Optical recording reveals novel properties of GSK1016790A-induced vanilloid transient receptor potential channel TRPV4 activity in primary human endothelial cells

Molecular Pharmacology

Volumn 82, Issue 3, 2012, Pages 464-472

  Sullivan, Michelle N ^a   Francis, Michael ^b   Pitts, Natalie L ^a   Taylor, Mark S ^b   Earley, Scott ^a  

^a Department of Environmental and Radiological Health Sciences   (United States)

^b UNIVERSITY OF SOUTH ALABAMA COLLEGE OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CALCIUM CHANNEL; CALCIUM ION; GSK 1016790 A; N [1 [[4 [2 [((2,4 DICHLOROPHENYL)SULFONYL)AMINO] 3 HYDROXYPROPANOYL] 1 PIPERAZINYL]CARBONYL] 3 METHYLBUTYL] 1 BENZOTHIOPHENE 2 CARBOXAMIDE; UNCLASSIFIED DRUG; VANILLOID RECEPTOR 4; VANILLOID RECEPTOR AFFECTING AGENT;

ARTICLE; CELL ACTIVITY; CELL MEMBRANE; COMPUTER PROGRAM; CONTROLLED STUDY; ENDOTHELIUM CELL; FLUORESCENCE MICROSCOPY; HUMAN; HUMAN CELL; NEWBORN; OPTICS; PRIORITY JOURNAL;

CALCIUM; CELL MEMBRANE; CELLS, CULTURED; ENDOTHELIAL CELLS; ENDOTHELIUM, VASCULAR; HUMANS; LEUCINE; MICROSCOPY, FLUORESCENCE; SULFONAMIDES; TRPV CATION CHANNELS;

EID: 84865212470     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.112.078584     Document Type: Article

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