메뉴 건너뛰기




Volumn 26, Issue 1, 2012, Pages 86-90

Investigation of UDP-glucuronosyltransferases (UGTs) inhibitory properties of carvacrol

Author keywords

carvacrol; drug drug interactions (DDIs); UDP glucuronosyltransferases (UGTs)

Indexed keywords

CARVACROL; GLUCURONOSYLTRANSFERASE; GLUCURONOSYLTRANSFERASE 1A9; HYMECROMONE; PROPOFOL;

EID: 84855684309     PISSN: 0951418X     EISSN: 10991573     Source Type: Journal    
DOI: 10.1002/ptr.3525     Document Type: Article
Times cited : (67)

References (25)
  • 1
    • 0023198881 scopus 로고
    • Metabolism in rats of p-cymene derivatives: Carvacrol and thymol
    • Austgulen LT, Solheim E, Scheline RR,. 1987. Metabolism in rats of p-cymene derivatives: carvacrol and thymol. Pharmacol Toxicol 61: 98-102. (Pubitemid 17136709)
    • (1987) Pharmacology and Toxicology , vol.61 , Issue.2 , pp. 98-102
    • Austgulen, L.-T.1    Solheim, E.2    Scheline, R.R.3
  • 3
    • 8844239121 scopus 로고    scopus 로고
    • Evaluation of carvacrol and eugenol as prophylaxis and treatment of vaginal candidiasis in an immunosuppressed rat model
    • DOI 10.1093/jac/dkh436
    • Chami F, Chami N, Bennis S, Trouillas J, Remmal A,. 2004. Evaluation of carvacrol and eugenol as prophylaxis and treatment of vaginal candidiasis in an immunosuppressed rat model. J Antimicrob Chemother 54: 909-914. (Pubitemid 39529986)
    • (2004) Journal of Antimicrobial Chemotherapy , vol.54 , Issue.5 , pp. 909-914
    • Chami, F.1    Chami, N.2    Bennis, S.3    Trouillas, J.4    Remmal, A.5
  • 4
    • 0033569516 scopus 로고    scopus 로고
    • Pharmacogenomics: Translating functional genomics into rational therapeutics
    • Evans WE, Relling MV,. 1999. Pharmacogenomics: translating functional genomics into rational therapeutics. Science 286: 487-491.
    • (1999) Science , vol.286 , pp. 487-491
    • Evans, W.E.1    Relling, M.V.2
  • 5
    • 33749550685 scopus 로고    scopus 로고
    • Essential oils - Their antimicrobial activity against Escherichia coli and effect on intestinal cell viability
    • Fabian D, Sabol M, Domaracka K, Bujnakova D,. 2006. Essential oils-their antimicrobial activity against Escherichia coli and effect on intestinal cell viability. Toxicol Vitro 20: 1435-1445.
    • (2006) Toxicol Vitro , vol.20 , pp. 1435-1445
    • Fabian, D.1    Sabol, M.2    Domaracka, K.3    Bujnakova, D.4
  • 6
    • 75149152466 scopus 로고    scopus 로고
    • Time-dependent inhibition of CYP3A4 and CYP2C9 by noscapine potentially explains clinical noscapine-warfarin interaction
    • Fang ZZ, Zhang YY, Ge GB, Huo H, Liang SC, Yang L,. 2010. Time-dependent inhibition of CYP3A4 and CYP2C9 by noscapine potentially explains clinical noscapine-warfarin interaction. Br J Clin Pharmacol 69: 193-199.
    • (2010) Br J Clin Pharmacol , vol.69 , pp. 193-199
    • Fang, Z.Z.1    Zhang, Y.Y.2    Ge, G.B.3    Huo, H.4    Liang, S.C.5    Yang, L.6
  • 7
    • 49949113587 scopus 로고    scopus 로고
    • Structure-activity relationship and substrate-dependent phenomena in effects of ginsenosides on activities of drug-metabolizing P450 enzymes
    • Hao M, Zhao Y, Chen P, et al,. 2008. Structure-activity relationship and substrate-dependent phenomena in effects of ginsenosides on activities of drug-metabolizing P450 enzymes. PloS One 3: 1-10.
    • (2008) PloS One , vol.3 , pp. 1-10
    • Hao, M.1    Zhao, Y.2    Chen, P.3
  • 8
    • 78650281301 scopus 로고    scopus 로고
    • Strong inhibitory effect of medroxyprogesterone acetate (MPA) on UDP-glucurosyltransferase (UGT) 2B7 might induce drug-drug interactions
    • Huang T, Fang ZZ, Yang L,. 2010. Strong inhibitory effect of medroxyprogesterone acetate (MPA) on UDP-glucurosyltransferase (UGT) 2B7 might induce drug-drug interactions. Pharmazie 65: 919-921.
    • (2010) Pharmazie , vol.65 , pp. 919-921
    • Huang, T.1    Fang, Z.Z.2    Yang, L.3
  • 9
    • 15244342411 scopus 로고    scopus 로고
    • UDP-glucurosyltransferases and clinical drug-drug interactions
    • Kiang TKL, Ensom MHH, Chang TKH,. 2005. UDP-glucurosyltransferases and clinical drug-drug interactions. Pharmacol Ther 106: 97-132.
    • (2005) Pharmacol Ther , vol.106 , pp. 97-132
    • Kiang, T.K.L.1    Ensom, M.H.H.2    Chang, T.K.H.3
  • 10
    • 18944384699 scopus 로고    scopus 로고
    • Effective treatment of experimental acute otitis media by application of volatile fluids into the ear canal
    • DOI 10.1086/430003
    • Kristinsson KG, Magnusdottir AB, Petersen H, Hermansson A,. 2005. Effective treatment of experimental acute otitis media by application of volatile fluids into the ear canal. J Infect Dis 191: 1876-1880. (Pubitemid 40705395)
    • (2005) Journal of Infectious Diseases , vol.191 , Issue.11 , pp. 1876-1880
    • Kristinsson, K.G.1    Magnusdottir, A.B.2    Petersen, H.3    Hermansson, A.4
  • 11
    • 77957018120 scopus 로고    scopus 로고
    • Determination of propofol UDP-glucuronosyltransferase (UGT) activities in hepatic microsomes from different species by UFLC-ESI-MS
    • Liang SC, Ge GB, Liu HX, et al,. 2011. Determination of propofol UDP-glucuronosyltransferase (UGT) activities in hepatic microsomes from different species by UFLC-ESI-MS. J Pharm Biomed Anal 54: 236-241.
    • (2011) J Pharm Biomed Anal , vol.54 , pp. 236-241
    • Liang, S.C.1    Ge, G.B.2    Liu, H.X.3
  • 12
    • 0031472588 scopus 로고    scopus 로고
    • Role of pharmacokinetics and metabolism in drug discovery and development
    • Lin JH, Lu AYH,. 1997. Role of pharmacokinetics and metabolism in drug discovery and development. Pharmacol Rev 49: 403-449. (Pubitemid 28030947)
    • (1997) Pharmacological Reviews , vol.49 , Issue.4 , pp. 403-449
    • Lin, J.H.1    Lu, A.Y.H.2
  • 13
    • 73149090339 scopus 로고    scopus 로고
    • Comparison of the drug-drug interactions potential of erlotinib and gefitinib via inhibition of UDP-glucuronosyltransferases
    • Liu Y, Ramirez J, House L, Ratain MJ,. 2010. Comparison of the drug-drug interactions potential of erlotinib and gefitinib via inhibition of UDP-glucuronosyltransferases. Drug Metab Dispos 38: 32-39.
    • (2010) Drug Metab Dispos , vol.38 , pp. 32-39
    • Liu, Y.1    Ramirez, J.2    House, L.3    Ratain, M.J.4
  • 15
    • 0031975185 scopus 로고    scopus 로고
    • Update: Clinically significant cytochrome P-450 drug interactions
    • Michalets EL,. 1998. Update: clinically significant cytochrome P450 drug interactions. Pharmacotherapy 18: 84-112. (Pubitemid 28059007)
    • (1998) Pharmacotherapy , vol.18 , Issue.1 , pp. 84-112
    • Michalets, E.L.1
  • 16
    • 15444378115 scopus 로고    scopus 로고
    • A historical overview of the heterologous expression of mammalian UDP-glucuronosyltransferase isoforms over the past twenty years
    • DOI 10.2174/1389200053586127
    • Radominska-Pandya A, Bratton S, Little JM,. 2005. A historical overview of the heterologous expression of mammalian UDP-glucuronosyltransferase isoforms over the past twenty years. Curr Drug Metab 6: 141-160. (Pubitemid 40394342)
    • (2005) Current Drug Metabolism , vol.6 , Issue.2 , pp. 141-160
    • Radominska-Pandya, A.1    Bratton, S.2    Little, J.M.3
  • 17
    • 0034534895 scopus 로고    scopus 로고
    • Roles of glucuronidation and UDP-glucuronosyltransferases in xenobiotic bioactivation reactions
    • DOI 10.1016/S0009-2797(00)00198-8, PII S0009279700001988
    • Ritter JK,. 2000. Roles of glucuronidation and UDP- glucuronosyltransferases in xenobiotic bioactivation reactions. Chem Biol Interact 129: 171-193. (Pubitemid 32061059)
    • (2000) Chemico-Biological Interactions , vol.129 , Issue.1-2 , pp. 171-193
    • Ritter, J.K.1
  • 18
    • 0242668347 scopus 로고    scopus 로고
    • Pharmacophore and quantitative structure-activity relationship modeling: Complementary approaches for the rationalization and prediction of UDP-glucuronosyltransferase 1A4 substrate selectivity
    • DOI 10.1021/jm020397c
    • Smith PA, Sorich MJ, McKinnon RA, Miners JO,. 2003. Pharmacophore and quantitative structure-activity relationship modeling: complementary approaches for the rationalization and prediction of UDP-glucuronosyltransferase 1A4 substrate selectivity. J Med Chem 46: 1617-1626. (Pubitemid 36444215)
    • (2003) Journal of Medicinal Chemistry , vol.46 , Issue.9 , pp. 1617-1626
    • Smith, P.A.1    Sorich, M.J.2    McKinnon, R.A.3    Miners, J.O.4
  • 19
    • 0032882744 scopus 로고    scopus 로고
    • Toxicity of selected plant volatiles in microbial and mammalian short-term assays
    • DOI 10.1016/S0278-6915(99)00075-7, PII S0278691599000757
    • Stammati A, Bonsi P, Zucco F, Moezelaar R, Alakomi HL, vonWright A,. 1999. Toxicity of selected plant volatiles in microbial and mammalian short-term assays. Food Chem Toxicol 37: 813-823. (Pubitemid 29472432)
    • (1999) Food and Chemical Toxicology , vol.37 , Issue.8 , pp. 813-823
    • Stammati, A.1    Bonsi, P.2    Zucco, F.3    Moezelaar, R.4    Alakomi, H.-L.5    Von Wright, A.6
  • 20
    • 0033664783 scopus 로고    scopus 로고
    • Substrate-dependent modulation of CYP3A4 catalytic activity: Analysis of 27 test compounds with four fluorometric substrates
    • Stresser DM, Blanchard AP, Turner SD, et al,. 2000. Substrate-dependent modulation of CYP3A4 catalytic activity: analysis of 27 test compounds with four fluorometric substrates. Drug Metab Dispos 28: 1440-1448.
    • (2000) Drug Metab Dispos , vol.28 , pp. 1440-1448
    • Stresser, D.M.1    Blanchard, A.P.2    Turner, S.D.3
  • 21
    • 77955646498 scopus 로고    scopus 로고
    • Inhibitory effects of curcumenol on human liver cytochrome P450 enzymes
    • Sun DX, Fang ZZ, Zhang YY, Cao YF, Yang L, Yin J,. 2010. Inhibitory effects of curcumenol on human liver cytochrome P450 enzymes. Phytother Res 24: 1213-1216.
    • (2010) Phytother Res , vol.24 , pp. 1213-1216
    • Sun, D.X.1    Fang, Z.Z.2    Zhang, Y.Y.3    Cao, Y.F.4    Yang, L.5    Yin, J.6
  • 22
    • 0032456884 scopus 로고    scopus 로고
    • Clinically important pharmacokinetic drug-drug interactions: Role of cytochrome P450 enzymes
    • DOI 10.1046/j.1365-2710.1998.00086.x
    • Tanaka E,. 1998. Clinically important pharmacokinetic drug-drug interactions: role of cytochrome P450 enzymes. J Clin Pharm Ther 23: 403-416. (Pubitemid 29060690)
    • (1998) Journal of Clinical Pharmacy and Therapeutics , vol.23 , Issue.6 , pp. 403-416
    • Tanaka, E.1
  • 23
    • 0034128936 scopus 로고    scopus 로고
    • Human UDP-glucuronosyltransferases: Metabolism, expression, and disease
    • DOI 10.1146/annurev.pharmtox.40.1.581
    • Tukey RH, Strassburg CP,. 2000. Human UDP-glucuronosyltransferases: metabolism, expression, and disease. Annu Rev Pharmacol Toxicol 40: 581-616. (Pubitemid 30340694)
    • (2000) Annual Review of Pharmacology and Toxicology , vol.40 , pp. 581-616
    • Tukey, R.H.1    Strassburg, C.P.2
  • 25
    • 2342500889 scopus 로고    scopus 로고
    • Immunostimulatory effect of dietary oregano etheric oils on lymphocytes from growth-retarded, low-weight growing-finishing pigs and productivity
    • Walter BM, Bilkei G,. 2004. Immunostimulatory effect of dietary oregano etheric oils on lymphocytes from growth-retarded, low-weight growing-finishing pigs and productivity. Tijdschrift voor diergeneeskundeunde 129: 178-181. (Pubitemid 38609950)
    • (2004) Tijdschrift voor Diergeneeskunde , vol.129 , Issue.6 , pp. 178-181
    • Walter, B.M.1    Bilkei, G.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.