Nimesulide PLA microspheres as a potential sustained release system for the treatment of inflammatory diseases

International Journal of Pharmaceutics

Volumn 295, Issue 1-2, 2005, Pages 201-211

  Freitas, M N ^a   Marchetti, J M ^a  

^a UNIVERSITY OF SÃO PAULO   (Brazil)

Author keywords

Emulsion solvent evaporation method; Microspheres; Nimesulide; Polylactic acid; Sustained release system

Indexed keywords

DRUG CARRIER; MICROSPHERE; NIMESULIDE; NONSTEROID ANTIINFLAMMATORY AGENT; POLYLACTIC ACID;

ARTICLE; BIODEGRADABILITY; DISSOLUTION; DRUG INDICATION; EMULSION; EVAPORATION; INFLAMMATORY DISEASE; PARTICLE SIZE; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; SCANNING ELECTRON MICROSCOPY; SUSTAINED DRUG RELEASE;

EID: 17644387694     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2005.03.003     Document Type: Article

References (44)

1. R.W. Baker, and H.S. Lonsdale Controlled Release of Biologically Active Agents 1974 Plenum Press New York pp. 15-71
2. T.D. Birnbaum, D.J. Kosmala, B.D. Henthorn, and L. Peppas-Brannon Controlled release of 17-β-estradiol from PLGA microparticles: the effect of organic phase solvent on encapsulation and release J. Control. Release 65 2000 375 387
3. F. Boury, T. Ivanova, I. Panaiotov, J.E. Proust, A. Bois, and J. Richou Dynamical properties of poly(d-l-lactide) monolayers at the air/water and at the dichloromethane/water interfaces J. Colloid Interface Sci. 169 1995 380 392
4. R.S. Branja, and T.K. Pal In vitro release kinetics of salbutamol sulphate microcapsules coated with both Eudragit RS 100 and Eudragit RL 100 Drug Dev. Ind. Pharm. 20 1994 375 386
5. R.K. Chang, J.C. Price, and C.W. Whithworth Control of drug release rates through the use of mixtures of policaprolactone and cellulose propionate polymers Pharm. Technol. 10 1986 24 33
6. P. Costa, D.C. Ferreira, and J.M. Souza Lobo Nitroglicerina em sistemas de liberação transdérmica-determinação da velocidade de libertação Rev. Port. Farm. 46 1996 4 8
7. P. Costa, and J.M. Souza Lobo Modeling and comparison of dissolution profiles Eur. J. Pharm. Sci. Rev. 13 2001 123 133
8. P. Couvreur, C. Dubernet, and P. Puisideux Eur. J. Pharm. Biopharm. 41 1995 2
9. P.B. Deasy, M.R. Brophy, B. Ecanow, and M. Joy J. Pharm. Pharmacol. 32 1980 15 20
10. S.J. Desai, P. Singh, A.P. Simonelli, and W.I. Higuchi Investigation of factors influencing release of solid drug dispersed in inert matrices. III. Quantitative studies involving the polyethylene plastic matrix J. Pharm. Sci. 55 1966 1230 1234
11. S.J. Desai, P. Singh, A.P. Simonelli, and W.I. Higuchi Investigation of factors influencing release of solid drug dispersed in inert matrices. IV. Some studies involving the polyvinyl choride matrix J. Pharm. Sci. 55 1966 1235 1239
12. S.J. Douglas, S.S. Davis, L. Davis, and L. Illum Nanoparticles in drug delivery, CRC Crit. Rev. Ther. Drug Carrier Syst. 3 1987 233 261
13. Ferraz, H.G., 1997. Avaliação biofarmacêutica in vitro in vivo (bioequivalência) de comprimidos de ampicilina 500 mg comercializados no Brazil (Tese de doutoramento, Faculdade de Ciências Farmacêuticas da Universidade de São Paulo). São Paulo, p. 135.
14. H. Fessi, F. Puisieux, J.PH. Devissaguet, N. Ammony, and S. Benita Nanocapsulde formation by interfacial deposition following solvent displcement Int. J. Pharm. 55 1989 R1-R4
15. G. Haixiong, H. Yong, Y. Shicheng, J. Xiqun, and Y. Changzheng Preparation, characterization, and drug release behaviours of drug-loaded e-caprolactone/l-lactide copolymer nanoparticles J. Appl. Polym. Sci. 75 2000 874 882
16. T. Higuchi Rate of release of medicaments from ointment bases containing drugs in suspension J. Pharm. Sci. 50 1961 874 875
17. T. Higuchi Mechanism of sustained-action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices J. Pharm. Sci. 51 1963 802 804
18. Huang, X., Brazel, C.S., 2001. On the importance and mechanisms of burst release in matrix-controlled drug delivery systems. J. Control. Release 73, 121-136.
19. I. Jalsenjak, and T. Kondo Effect of capsule size on permeability of gelatin-acacia microcapsules toward sodium chloride J. Pharm. Sci. 70 1981 456 457
20. H. Jeffery, S.S. Davis, and D.T. O'Hagan The preparation and characterization of poly(lactide-co-glycolide) microparticles. I. Oil-in-water emulsion solvent evaporation Int. J. Pharm. 77 1991 169 175
21. H.W. Jun, and J.W. Lai Preparation and in vitro dissolution tests of egg albumin microcapsules of nitrofurantion Int. J. Pharm. 16 1983 65 77
22. M.Z.I. Khan Dissolution testing for sustained or controlled release oral dosage forms and correlation with in vivo data: challenges and opportunities Int. J. Pharm. (Amsterdam) 140 1996 131 143
23. S.C. Lee, J.T. Oh, H.M. Jang, and L.S. Chung Quantitative analysis of polyvinyl alcohol on the surface of poly(d-,l-lactide-co-glycolide) microparticles prepared by solvent evaporation method: effect of particle size and PVA concentration J. Control. Release 59 1999 123 132
24. C. Michael, M.D. Ilia Fishbein, D.D. Haim, and G. Gershon Lipophilic drug nanospheres prepared by nanoprecipitaion: effect of formulation variables on size, drug recovery and release kinetics J. Control. Release 83 2002 389 400
25. M. Mortada Preparation of ethyl cellulose microcapsules using the complex emulsion method Pharmazie 37 1982 427 429
26. T. Niwa, H. Takeuchi, T. Hino, N. Kunou, and Y. Kawashima Preparation of biodegradable nanospheres of water-soluble and insoluble drugs with d-,l-lactide/glycolide copolymer by a novel emulsification solvent diffusion method, and drug release behavior J. Control. Release 25 1993 89 98
27. P.B. O'Donnel Mcginity, preparation of microspheres by the solvent evaporation technique Adv. Drug Del. Rev. 228 1997 25 42
28. D.T. O'Hagan, D. Rahman, J.P. McGee, H. Jeffery, M.C. Davies, P. Williams, S.S. Davis, and S.J. Challacombe Biodegradable microparticles as controlled release antigen delivery systems Imunology 73 1991 239 242
29. P. Ptacek, J. Macek, and J. Klima Rapid and simple high performance liquid chromatograpic determination of nimesulide in human plasma J. Chromatogr. B 758 2001 183 188
30. M.P. Redmon, A.J. Hickey, and P.P. DeLuca Predinizolone-21-acetate poly(glycolic acid) microspheres; influence of matrix characteristics on release J. Control. Release 9 1989 99 109
31. R.S. Schaffazick, S.S. Guterres, L.L. Freitas, and A.R. Pohjmann Characterization and physico-chemical stability of polymeric nanoparticulated systems for drug administration Químca Nova 26 No. 5 2003 726 737
32. B.J. Schwartz, A.P. Simonelli, and W.I. Higuchi Drug release from wax matrices. I. Analysis of data with first order kinetics and with the diffusion-controlled model J. Pharm. Sci. 57 1968 274 277
33. B.J. Schwartz, A.P. Simonelli, and W.I. Higuchi Drug release from wax matrices. II. Application of a mixture theory to the sulfanilamide-wax system J. Pharm. Sci. 57 1968 278 282
34. T. Seki, T. Kawaguchi, H. Endoh, K. Ishikawa, K. Juni, and M. Nakano Controle release of 3,5-diester prodrugs of 5-fluoro-2-deoxyuridine from poly-l-lactic acid microspheres J. Pharm. Sci. 79 1980 985 987
35. K.M. Shakessheff, C. Evora, I. Soriano, and R. Langer The absorption of poly(vinyl alcohol) to biodegradable micorparticles studied by X-ray photoelectron spectroscopy (XPS) J. Colloid Interface Sci. 185 1997 538 547
36. A.J. Shukla, and J.C. Price Effect of drug loading and molecular weight of cellulose acetate propionate on the release characteristics of theophyline microspheres Pharm. Res. 8 1991 1369 1400
37. C. Thies Formulation of degradable drug-loaded microparticles by in in-liquid drying processes M. Dunbrow Microcapsules and Nanoparticles in Medicine and Pharmacy 1992 CRC Press Boca Raton, FL 47 71
38. G. Thirumala, S. Snjezana, C.G. Martin, I. Lisbeth, and S.D. Stanley PLGA nanoparticles prepared by nanoprecipitation: drug loading and release studies of a water soluble drugs J. Control. Release 57 1999 171 185
39. S. Tognella Nimesulide: new clinical opportunities. Drugs 46 1993 275 276
40. T. Uchida, M. Kawata, and S.J. Goto In vivo evaluation of ethyl cellulose microcapsules containing ampicillin using rabbits, beagle dogs and humans Pharmacobio-Dyn. 9 1986 631 637
41. C.G. Varelas, D.G. Dixon, and C. Steiner Zero order release from biphasic polymer hydrogels J. Control. Release 34 1995 185 192
42. T. Verrecchia, P. Huve, D.V. Brazile, M. Veillard, G. Spenlehauer, and P. Couvreur Adsorption/desorption human serum albumin at the surface of poly(lactid acid) nanoparticles prepared by a solvent evaporation process J. Biomed. Mater. Res. 27 1993 1019 1028
43. R. Wada, S.H. Hyon, and Y. Ikada Lactic acid oligomer microspheres containing hydrophilic drugs J. Pharm. Sci. 79 1990 919 924
44. ®les and morphology of biodegradable microcapsules containing an oily core J. Control. Release 76 2001 313 326