Radiolabeling of RGD peptide and preliminary biological evaluation in mice bearing U87MG tumors

Bioorganic and Medicinal Chemistry

Volumn 20, Issue 12, 2012, Pages 3850-3855

  Li, Jianbo ^a,b   Shi, Lingli ^a,b   Jia, Lina ^a,b   Jiang, Dawei ^a,b   Zhou, Wei ^a   Hu, Weiqing ^a   Qi, Yujin ^a   Zhang, Lan ^a  

^a SHANGHAI INSTITUTE OF APPLIED PHYSICS   (China)

^b UNIVERSITY OF CHINESE ACADEMY OF SCIENCES   (China)

Author keywords

Click reaction; Fluorion 18; Micro PET imaging; Radiolabeling; RGD peptide

Indexed keywords

2 AZIDOETHYL 4 TOLUENESULFONIC ACID; 2 FLUOROETHYLAZIDE F 18; ALKYNE; ARGINYLGLYCYLASPARTYLPHENYLALANYLLYSINE; COPPER; PENTAPEPTIDE; PHOSPHATE BUFFERED SALINE; RADIOPHARMACEUTICAL AGENT; TOLUENESULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; VITRONECTIN RECEPTOR;

ANIMAL EXPERIMENT; BINDING AFFINITY; CATALYST; CHEMICAL REACTION; CLICK CHEMISTRY; CONCENTRATION (PARAMETERS); CONFERENCE PAPER; CYCLOADDITION; DRUG ACCUMULATION; DRUG CLEARANCE; DRUG STRUCTURE; DRUG TUMOR LEVEL; FLUORINATION; GLIOBLASTOMA; ISOTOPE LABELING; MALE; MICRO-POSITRON EMISSION TOMOGRAPHY; MOUSE; NEWBORN CALF SERUM; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RADIOCHEMISTRY; RADIOFLUORINATION; RADIOISOTOPE DECAY; REACTION TIME; RECEPTOR BINDING; SERUM; SYNTHESIS; TEMPERATURE;

ANIMALS; CELL LINE, TUMOR; FLUORINE RADIOISOTOPES; HUMANS; MICE; MICE, INBRED STRAINS; NEOPLASMS, EXPERIMENTAL; OLIGOPEPTIDES; TISSUE DISTRIBUTION;

MUS;

EID: 84861574314     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2012.04.037     Document Type: Conference Paper

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