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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 1, 2012, Pages 523-526

(±)-2-(N-tert-Butylamino)-3′-[ 125I]-iodo-4′- azidopropiophenone: A dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban)

(9) Lapinsky, David J a Aggarwal, Shaili a Nolan, Tammy L a Surratt, Christopher K a Lever, John R b,c Acharya, Rejwi d Vaughan, Roxanne A d Pandhare, Akash e Blanton, Michael P e

a DUQUESNE UNIVERSITY (United States)

b University of Missouri (United States)

c VETERANS AFFAIRS MEDICAL CENTER (United States)

d UNIVERSITY OF NORTH DAKOTA SCHOOL OF MEDICINE AND HEALTH SCIENCES (United States)

e TEXAS TECH UNIVERSITY (United States)

Author keywords

Bupropion; Dopamine transporter; Nicotinic acetylcholine receptor; Photoaffinity labeling

Indexed keywords

2 (N TERT BUTYLAMINO) 3' [IODINE 125]IODO 4' AZIDOPROPIOPHENONE; AMFEBUTAMONE; AZIDE; COCAINE; DOPAMINE TRANSPORTER; IODINE; LIPID; NICOTINIC RECEPTOR; PROPIOPHENONE DERIVATIVE; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; CELL CULTURE; CELL MEMBRANE; CHANNEL GATING; CONTROLLED STUDY; COVALENT BOND; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; INCUBATION TEMPERATURE; INCUBATION TIME; PHOTOAFFINITY LABELING; PHOTOREACTIVITY; PROTEIN PURIFICATION; RADIOIODINATION;

AZIDES; BUPROPION; CHEMISTRY, PHARMACEUTICAL; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; DRUG DESIGN; HUMANS; IODINE; IODINE RADIOISOTOPES; KINETICS; LIGANDS; MODELS, CHEMICAL; PHOTOCHEMISTRY; RECEPTORS, NICOTINIC;

EID: 84655164867 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.10.086 Document Type: Article

Times cited : (10)

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