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Volumn 60, Issue 32, 2012, Pages 7949-7956

Effects of estrogen and estrus cycle on pharmacokinetics, absorption, and disposition of genistein in female sprague-dawley rats

Author keywords

estrogen; estrus cycle; genistein; oral bioavailability; pharmacokinetics

Indexed keywords

AGLYCONES; ANTICANCER ACTIVITIES; BASAL LEVELS; ESTROGEN; ESTRUS CYCLE; FEMALE RAT; GENISTEIN; GLUCURONIDATION; HEPATIC ENZYMES; ISOFLAVONES; MALE RATS; ORAL BIOAVAILABILITY; PERFUSION STUDIES; SPRAGUE-DAWLEY RATS;

EID: 84865146287     PISSN: 00218561     EISSN: 15205118     Source Type: Journal    
DOI: 10.1021/jf204755g     Document Type: Article
Times cited : (11)

References (26)
  • 1
    • 0036201358 scopus 로고    scopus 로고
    • Absorption and metabolism of flavonoids in the Caco-2 cell culture model and a perfused rat intestinal model
    • DOI 10.1124/dmd.30.4.370
    • Liu, Y.; Hu, M. Absorption and metabolism of flavonoids in the caco-2 cell culture model and a perused rat intestinal model Drug Metab. Dispos. 2002, 30 (4) 370-377 (Pubitemid 34263820)
    • (2002) Drug Metabolism and Disposition , vol.30 , Issue.4 , pp. 370-377
    • Liu, Y.1    Hu, M.2
  • 3
    • 18144386028 scopus 로고    scopus 로고
    • The role of isoflavones in cancer chemoprevention
    • Sarkar, F. H.; Li, Y. The role of isoflavones in cancer chemoprevention Front. Biosci. 2004, 9, 2714-2724
    • (2004) Front. Biosci. , vol.9 , pp. 2714-2724
    • Sarkar, F.H.1    Li, Y.2
  • 5
    • 0035073833 scopus 로고    scopus 로고
    • Genistein, daidzein and glycitein inhibit growth and DNA synthesis of aortic smooth muscle cells from stroke-prone spontaneously hypertensive rats
    • Pan, W.; Ikeda, K.; Takebe, M.; Yamori, Y. Genistein, daidzein and glycitein inhibit growth and DNA synthesis of aortic smooth muscle cells from stroke-prone spontaneously hypertensive rats J. Nutr. 2001, 131 (4) 1154-1158 (Pubitemid 32275092)
    • (2001) Journal of Nutrition , vol.131 , Issue.4 , pp. 1154-1158
    • Pan, W.1    Ikeda, K.2    Takebe, M.3    Yamori, Y.4
  • 6
    • 0036825350 scopus 로고    scopus 로고
    • 14C] genistein in the rat; plasma pharmacokinetics of parent compound, genistein glucuronide and total radioactivity
    • Coldham, N. G.; Zhang, A. Q.; Key, P.; Sauer, M. J. Absolute bioavailability of [14C] genistein in the rat; plasma pharmacokinetics of parent compound, genistein glucuronide and total radioactivity Eur. J. Drug Metab. Pharmacokinet. 2002, 27 (4) 249-258 (Pubitemid 36205472)
    • (2002) European Journal of Drug Metabolism and Pharmacokinetics , vol.27 , Issue.4 , pp. 249-258
    • Coldham, N.G.1    Zhang, A.-Q.2    Key, P.3    Sauer, M.J.4
  • 7
    • 77953497158 scopus 로고    scopus 로고
    • Lesson learned from nature for the development of novel anti-cancer agents: Implication of isoflavone, curcumin, and their synthetic analogs
    • Sarkar, F. H.; Li, Y.; Wang, Z.; Padhye, S. Lesson learned from nature for the development of novel anti-cancer agents: implication of isoflavone, curcumin, and their synthetic analogs Curr. Pharm. Des. 2010, 16 (16) 1801-1812
    • (2010) Curr. Pharm. Des. , vol.16 , Issue.16 , pp. 1801-1812
    • Sarkar, F.H.1    Li, Y.2    Wang, Z.3    Padhye, S.4
  • 9
    • 0019349644 scopus 로고
    • The role of a high-fat diet in enhancing the development of mammary tumors in ovariectomized rats
    • DOI 10.1002/1097-0142(19810101)47:1<66::AID-CNCR2820470113>3.0. CO;2-M
    • Cohen, L. A.; Chan, P. C.; Wynder, E. L. The role of a high-fat diet in enhancing the development of mammary tumors in ovariectomized rats Cancer 1981, 47 (1) 66-71 (Pubitemid 11167362)
    • (1981) Cancer , vol.47 , Issue.1 , pp. 66-71
    • Cohen, L.A.1    Chan, P.C.2    Wynder, E.L.3
  • 10
    • 0017372823 scopus 로고
    • Effects of tamoxifen in relation to breast cancer
    • Jordan, V. C. Effects of tamoxifen in relation to breast cancer Br. Med. J. 1977, 1 (6075) 1534-1535 (Pubitemid 8115362)
    • (1977) British Medical Journal , vol.1 , Issue.6075 , pp. 1534-1535
    • Jordan, V.C.1
  • 11
    • 69349094410 scopus 로고    scopus 로고
    • Tamoxifen produces conditioned taste avoidance in male rats: An analysis of microstructural licking patterns and taste reactivity
    • Fudge, M. A.; Kavaliers, M.; Baird, J. P.; Ossenkopp, K. P. Tamoxifen produces conditioned taste avoidance in male rats: an analysis of microstructural licking patterns and taste reactivity Horm. Behav. 2009, 56 (3) 322-331
    • (2009) Horm. Behav. , vol.56 , Issue.3 , pp. 322-331
    • Fudge, M.A.1    Kavaliers, M.2    Baird, J.P.3    Ossenkopp, K.P.4
  • 12
    • 69749125067 scopus 로고    scopus 로고
    • Antitumor and antiangiogenic activity of soy phytoestrogen on 7,12-dimethylbenz[alpha]anthracene-induced mammary tumors following ovariectomy in Sprague-Dawley rats
    • Kang, X.; Jin, S.; Zhang, Q. Antitumor and antiangiogenic activity of soy phytoestrogen on 7,12-dimethylbenz[alpha]anthracene-induced mammary tumors following ovariectomy in Sprague-Dawley rats J. Food Sci. 2009, 74 (7) H237-H242
    • (2009) J. Food Sci. , vol.74 , Issue.7
    • Kang, X.1    Jin, S.2    Zhang, Q.3
  • 13
    • 59849085757 scopus 로고    scopus 로고
    • Tamoxifen and raloxifene produce conditioned taste avoidance in female rats: A microstructural analysis of licking patterns
    • Fudge, M. A.; Kavaliers, M.; Baird, J. P.; Ossenkopp, K. P. Tamoxifen and raloxifene produce conditioned taste avoidance in female rats: a microstructural analysis of licking patterns Life Sci. 2009, 84 (9-10) 282-289
    • (2009) Life Sci. , vol.84 , Issue.9-10 , pp. 282-289
    • Fudge, M.A.1    Kavaliers, M.2    Baird, J.P.3    Ossenkopp, K.P.4
  • 14
    • 0017735687 scopus 로고
    • Ovarian and adrenal steroids during pregnancy and the oestrous cycle in the rat
    • Ogle, T. F.; Kitay, J. I. Ovarian and adrenal steroids during pregnancy and the oestrous cycle in the rat J. Endocrinol. 1977, 74 (1) 89-98 (Pubitemid 8139416)
    • (1977) Journal of Endocrinology , vol.74 , Issue.1 , pp. 89-98
    • Ogle, T.F.1    Kitay, J.I.2
  • 15
    • 0003255738 scopus 로고    scopus 로고
    • Determination of the estrous cycle phases of rats: Some helpful considerations
    • Marcondes, F. K.; Bianchi, F. J.; Tanno, A. P. Determination of the estrous cycle phases of rats: some helpful considerations Braz. J. Biol. 2002, 62 (4A) 609-614
    • (2002) Braz. J. Biol. , vol.62 , Issue.4 A , pp. 609-614
    • Marcondes, F.K.1    Bianchi, F.J.2    Tanno, A.P.3
  • 16
    • 0035851899 scopus 로고    scopus 로고
    • Estrous cycle influences the response of female rats in the elevated plus-maze test
    • DOI 10.1016/S0031-9384(01)00593-5, PII S0031938401005935
    • Marcondes, F. K.; Miguel, K. J.; Melo, L. L.; Spadari-Bratfisch, R. C. Estrous cycle influences the response of female rats in the elevated plus-maze test Physiol. Behav. 2001, 74 (4-5) 435-440 (Pubitemid 34076588)
    • (2001) Physiology and Behavior , vol.74 , Issue.4-5 , pp. 435-440
    • Marcondes, F.K.1    Miguel, K.J.2    Melo, L.L.3    Spadari-Bratfisch, R.C.4
  • 17
    • 77952323519 scopus 로고    scopus 로고
    • Simultaneous determination of genistein and its four phase II metabolites in blood by a sensitive and robust UPLC-MS/MS method: Application to an oral bioavailability study of genistein in mice
    • Yang, Z.; Zhu, W.; Gao, S.; Xu, H.; Wu, B.; Kulkarni, K.; Singh, R.; Tang, L.; Hu, M. Simultaneous determination of genistein and its four phase II metabolites in blood by a sensitive and robust UPLC-MS/MS method: application to an oral bioavailability study of genistein in mice J. Pharm. Biomed. Anal. 2010, 53 (1) 81-89
    • (2010) J. Pharm. Biomed. Anal. , vol.53 , Issue.1 , pp. 81-89
    • Yang, Z.1    Zhu, W.2    Gao, S.3    Xu, H.4    Wu, B.5    Kulkarni, K.6    Singh, R.7    Tang, L.8    Hu, M.9
  • 18
    • 0031849072 scopus 로고    scopus 로고
    • Determination of absorption characteristics of AG337, a novel thymidylate synthase inhibitor, using a perfused rat intestinal model
    • DOI 10.1021/js970251e
    • Hu, M.; Roland, K.; Ge, L.; Chen, J.; Li, Y.; Tyle, P.; Roy, S. Determination of absorption characteristics of AG337, a novel thymidylate synthase inhibitor, using a perfused rat intestinal model J. Pharm. Sci. 1998, 87 (7) 886-890 (Pubitemid 28319421)
    • (1998) Journal of Pharmaceutical Sciences , vol.87 , Issue.7 , pp. 886-890
    • Hu, M.1    Roland, K.2    Ge, L.3    Chen, J.4    Li, Y.5    Tyle, P.6    Roy, S.7
  • 19
    • 0023924860 scopus 로고
    • Membrane permeability parameters for some amino acids and beta-lactam antibiotics: Application of the boundary layer approach
    • Hu, M.; Sinko, P. J.; deMeere, A. L.; Johnson, D. A.; Amidon, G. L. Membrane permeability parameters for some amino acids and beta-lactam antibiotics: application of the boundary layer approach J. Theor. Biol. 1988, 131 (1) 107-114
    • (1988) J. Theor. Biol. , vol.131 , Issue.1 , pp. 107-114
    • Hu, M.1    Sinko, P.J.2    Demeere, A.L.3    Johnson, D.A.4    Amidon, G.L.5
  • 20
    • 0037371414 scopus 로고    scopus 로고
    • Metabolism of flavonoids via enteric recycling: Role of intestinal disposition
    • DOI 10.1124/jpet.102.046409
    • Chen, J.; Lin, H.; Hu, M. Metabolism of flavonoids via enteric recycling: role of intestinal disposition J. Pharmacol. Exp. Ther. 2003, 304 (3) 1228-1235 (Pubitemid 36254436)
    • (2003) Journal of Pharmacology and Experimental Therapeutics , vol.304 , Issue.3 , pp. 1228-1235
    • Chen, J.1    Lin, H.2    Hu, M.3
  • 21
    • 33751113603 scopus 로고    scopus 로고
    • Disposition of flavonoids via enteric recycling: Structural effects and lack of correlations between in vitro and in situ metabolic properties
    • DOI 10.1124/dmd.106.009910
    • Wang, S. W.; Chen, J.; Jia, X.; Tam, V. H.; Hu, M. Disposition of flavonoids via enteric recycling: structural effects and lack of correlations between in vitro and in situ metabolic properties Drug Metab. Dispos. 2006, 34 (11) 1837-1848 (Pubitemid 44771711)
    • (2006) Drug Metabolism and Disposition , vol.34 , Issue.11 , pp. 1837-1848
    • Wang, S.W.J.1    Chen, J.2    Jia, X.3    Tam, V.H.4    Hu, M.5
  • 22
    • 66749132077 scopus 로고    scopus 로고
    • Disposition of Flavonoids via Enteric Recycling: UGT1As Deficiency in Gunn Rats Is Compensated by Increases in UGT2Bs Activities
    • Wang, S.; Kulkarni, K. H.; Tang, L; Wang, J; Daidoji, T; Yokota, H.; Hu, M. Disposition of Flavonoids via Enteric Recycling: UGT1As Deficiency in Gunn Rats Is Compensated by Increases in UGT2Bs Activities J. Pharmacol. Exp. Ther. 2009, 329, 1023-1031
    • (2009) J. Pharmacol. Exp. Ther. , vol.329 , pp. 1023-1031
    • Wang, S.1    Kulkarni, K.H.2    Tang, L.3    Wang, J.4    Daidoji, T.5    Yokota, H.6    Hu, M.7
  • 23
    • 66749132077 scopus 로고    scopus 로고
    • Disposition of flavonoids via enteric recycling: UDP- glucuronosyltransferase (UGT) 1As deficiency in Gunn rats is compensated by increases in UGT2Bs activities
    • Wang, S. W.; Kulkarni, K. H.; Tang, L.; Wang, J. R.; Yin, T.; Daidoji, T.; Yokota, H.; Hu, M. Disposition of flavonoids via enteric recycling: UDP-glucuronosyltransferase (UGT) 1As deficiency in Gunn rats is compensated by increases in UGT2Bs activities J. Pharmacol. Exp. Ther. 2009, 329 (3) 1023-1031
    • (2009) J. Pharmacol. Exp. Ther. , vol.329 , Issue.3 , pp. 1023-1031
    • Wang, S.W.1    Kulkarni, K.H.2    Tang, L.3    Wang, J.R.4    Yin, T.5    Daidoji, T.6    Yokota, H.7    Hu, M.8
  • 25
    • 77957555079 scopus 로고    scopus 로고
    • Canola oil inhibits breast cancer cell growth in cultures and in vivo and acts synergistically with chemotherapeutic drugs
    • Cho, K.; Mabasa, L.; Fowler, A. W.; Walsh, D. M.; Park, C. S. Canola oil inhibits breast cancer cell growth in cultures and in vivo and acts synergistically with chemotherapeutic drugs Lipids 2010, 45 (9) 777-784
    • (2010) Lipids , vol.45 , Issue.9 , pp. 777-784
    • Cho, K.1    Mabasa, L.2    Fowler, A.W.3    Walsh, D.M.4    Park, C.S.5
  • 26
    • 59849085757 scopus 로고    scopus 로고
    • Tamoxifen and raloxifene produce conditioned taste avoidance in female rats: A microstructural analysis of licking patterns
    • Fudge, M. A.; Kavaliers, M.; Baird, J. P.; Ossenkopp, K. P. Tamoxifen and raloxifene produce conditioned taste avoidance in female rats: a microstructural analysis of licking patterns Life Sci. 2009, 84 (9-10) 282-289
    • (2009) Life Sci. , vol.84 , Issue.9-10 , pp. 282-289
    • Fudge, M.A.1    Kavaliers, M.2    Baird, J.P.3    Ossenkopp, K.P.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.