Development of biochemical assays for the identification of eIF4E-specific inhibitors

Journal of Biomolecular Screening

Volumn 17, Issue 5, 2012, Pages 581-592

  Visco, Carlo ^a   Perrera, Claudia ^a   Thieffine, Sandrine ^a   Sirtori, Federico Riccardi ^b   D'Alessio, Roberto ^b   Magnaghi, Paola ^c  

^a Biotechnology Department   (Italy)

^b Chemistry Department   (Italy)

^c NERVIANO MEDICAL SCIENCES   (Italy)

Author keywords

CBP80 CBP20; eIF4E; fluorescence polarization; screening; surface plasmon resonance

Indexed keywords

GUANOSINE DIPHOSPHATE; GUANOSINE TRIPHOSPHATE DERIVATIVE; INITIATION FACTOR 4E; MESSENGER RNA; OLIGONUCLEOTIDE;

ARTICLE; ASSAY; CANCER THERAPY; CELL CYCLE; DRUG TARGETING; FLUORESCENCE POLARIZATION; HUMAN; MOLECULARLY TARGETED THERAPY; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN PURIFICATION; RNA TRANSLATION; SCREENING; SURFACE PLASMON RESONANCE; TUMOR CELL LINE; TUMOR XENOGRAFT;

DRUG DISCOVERY; EUKARYOTIC INITIATION FACTOR-4E; FLUORESCENCE POLARIZATION; HUMANS; KINETICS; NUCLEAR CAP-BINDING PROTEIN COMPLEX; PROTEIN BINDING; REPRODUCIBILITY OF RESULTS; RNA CAPS; SURFACE PLASMON RESONANCE;

EUKARYOTA;

EID: 84861832788     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057112438554     Document Type: Article

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