메뉴 건너뛰기




Volumn 56, Issue 3, 2012, Pages 1564-1570

Novel potent metallocenes against liver stage malaria

Author keywords

[No Author keywords available]

Indexed keywords

ANTIMALARIAL AGENT; FERROCENE DERIVATIVE; PRIMACENE; PRIMAQUINE; UNCLASSIFIED DRUG;

EID: 84857165822     PISSN: 00664804     EISSN: 10986596     Source Type: Journal    
DOI: 10.1128/AAC.05345-11     Document Type: Article
Times cited : (37)

References (34)
  • 3
    • 67651004913 scopus 로고    scopus 로고
    • Resistance to therapies for infection by Plasmodium vivax
    • Baird JK. 2009. Resistance to therapies for infection by Plasmodium vivax. Clin. Microbiol. Rev. 22:508-534.
    • (2009) Clin. Microbiol. Rev. , vol.22 , pp. 508-534
    • Baird, J.K.1
  • 4
    • 0242487691 scopus 로고    scopus 로고
    • Synthesis and antimalarial activity in vitro of new heterobimetallic complexes: Rh and Au derivatives of chloroquine and a series of ferrocenyl-4-amino-7-chloroquinolines
    • Blackie MAL, et al. 2003. Synthesis and antimalarial activity in vitro of new heterobimetallic complexes: Rh and Au derivatives of chloroquine and a series of ferrocenyl-4-amino-7-chloroquinolines. J. Organomet. Chem. 688:144-152.
    • (2003) J. Organomet. Chem. , vol.688 , pp. 144-152
    • Blackie, M.A.L.1
  • 5
    • 79959959354 scopus 로고    scopus 로고
    • The state of the art in antimalarial drug discovery and development
    • Burrows JN, Chibale K, Wells TNC. 2011. The state of the art in antimalarial drug discovery and development. Curr. Top. Med. Chem. 11:1226-1254.
    • (2011) Curr. Top. Med. Chem. , vol.11 , pp. 1226-1254
    • Burrows, J.N.1    Chibale, K.2    Wells, T.N.C.3
  • 6
    • 0000315307 scopus 로고
    • Steric effects. I. Esterification and acid-catalyzed hydrolysis of esters
    • Charton M. 1975. Steric effects. I. Esterification and acid-catalyzed hydrolysis of esters. J. Am. Chem. Soc. 97:1552-1556.
    • (1975) J. Am. Chem. Soc. , vol.97 , pp. 1552-1556
    • Charton, M.1
  • 7
    • 33646352709 scopus 로고    scopus 로고
    • Assessment of Plasmodium falciparum resistance to ferroquine (SSR97193) in field isolates and in W2 strain under pressure
    • Daher W, et al. 2006. Assessment of Plasmodium falciparum resistance to ferroquine (SSR97193) in field isolates and in W2 strain under pressure. Malar. J. 5:11.
    • (2006) Malar. J. , vol.5 , pp. 11
    • Daher, W.1
  • 8
    • 79953322662 scopus 로고    scopus 로고
    • Towards an in vitro model of Plasmodium hypnozoites suitable for drug discovery
    • Dembele L, et al. 2011. Towards an in vitro model of Plasmodium hypnozoites suitable for drug discovery. PLoS One 6:e18162.
    • (2011) PLoS One , vol.6
    • Dembele, L.1
  • 9
    • 73249120807 scopus 로고    scopus 로고
    • Enhancement of the antimalarial activity of ciprofloxacin using a double prodrug/bioorganometallic approach
    • Dubar F, et al. 2009. Enhancement of the antimalarial activity of ciprofloxacin using a double prodrug/bioorganometallic approach. J. Med. Chem. 52:7954-7957.
    • (2009) J. Med. Chem. , vol.52 , pp. 7954-7957
    • Dubar, F.1
  • 10
    • 58149387664 scopus 로고    scopus 로고
    • Ferroquine, an ingenious antimalarial drug - Thoughts on the mechanism of action
    • Dubar F, Khalife J, Brocard J, Dive D, Biot C. 2008. Ferroquine, an ingenious antimalarial drug - thoughts on the mechanism of action. Molecules 13:2900-2907.
    • (2008) Molecules , vol.13 , pp. 2900-2907
    • Dubar, F.1    Khalife, J.2    Brocard, J.3    Dive, D.4    Biot, C.5
  • 12
    • 57649149608 scopus 로고    scopus 로고
    • Plasmodium vivax: Who cares?
    • Galinski MR, Barnwell JW. 2008. Plasmodium vivax: who cares? Malar. J. 7(Suppl 1):S9.
    • (2008) Malar. J. , vol.7 , Issue.SUPPL. 1
    • Galinski, M.R.1    Barnwell, J.W.2
  • 13
    • 39749181550 scopus 로고    scopus 로고
    • Generation of a set of simple, interpretable ADMET rules of thumb
    • DOI 10.1021/jm701122q
    • Gleeson MP. 2008. Generation of a set of simple, interpretable ADMET rules of thumb. J. Med. Chem. 51:817-834. (Pubitemid 351304691)
    • (2008) Journal of Medicinal Chemistry , vol.51 , Issue.4 , pp. 817-834
    • Gleeson, M.P.1
  • 14
    • 77956544478 scopus 로고    scopus 로고
    • The international limits and population at risk of Plasmodium vivax transmission in 2009
    • Guerra CA, et al. 2010. The international limits and population at risk of Plasmodium vivax transmission in 2009. PLoS Negl. Trop. Dis. 4:e774.
    • (2010) PLoS Negl. Trop. Dis. , vol.4
    • Guerra, C.A.1
  • 16
    • 77954309291 scopus 로고    scopus 로고
    • Quinolines and structurally related heterocycles as antimalarials
    • Kaur K, Jain M, Reddy RP, Jain R. 2010. Quinolines and structurally related heterocycles as antimalarials. Eur. J. Med. Chem. 45:3245-3264.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 3245-3264
    • Kaur, K.1    Jain, M.2    Reddy, R.P.3    Jain, R.4
  • 17
    • 78650724579 scopus 로고    scopus 로고
    • Synthesis, antiprotozoal, antimicrobial, β-hematin inhibition, cytotoxicity and methemoglobin (MetHb) formation activities of bis(8-aminoquinolines)
    • Kaur K, et al. 2011. Synthesis, antiprotozoal, antimicrobial, β-hematin inhibition, cytotoxicity and methemoglobin (MetHb) formation activities of bis(8-aminoquinolines). Bioorg. Med. Chem. 19:197-210.
    • (2011) Bioorg. Med. Chem. , vol.19 , pp. 197-210
    • Kaur, K.1
  • 18
    • 78751581687 scopus 로고    scopus 로고
    • The hypnozoite concept, with particular reference to malaria
    • Markus MB. 2011. The hypnozoite concept, with particular reference to malaria. Parasitol. Res. 108:247-252.
    • (2011) Parasitol. Res. , vol.108 , pp. 247-252
    • Markus, M.B.1
  • 19
    • 79952524600 scopus 로고    scopus 로고
    • Primacenes: Novel non-cytotoxic primaquine ferrocene-conjugates with anti-Pneumocystis carinii activity
    • Matos J, et al. 2010. Primacenes: novel non-cytotoxic primaquine ferrocene-conjugates with anti-Pneumocystis carinii activity. Medchemcomm 1:199-201.
    • (2010) Medchemcomm , vol.1 , pp. 199-201
    • Matos, J.1
  • 20
    • 0019830934 scopus 로고
    • Considerations about the structure-activity relationships of 8-aminoquinoline antimalarial drugs
    • McChesney JD. 1981. Considerations about the structure-activity relationships of 8-aminoquinoline antimalarial drugs. Bull. World Health Organ. 59:459-462. (Pubitemid 11024769)
    • (1981) Bulletin of the World Health Organization , vol.59 , Issue.3 , pp. 459-462
    • McChesney, J.D.1
  • 22
    • 77958490216 scopus 로고    scopus 로고
    • Iron potentiates acetaminophen-induced oxidative stress and mitochondrial dysfunction in cultured mouse hepatocytes
    • Moon MS, Richie JP, Isom HC. 2010. Iron potentiates acetaminophen-induced oxidative stress and mitochondrial dysfunction in cultured mouse hepatocytes. Toxicol. Sci. 118:119-127.
    • (2010) Toxicol. Sci. , vol.118 , pp. 119-127
    • Moon, M.S.1    Richie, J.P.2    Isom, H.C.3
  • 23
    • 68949106269 scopus 로고    scopus 로고
    • Key gaps in the knowledge of Plasmodium vivax, a neglected human malaria parasite
    • Mueller I, et al. 2009. Key gaps in the knowledge of Plasmodium vivax, a neglected human malaria parasite. Lancet Infect. Dis. 9:555-566.
    • (2009) Lancet Infect. Dis. , vol.9 , pp. 555-566
    • Mueller, I.1
  • 24
    • 77957557403 scopus 로고    scopus 로고
    • Declining in efficacy of a three-day combination regimen of mefloquine-artesunate in a multi-drug resistance area along the Thai-Myanmar border
    • Na-Bangchang K, Ruengweerayut R, Mahamad P, Ruengweerayut K, Chaijaroenkul W. 2010. Declining in efficacy of a three-day combination regimen of mefloquine-artesunate in a multi-drug resistance area along the Thai-Myanmar border. Malar. J. 9:273.
    • (2010) Malar. J. , vol.9 , pp. 273
    • Na-Bangchang, K.1    Ruengweerayut, R.2    Mahamad, P.3    Ruengweerayut, K.4    Chaijaroenkul, W.5
  • 27
    • 70849097089 scopus 로고    scopus 로고
    • Visualization and quantitative analysis of the rodent malaria liver stage by real time imaging
    • Ploemen IHJ, et al. 2009. Visualization and quantitative analysis of the rodent malaria liver stage by real time imaging. PLoS One 4:e7881.
    • (2009) PLoS One , vol.4
    • Ploemen, I.H.J.1
  • 28
    • 34247266100 scopus 로고    scopus 로고
    • Plasmodium vivax in Africa: hidden in plain sight?
    • DOI 10.1016/j.pt.2007.02.009, PII S1471492207000554
    • Rosenberg R. 2007. Plasmodium vivax in Africa: hidden in plain sight? Trends Parasitol. 23:193-196. (Pubitemid 46618122)
    • (2007) Trends in Parasitology , vol.23 , Issue.5 , pp. 193-196
    • Rosenberg, R.1
  • 29
    • 78651096930 scopus 로고    scopus 로고
    • Antimalarial activity of novel 5-aryl-8-aminoquinoline derivatives
    • Shiraki H, et al. 2011. Antimalarial activity of novel 5-aryl-8-aminoquinoline derivatives. J. Med. Chem. 54:131-142.
    • (2011) J. Med. Chem. , vol.54 , pp. 131-142
    • Shiraki, H.1
  • 30
    • 60549099364 scopus 로고    scopus 로고
    • Primaquine revisited six decades after its discovery
    • Vale N, Moreira R, Gomes P. 2009. Primaquine revisited six decades after its discovery. Eur. J. Med. Chem. 44:937-953.
    • (2009) Eur. J. Med. Chem. , vol.44 , pp. 937-953
    • Vale, N.1    Moreira, R.2    Gomes, P.3
  • 31
    • 72249095184 scopus 로고    scopus 로고
    • Imidazoquines as antimalarial and antipneumocystis agents
    • Vale N, et al. 2009. Imidazoquines as antimalarial and antipneumocystis agents. J. Med. Chem. 52:7800-7807.
    • (2009) J. Med. Chem. , vol.52 , pp. 7800-7807
    • Vale, N.1
  • 32
    • 79551534432 scopus 로고    scopus 로고
    • Plasmodium vivax sub-patent infections after radical treatment are common in Peruvian patients: Results of a 1-year prospective cohort study
    • Van den Eede P, et al. 2011. Plasmodium vivax sub-patent infections after radical treatment are common in Peruvian patients: results of a 1-year prospective cohort study. PLoS One 6:e16257.
    • (2011) PLoS One , vol.6
    • Van Den Eede, P.1
  • 33
    • 76749083725 scopus 로고    scopus 로고
    • Targeting the hypnozoite reservoir of Plasmodium vivax: The hidden obstacle to malaria elimination
    • Wells TNC, Burrows JN, Baird JK. 2010. Targeting the hypnozoite reservoir of Plasmodium vivax: the hidden obstacle to malaria elimination. Trends Parasitol. 26:145-151.
    • (2010) Trends Parasitol. , vol.26 , pp. 145-151
    • Wells, T.N.C.1    Burrows, J.N.2    Baird, J.K.3
  • 34
    • 2142659388 scopus 로고    scopus 로고
    • Antimalarial drug resistance
    • DOI 10.1172/JCI200421682
    • White NJ. 2004. Antimalarial drug resistance. J. Clin. Invest. 113:1084-1092. (Pubitemid 38544090)
    • (2004) Journal of Clinical Investigation , vol.113 , Issue.8 , pp. 1084-1092
    • White, N.J.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.