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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 2, 2012, Pages 820-823

Synthesis, pharmacological evaluation and docking studies of N-(benzo[d]thiazol-2-yl)-2-(piperazin-1-yl)acetamide analogs as COX-2 inhibitors

(4) Raghavendra, Nulgumnalli Manjunathaiah a Jyothsna, Aitha a Venkateswara Rao, Alapati a Subrahmanyam, C V S a

a Osmania University (India)

Author keywords

2 Amino benzothiazole; Anti inflammatory activity; Computer aided drug design; Docking studies; Piperazine; Ulcerogenic activity

Indexed keywords

ANTIINFLAMMATORY AGENT; CYCLOOXYGENASE 2; N (BENZO[D]THIAZOL 2 YL) 2 (PIPERAZIN 1 YL)ACETAMIDE DERIVATIVE; NAPROXEN; ROFECOXIB; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG PROTEIN BINDING; DRUG SCREENING; DRUG SYNTHESIS; IN VIVO STUDY; MOLECULAR DOCKING; NONHUMAN; PAW EDEMA; RAT;

ACETAMIDES; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; BENZOTHIAZOLES; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITORS; DRUG DISCOVERY; MODELS, MOLECULAR; MOLECULAR STRUCTURE; STEREOISOMERISM;

RUMEX;

EID: 84855655313 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.12.062 Document Type: Article

Times cited : (42)

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