Synthesis and biological evaluation of a series of novel salicylanilides as inhibitors of EGFR protein tyrosine kinases

Chinese Chemical Letters

Volumn 23, Issue 5, 2012, Pages 529-532

  Ding, Ning ^a   Zhang, Wei ^a   Xiao, Hua Ling ^b   Wang, Peng ^b   Li, Ying Xia ^a  

^a FUDAN UNIVERSITY   (China)

^b OCEAN UNIVERSITY OF CHINA   (China)

Author keywords

EGFR; HER2; Salicylanilides; Tyrosine kinase inhibitor

Indexed keywords

EID: 84860369237     PISSN: 10018417     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cclet.2012.03.016     Document Type: Article

References (34)

1. C.T. Supuran, and A. Scozzafava Expert Opin. Ther. Patents 14 2004 35
2. Y. Yarden, and M.X. Sliwkowski Nat. Rev. Mol. Biol. 2 2001 127
3. J.B. Johnston, S. Navaratnam, and M.W. Pitz Curr. Med. Chem. 13 2006 3483
4. P.A. Bunn Jr., B. Helfrich, and A.F. Soriano Clin. Cancer Res. 7 2001 3239
5. R.S. Herbst, and A.B. Sandler Clin. Lung Cancer 6 Suppl. 1 2004 S7
6. E. Raymond, S. Faivre, and J.P. Armand Drugs 60 2000 15
7. A. Levitzki, and A. Gazit Science 267 1995 1782
8. E.K. Rowinsky Annu. Rev. Med. 55 2004 433
9. J. Dumas Curr. Opin. Drug Discov. Devel. 4 2001 378
10. H.C. Maguire Jr., and M.I. Greene Semin. Oncol. 16 1989 148
11. Y. Yarden, and M.X. Sliwkowski Nat. Rev. Mol. Cell Biol. 2 2001 127
12. H.K. Koeppen, B.D. Wright, and A.D. Burt Histopathology 38 2001 96
13. V. Aparna, G. Rambabu, and S.K. Panigrahi J. Chem. Inf. Model. 45 2005 725
14. G. Speake, B. Holloway, and G. Costello Curr. Opin. Pharmacol. 5 2005 343
15. K.G. Petrov, Y. Zhang, and M. Carter Bioorg. Med. Chem. Lett. 16 2006 4686
16. A.J. Barker, K.H. Gibson, and W. Grudy Bioorg. Med. Chem. Lett. 11 2001 1191
17. A.M. Bulgaru, S. Mani, and S. Goel Expert Rev. Anticancer Ther. 3 2003 269
18. D.W. Rusnak, K. Lackey, and K. Affleck Mol. Cancer Ther. 1 2001 85
19. L. Kopper Pathol. Oncol. Res. 14 2008 1
20. S. Dhillon, and A.J. Wagstaff Drugs 67 2007 2101
21. J. Stamos, M.X. Sliwkowski, and C. Eigenbrot J. Biol. Chem. 48 2002 46265
22. J.J. Liao J. Med. Chem. 50 2007 409
23. S. Garofalo, R. Rosa, and R. Bianco Expert Opin. Ther. Patents 18 2008 889
24. P. Traxler Expert Opin. Ther. Targets 7 2003 215
25. C.N. Hodge, and J. Pierce Bioorg. Med. Chem. Lett. 3 1993 1605
26. P. Traxler, J. Green, and H. Mett J. Med. Chem. 42 1999 1018
27. H. Suezawa, M. Hirota, and T. Yuzuri Bull. Chem. Soc. Jpn. 73 2000 2335
28. C. Liechti, U. Séquin, and G. Bold Eur. J. Med. Chem. 39 2004 11
29. L. Guo, Q. Wang, and Q.Q. Jiang J. Org. Chem. 72 2007 9947
30. W. Deng, Z. Guo, and Y. Guo Bioorg. Med. Chem. Lett. 16 2006 469
31. P. Knesl, D. Röseling, and U. Jordis Molecules 11 2006 286
32. T. Cohen, A.G. Dietz Jr., and J.R. Miser J. Org. Chem. 42 1977 2053
33. R.J. Edsall Jr., H.A. Harris, and E.S. Manasa Bioorg. Med. Chem. 11 2003 3457
34. P.S. Brignola, K. Lackey, and S.H. Kadwell J. Biol. Chem. 277 2002 1576