Druggability of methyl-lysine binding sites

Journal of Computer-Aided Molecular Design

Volumn 25, Issue 12, 2011, Pages 1171-1178

  Santiago, C ^a   Nguyen, K ^a   Schapira, M ^b  

^a UNIVERSITY OF TORONTO   (Canada)

^b UNIVERSITY OF TORONTO   (Canada)

Author keywords

Binding pocket; Druggability; Epigenetics; Inhibitors; Methyl lysine

Indexed keywords

AMINO ACIDS; BINDING SITES; GENE EXPRESSION REGULATION; PROTEINS;

BINDING POCKETS; DRUGGABILITY; EPIGENETIC REGULATION; EPIGENETICS; INHIBITOR; LYSINE RESIDUES; LYSINE-BINDING SITES; MEDIATED SIGNALLING; METHYL-LYSINE; STRUCTURAL MODULE;

GENE EXPRESSION;

HISTONE; LYSINE;

ARTICLE; BINDING SITE; HISTONE MODIFICATION; MOLECULAR INTERACTION; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN FUNCTION; PROTEIN SECONDARY STRUCTURE; PROTEIN TARGETING; SIGNAL TRANSDUCTION; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

EID: 84855194838     PISSN: 0920654X     EISSN: 15734951     Source Type: Journal    
DOI: 10.1007/s10822-011-9505-2     Document Type: Article

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