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ChemMedChem

Volumn 7, Issue 2, 2012, Pages 233-236

Application of Barluenga Boronic Coupling (BBC) to the Parallel Synthesis of Drug-like and Drug Fragment-like Molecules

(6) Nakagawa, Shoko a Bainbridge, Katie A a Butcher, Ken a Ellis, Dave a Klute, Wolfgang a Ryckmans, Thomas a,b

a PFIZER GLOBAL RESEARCH AND DEVELOPMENT (United Kingdom)

b H LUNDBECK A S (Denmark)

Author keywords

Array synthesis; Barluenga boronic coupling; C C bond formation; Drug likeness

Indexed keywords

AZAINDOLE DERIVATIVE; AZETIDINE DERIVATIVE; BORONIC ACID DERIVATIVE; CARBON; IMIDAZOLE DERIVATIVE; INDOLE DERIVATIVE; NITROGEN; OXYGEN; UNCLASSIFIED DRUG;

ACYLATION; ARTICLE; BARLUENGA BORONIC COUPLING; CHEMICAL BOND; CHEMICAL REACTION; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROGEN BOND; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

ALDEHYDES; BORONIC ACIDS; CARBON; HYDRAZONES; PHARMACEUTICAL PREPARATIONS; TOSYL COMPOUNDS;

EID: 84856402670 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100339 Document Type: Article

Times cited : (33)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.