High-throughput screening of potassium-competitive acid blockers

Journal of Biomolecular Screening

Volumn 17, Issue 2, 2012, Pages 177-182

  Kondo, Mitsuyo ^a   Kawamoto, Makiko ^a   Hasuoka, Atsushi ^a   Kajino, Masahiro ^a   Inatomi, Nobuhiro ^a   Tarui, Naoki ^a  

^a TAKEDA PHARMACEUTICAL COMPANY LIMITED   (Japan)

Author keywords

affinity selection mass spectrometry; gastroesophageal reflux disease; H+; high throughput screening; K+ ATPase; potassium competitive acid blocker

Indexed keywords

1 [5 (2 FLUOROPHENYL) 1 (PYRIDIN 3 YLSULFONYL) 1H PYRROL 3 YL]N METHYLMETHANAMINE MONOFUMARATE; 8 BENZYLOXY 2 METHYLIMIDAZO[1,2 A]PYRIDINE 3 ACETONITRILE; HYDROGEN POTASSIUM ADENOSINE TRIPHOSPHATASE; LANSOPRAZOLE; POTASSIUM COMPETITIVE ACID BLOCKER; PYRROLE DERIVATIVE; TAK 438; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; HIGH THROUGHPUT SCREENING; PRIORITY JOURNAL;

ANIMALS; H(+)-K(+)-EXCHANGING ATPASE; HIGH-THROUGHPUT SCREENING ASSAYS; PROTON PUMP INHIBITORS; PYRROLES; SMALL MOLECULE LIBRARIES; SULFONAMIDES; SWINE;

EID: 84856256407     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057111421004     Document Type: Article

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