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Volumn 14, Issue 3, 2012, Pages 580-585

One-pot synthesis of useful heterocycles in medicinal chemistry using a cascade strategy

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EID: 84863270175     PISSN: 14639262     EISSN: 14639270     Source Type: Journal    
DOI: 10.1039/c2gc16457d     Document Type: Article
Times cited : (34)

References (73)
  • 7
    • 53849120603 scopus 로고    scopus 로고
    • For a review of recent applications of cascade reactions to natural product synthesis, see
    • I. Nicolas L. Rodolfo Chem.–Eur. J. 2008 14 8444-8454; For a review of recent applications of cascade reactions to natural product synthesis, see.
    • (2008) Chem.–Eur. J. , vol.14 , pp. 8444-8454
    • Nicolas, I.1    Rodolfo, L.2
  • 12
    • 85034327954 scopus 로고    scopus 로고
    • Northwestern University US20080051410
    • Watterson, D. M., Van Eldik, L. J. Northwestern University US20080051410, 2008.
    • (2008)
    • Watterson, D.M.1    Van Eldik, L.J.2
  • 21
    • 85034374327 scopus 로고    scopus 로고
    • N30 Pharmaceuticals, LLC. WO2011038204
    • Sun, X., Qiu, J. N30 Pharmaceuticals, LLC. WO2011038204, 2011.
    • (2011)
    • Sun, X.1    Qiu, J.2
  • 22
    • 33845374099 scopus 로고
    • For reviews on benzofurans see
    • For reviews on benzofurans see: B. H. Lipshutz Chem. Rev. 1986 86 795-819.
    • (1986) Chem. Rev. , vol.86 , pp. 795-819
    • Lipshutz, B.H.1
  • 23
    • 84943380362 scopus 로고
    • Furans and Their Benzo Derivatives: (iii) Synthesis and Applications
    • A. R. Katritzky, Ed., Pergamon, New York
    • D. M. X. Donelly, M. J. Meegan Furans and Their Benzo Derivatives: (iii) Synthesis and Applications, In Comprehensive Heterocyclic Chemistry, A. R. Katritzky, Ed., Pergamon, New York, 1984, Vol. 4, pp 657–712.
    • (1984) Comprehensive Heterocyclic Chemistry , vol.4 , pp. 657-712
    • Donelly, D.M.X.1    Meegan, M.J.2
  • 25
    • 84943376011 scopus 로고
    • Synthesis of Five-membered Rings with One Heteroatom
    • A. R. KatritzkyPergamon, New York, For recent discovery of novel benzofurans as lignan derivatives, see
    • C. W. Bird, G. W. H. Cheeseman Synthesis of Five-membered Rings with One Heteroatom. In Comprehensive Heterocyclic Chemistry, A. R. Katritzky, Ed., Pergamon, New York, 1984, Vol. 4, pp 89153. For recent discovery of novel benzofurans as lignan derivatives, see.
    • (1984) Comprehensive Heterocyclic Chemistry , vol.4 , pp. 89153
    • Bird, C.W.1    Cheeseman, G.W.H.2
  • 27
    • 84943407995 scopus 로고
    • For reviews on indazoles see, A. R. Katrizky, C. W. Rees, Eds., Pergamon Press, New York
    • For reviews on indazoles see: J. Elguero In Comprehensi e Heterocyclic Chemistry, A. R. Katrizky, C. W. Rees, Eds., Pergamon Press, New York, 1984, Vol. 5, p 167.
    • (1984) Comprehensi E Heterocyclic Chemistry , vol.5 , pp. 167
    • Elguero, J.1
  • 34
    • 0003678023 scopus 로고
    • ACS Monograph 186, American Chemical Society, Washington, DC
    • M. Hudlicky, Oxidations in Organic Chemistry, ACS Monograph 186, American Chemical Society, Washington, DC, 1990.
    • (1990) Oxidations in Organic Chemistry
    • Hudlicky, M.1
  • 38
  • 52
    • 84979132760 scopus 로고
    • For selected examples, see
    • For selected examples, see: L. Claisen O. Lowman Ber. 1887 20 651-654.
    • (1887) Ber. , vol.20 , pp. 651-654
    • Claisen, L.1    Lowman, O.2
  • 61
    • 85034321300 scopus 로고    scopus 로고
    • FR 2880023, For examples of Claisen condensation using malonic acid mono esters, see
    • Barth, F., Congy, C., Ducoux, J. P., Rinaldi, C. M. FR 2880023, 2006. For examples of Claisen condensation using malonic acid mono esters, see.
    • (2006)
    • Barth, F.1    Congy, C.2    Ducoux, J.P.3    Rinaldi, C.M.4
  • 73
    • 85034341382 scopus 로고    scopus 로고
    • The scale-up was performed using 3 grams of 2-(2-bromophenyl)acetic acid. The desired product, methyl stemofuran, was obtained in 66% yield. See supporting information for experimental details
    • The scale-up was performed using 3 grams of 2-(2-bromophenyl)acetic acid. The desired product, methyl stemofuran, was obtained in 66% yield. See supporting information for experimental details.


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