LDV peptidomimetics equipped with biotinylated spacer-arms: Synthesis and biological evaluation on CCRF-CEM cell line

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 1, 2012, Pages 586-590

  Gérard, Estelle ^a   Meulle, Aline ^a   Feron, Olivier ^a   Marchand Brynaert, Jacqueline ^a  

^a UNIVERSITÉ CATHOLIQUE DE LOUVAIN   (Belgium)

Author keywords

4 1 Integrin antagonists; Biotin conjugated peptidomimetics; CCRF CEM cell line; LDV peptidomimetics

Indexed keywords

AVIDIN; BIOTIN; BIOTIN CONJUGATED LEUCYLASPARTYLVALINE; NEUTRAVIDIN; PEPTIDOMIMETIC AGENT; TRIPEPTIDE; UNCLASSIFIED DRUG; VERY LATE ACTIVATION ANTIGEN 4;

ADHESION; ARTICLE; BIOTINYLATION; CHEMICAL INTERACTION; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; FLUORESCENCE; HUMAN; HUMAN CELL; LEUKAPHERESIS; LEUKEMIA CELL LINE;

ANTINEOPLASTIC AGENTS; BIOTIN; CELL ADHESION; CELL LINE; CELL LINE, TUMOR; CHEMISTRY, PHARMACEUTICAL; DRUG DESIGN; GENE EXPRESSION REGULATION, LEUKEMIC; HUMANS; INHIBITORY CONCENTRATION 50; INTEGRIN ALPHA4BETA1; KINETICS; LEUKEMIA; MODELS, CHEMICAL; OLIGOPEPTIDES; PEPTIDES; PEPTIDOMIMETICS;

EID: 84655169565     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.10.078     Document Type: Article

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