Bio-relevant media to assess drug permeability: Sodium taurocholate and lecithin combination or crude bile?

International Journal of Pharmaceutics

Volumn 429, Issue 1-2, 2012, Pages 22-30

  Berginc, Katja ^a   Trontelj, Jurij ^a   Kristl, Albin ^a  

^a UNIVERSITY OF LJUBLJANA   (Slovenia)

Author keywords

Bile; Bio relevant conditions; Drug binding; Lecithin; Permeability; Taurocholate

Indexed keywords

ACICLOVIR; AMITRIPTYLINE; ATENOLOL; BENDROFLUMETHIAZIDE; CHLORPHENIRAMINE; CIMETIDINE; CLOMIPRAMINE; FELODIPINE; FEXOFENADINE; FLUINDOSTATIN; FUROSEMIDE; GUANABENZ; HYDROCHLOROTHIAZIDE; LISINOPRIL; LOPERAMIDE; METOPROLOL; NADOLOL; NITROFURANTOIN; NORFLOXACIN; PHENAZONE; PHOSPHATIDYLCHOLINE; PINDOLOL; PRAVASTATIN; RANITIDINE; SALAZOSULFAPYRIDINE; SERTRALINE; SUMATRIPTAN; TAUROCHOLIC ACID; TERBUTALINE; UNINDEXED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BILE; CELL STRAIN CACO 2; CELL VIABILITY; CONTROLLED STUDY; CORRELATION ANALYSIS; DIET RESTRICTION; DRUG ABSORPTION; DRUG METABOLISM; DRUG PENETRATION; HUMAN; HUMAN CELL; IN VITRO STUDY; IN VIVO STUDY; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; BILE; BIOLOGICAL TRANSPORT; CACO-2 CELLS; HUMANS; INTESTINAL ABSORPTION; INTESTINE, SMALL; LECITHINS; MICELLES; MODELS, BIOLOGICAL; PERMEABILITY; PHARMACEUTICAL PREPARATIONS; RATS; SURFACE-ACTIVE AGENTS; SWINE; TAUROCHOLIC ACID;

EID: 84859625940     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.03.015     Document Type: Article

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