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Volumn 30, Issue 4, 2011, Pages 403-409

T-type calcium channel blockers - New and notable

Author keywords

Dihydropyridines; Phenylakylamines; T type calcium channels; Zn 2+, Cu 2+, Ni 2+, Co 2+, Cd 2+, La 3+, Er 3+, Y 3+

Indexed keywords

AMLODIPINE; BENIDIPINE; CADMIUM; CALCIUM CHANNEL BLOCKING AGENT; CALCIUM CHANNEL L TYPE; CALCIUM CHANNEL T TYPE; COBALT; CUPRIC ION; DIHYDROPYRIDINE; EFONIDIPINE; HISTIDINE; ISRADIPINE; LANTHANIDE; LANTHANUM; NICKEL; NIFEDIPINE; NIMODIPINE; PHENYLALKYLAMINE; VERAPAMIL; VOLTAGE GATED CALCIUM CHANNEL; YTTRIUM; ZINC ION;

EID: 83155182705     PISSN: 02315882     EISSN: None     Source Type: Journal    
DOI: 10.4149/gpb_2011_04_403     Document Type: Short Survey
Times cited : (25)

References (63)
  • 2
    • 0036595607 scopus 로고    scopus 로고
    • Inhibition of transiently expressed low- and high-voltage-activated calcium channels by trivalent metal cations
    • DOI 10.1007/s00232-001-0166-2
    • Beedle A. M., Hamid J., Zamponi G. W. (2002): Inhibition of transiently expressed low- and high-voltage-activated calcium channels by trivalent metal cations. J. Membr. Biol. 187, 225-238 http://dx.doi.org/10.1007/s00232-001-0166- 2 (Pubitemid 34587778)
    • (2002) Journal of Membrane Biology , vol.187 , Issue.3 , pp. 225-238
    • Beedle, A.M.1    Hamid, J.2    Zamponi, G.W.3
  • 6
    • 82255177148 scopus 로고    scopus 로고
    • Nimodipine inhibits AP firing in cultured hippocampal neurons predominantly due to block of voltage-dependent potassium channels
    • Caro A., Tarabova B., Rojo-Ruiz J., Lacinova L. (2011): Nimodipine inhibits AP firing in cultured hippocampal neurons predominantly due to block of voltage-dependent potassium channels. Gen. Physiol. Biophys. 30 (Special Issue), S44-53
    • (2011) Gen. Physiol. Biophys. , vol.30 , Issue.SPEC. ISSUE
    • Caro, A.1    Tarabova, B.2    Rojo-Ruiz, J.3    Lacinova, L.4
  • 9
    • 74849102076 scopus 로고    scopus 로고
    • The dihydropyridine analogue cerebrocrast blocks both T-type and L-type calcium currents
    • Drigelova M., Tarabova B., Duburs G., Lacinova L. (2009): The dihydropyridine analogue cerebrocrast blocks both T-type and L-type calcium currents. Can. J. Physiol. Pharmacol. 87, 923-932 http://dx.doi.org/10.1139/Y09- 086
    • (2009) Can. J. Physiol. Pharmacol. , vol.87 , pp. 923-932
    • Drigelova, M.1    Tarabova, B.2    Duburs, G.3    Lacinova, L.4
  • 11
    • 0033135444 scopus 로고    scopus 로고
    • One calcium ion
    • may suffice to open the tetrameric cardiac ryanodine receptor in rat ventricular myocytes.
    • Fan J. S., Palade P. (1999): One calcium ion may suffice to open the tetrameric cardiac ryanodine receptor in rat ventricular myocytes. J. Physiol. 516, 769-780 http://dx.doi.org/10.1111/j.1469-7793.1999.0769u.x
    • (1999) J. Physiol. , vol.516 , pp. 769-780
    • Fan, J.S.1    Palade, P.2
  • 12
    • 0023518468 scopus 로고
    • Kinetic and pharmacological properties distinguishing three types of calcium currents in chick sensory neurones
    • Fox A. P., Nowycky M. C., Tsien R. W. (1987): Kinetic and pharmacological properties distinguishing three types of calcium currents in chick sensory neurones. J. Physiol. 394, 149-172 (Pubitemid 18005128)
    • (1987) Journal of Physiology , vol.394 , pp. 149-172
    • Fox, A.P.1    Nowycky, M.C.2    Tsien, R.W.3
  • 17
    • 14844323679 scopus 로고    scopus 로고
    • Effects of diltiazem and nifedipine on transient outward and ultra-rapid delayed rectifier potassium currents in human atrial myocytes
    • DOI 10.1038/sj.bjp.0706113
    • Gao Z., Sun H., Chiu S. W., Lau C. P., Li G. R. (2005): Effects of diltiazem and nifedipine on transient outward and ultra-rapid delayed rectifier potassium currents in human atrial myocytes. Br. J. Pharmacol. 144, 595-604 http://dx.doi.org/10.1038/sj.bjp.0706113 (Pubitemid 40349467)
    • (2005) British Journal of Pharmacology , vol.144 , Issue.4 , pp. 595-604
    • Gao, Z.1    Sun, H.2    Chiu, S.-W.3    Lau, C.-P.4    Li, G.-R.5
  • 18
    • 0025355645 scopus 로고
    • Calcium channels in vertebrate cells
    • Hess P. (1990): Calcium channels in vertebrate cells. Annu Rev Neurosci. 13, 337-356 http://dx.doi.org/10.1146/annurev.ne.13.030190.002005
    • (1990) Annu Rev Neurosci. , vol.13 , pp. 337-356
    • Hess, P.1
  • 19
    • 0029153731 scopus 로고
    • Molecular determinants of high affinity phenylalkylamine block of L-type calcium channels
    • Hockerman G. H., Johnson B. D., Scheuer T., Catterall W. A. (1995): Molecular determinants of high affinity phenylalkylamine block of L-type calcium channels. J. Biol. Chem. 270, 22119-22122 http://dx.doi.org/10.1074/jbc.270.38. 22119
    • (1995) J. Biol. Chem. , vol.270 , pp. 22119-22122
    • Hockerman, G.H.1    Johnson, B.D.2    Scheuer, T.3    Catterall, W.A.4
  • 20
    • 0026657389 scopus 로고
    • Impact of food on the pharmacokinetics and electrocardiographic effects of sustained release verapamil in normal subjects
    • Hoon T. J., McCollam P. L., Beckman K. J., Hariman R. J., Bauman J. L. (1992): Impact of food on the pharmacokinetics and electrocardiographic effects of sustained release verapamil in normal subjects. Am. J. Cardiol. 70, 1072-1076 http://dx.doi.org/10.1016/0002-9149(92)90363-4
    • (1992) Am. J. Cardiol. , vol.70 , pp. 1072-1076
    • Hoon, T.J.1    McCollam, P.L.2    Beckman, K.J.3    Hariman, R.J.4    Bauman, J.L.5
  • 22
    • 58149127278 scopus 로고    scopus 로고
    • Regulation of neuronal T-type calcium channels
    • Iftinca M. C., Zamponi G. W. (2009): Regulation of neuronal T-type calcium channels. Trends Pharmacol. Sci. 30, 32-40 http://dx.doi.org/10.1016/j. tips.2008.10.004
    • (2009) Trends Pharmacol. Sci. , vol.30 , pp. 32-40
    • Iftinca, M.C.1    Zamponi, G.W.2
  • 24
    • 0042833114 scopus 로고    scopus 로고
    • Divalent metals differentially block cloned T-type calcium channels
    • Jeong S. W., Park B. G., Park J. Y., Lee J. W., Lee J. H. (2003): Divalent metals differentially block cloned T-type calcium channels. Neuroreport 14, 1537-1540 http://dx.doi.org/10.1097/00001756-200308060-00028
    • (2003) Neuroreport , vol.14 , pp. 1537-1540
    • Jeong, S.W.1    Park, B.G.2    Park, J.Y.3    Lee, J.W.4    Lee, J.H.5
  • 25
    • 0029847081 scopus 로고    scopus 로고
    • Distinct effects of mutations in transmembrane segment IVS6 on block of L-type calcium channels by structurally similar phenylalkylamines
    • Johnson B. D., Hockerman G. H., Scheuer T., Catterall W. A. (1996): Distinct effects of mutations in transmembrane segment IVS6 on block of L-type calcium channels by structurally similar phenylalkylamines. Mol. Pharmacol. 50, 1388-1400 (Pubitemid 26384878)
    • (1996) Molecular Pharmacology , vol.50 , Issue.5 , pp. 1388-1400
    • Johnson, B.D.1    Hockerman, G.H.2    Scheuer, T.3    Catterall, W.A.4
  • 29
    • 78650645098 scopus 로고    scopus 로고
    • V3.1 channel affects amplitude but not voltage dependence of gating current
    • V3.1 channel affects amplitude but not voltage dependence of gating current. Gen. Physiol. Biophys. 29, 419-423 http://dx.doi.org/10.4149/gpb-2010-04-419
    • (2010) Gen. Physiol. Biophys. , vol.29 , pp. 419-423
    • Karmazinova, M.1    Lacinova, L.2
  • 31
    • 0028211303 scopus 로고
    • The stretch-activated ion channel blocker gadolinium also blocks L-type calcium channels in isolated ventricular myocytes of the guinea-pig
    • DOI 10.1016/0005-2736(94)90250-X
    • Lacampagne A., Gannier F., Argibay J., Garnier D., Le Guennec J. Y. (1994): The stretch-activated ion channel blocker gadolinium also blocks L-type calcium channels in isolated ventricular myocytes of the guinea-pig. Biochim. Biophys. Acta 1191, 205-208 http://dx.doi.org/10.1016/0005-2736(94)90250-X (Pubitemid 24133546)
    • (1994) Biochimica et Biophysica Acta - Biomembranes , vol.1191 , Issue.1 , pp. 205-208
    • Lacampagne, A.1    Gannier, F.2    Argibay, J.3    Garnier, D.4    Le, G.J.-Y.5
  • 32
    • 2642553932 scopus 로고    scopus 로고
    • Pharmacology of recombinant low-voltage activated calcium channels
    • Lacinova L. (2004): Pharmacology of recombinant low-voltage activated calcium channels. Curr. Drug Targets CNS Neurol. Disord. 3, 105-111 http://dx.doi.org/10.2174/1568007043482543
    • (2004) Curr. Drug Targets CNS Neurol. Disord. , vol.3 , pp. 105-111
    • Lacinova, L.1
  • 33
    • 0034018917 scopus 로고    scopus 로고
    • Regulation of the calcium channel α(1G) subunit by divalent cations and organic blockers
    • DOI 10.1016/S0028-3908(99)00202-6, PII S0028390899002026
    • Lacinova L., Klugbauer N., Hofmann F. (2000): Regulation of the calcium channel α1G subunit by divalent cations and organic blockers. Neuropharmacology 39, 1254-1266 http://dx.doi.org/10.1016/S0028-3908(99)00202-6 (Pubitemid 30173189)
    • (2000) Neuropharmacology , vol.39 , Issue.7 , pp. 1254-1266
    • Lacinova, L.1    Klugbauer, N.2    Hofmann, F.3
  • 35
    • 0029154693 scopus 로고
    • The block of the expressed L-type calcium channel is modulated by the β3 subunit
    • Lacinova L., Ludwig A., Bosse E., Flockerzi V., Hofmann F. (1995): The block of the expressed L-type calcium channel is modulated by the β3 subunit. FEBS Lett. 373, 103-107 http://dx.doi.org/10.1016/0014-5793(95)01013-5
    • (1995) FEBS Lett. , vol.373 , pp. 103-107
    • Lacinova, L.1    Ludwig, A.2    Bosse, E.3    Flockerzi, V.4    Hofmann, F.5
  • 36
    • 0026074308 scopus 로고
    • The calcium antagonist D600 inhibits calcium-independent transient outward current in isolated rat ventricular myocytes
    • Lefevre I. A., Coulombe A., Coraboeuf E. (1991): The calcium antagonist D600 inhibits calcium-independent transient outward current in isolated rat ventricular myocytes. J Physiol. 432, 65-80
    • (1991) J Physiol. , vol.432 , pp. 65-80
    • Lefevre, I.A.1    Coulombe, A.2    Coraboeuf, E.3
  • 37
    • 0034973174 scopus 로고    scopus 로고
    • Influence of permeating ions on Kv1.5 channel block by nifedipine
    • Lin S., Wang Z., Fedida D. (2001): Influence of permeating ions on Kv1.5 channel block by nifedipine. Am. J. Physiol. Heart Circ. Physiol. 280, H1160-1172
    • (2001) Am. J. Physiol. Heart Circ. Physiol. , vol.280
    • Lin, S.1    Wang, Z.2    Fedida, D.3
  • 39
    • 33746379873 scopus 로고    scopus 로고
    • Zinc and copper: Pharmacological probes and endogenous modulators of neuronal excitability
    • DOI 10.1016/j.pharmthera.2005.11.004, PII S0163725805002664
    • Mathie A., Sutton G. L., Clarke C. E., Veale E. L. (2006): Zinc and copper: pharmacological probes and endogenous modulators of neuronal excitability. Pharmacol. Ther. 111, 567-583 http://dx.doi.org/10.1016/j. pharmthera.2005.11.004 (Pubitemid 44118429)
    • (2006) Pharmacology and Therapeutics , vol.111 , Issue.3 , pp. 567-583
    • Mathie, A.1    Sutton, G.L.2    Clarke, C.E.3    Veale, E.L.4
  • 40
    • 0027268632 scopus 로고
    • Block of current through T-type calcium channels by trivalent metal cations and nickel in neural rat and human cells
    • Mlinar B., Enyeart J. J. (1993): Block of current through T-type calcium channels by trivalent metal cations and nickel in neural rat and human cells. J. Physiol. 469, 639-652 (Pubitemid 23281600)
    • (1993) Journal of Physiology , vol.469 , pp. 639-652
    • Mlinar, B.1    Enyeart, J.J.2
  • 42
    • 34547693209 scopus 로고    scopus 로고
    • Reducing agents sensitize C-type nociceptors by relieving high-affinity zinc inhibition of T-type calcium channels
    • DOI 10.1523/JNEUROSCI.1800-07.2007
    • Nelson M. T., Woo J., Kang H. W., Vitko I., Barrett P. Q., Perez-Reyes E., Lee J. H., Shin H. S., Todorovic S. M. (2007b): Reducing agents sensitize C-type nociceptors by relieving high-affinity zinc inhibition of T-type calcium channels. J. Neurosci. 27, 8250-8260 http://dx.doi.org/10.1523/JNEUROSCI.1800- 07.2007 (Pubitemid 47219607)
    • (2007) Journal of Neuroscience , vol.27 , Issue.31 , pp. 8250-8260
    • Nelson, M.T.1    Woo, J.2    Kang, H.-W.3    Vitko, I.4    Barrett, P.Q.5    Perez-Reyes, E.6    Lee, J.-H.7    Shin, H.-S.8    Todorovic, S.M.9
  • 43
    • 77952885871 scopus 로고    scopus 로고
    • 2+ enhances the intrinsic bursting activity of a rat thalamic relay neuron
    • 2+ enhances the intrinsic bursting activity of a rat thalamic relay neuron. Neurosci. Res. 67, 95-97 http://dx.doi.org/10.1016/j.neures.2010.01.008
    • (2010) Neurosci. Res. , vol.67 , pp. 95-97
    • Noh, J.1    Choi, H.J.2    Chung, J.M.3
  • 44
    • 77049105127 scopus 로고    scopus 로고
    • 2+ channels in a rat thalamic relay neuron
    • 2+ channels in a rat thalamic relay neuron. Neurosci. Res. 66, 353-358 http://dx.doi.org/10.1016/j. neures.2009.12.005
    • (2010) Neurosci. Res. , vol.66 , pp. 353-358
    • Noh, J.1    Kim, M.K.2    Chung, J.M.3
  • 47
    • 59649126705 scopus 로고    scopus 로고
    • 2+ channels: Block by antihypertensives, antiarrhythmics, and their analogs
    • 2+ channels: block by antihypertensives, antiarrhythmics, and their analogs. J. Pharmacol. Exp. Ther. 328, 621-627 http://dx.doi.org/10.1124/jpet.108.145672
    • (2009) J. Pharmacol. Exp. Ther. , vol.328 , pp. 621-627
    • Perez-Reyes, E.1    Van Deusen, A.L.2    Vitko, I.3
  • 48
    • 33750113366 scopus 로고    scopus 로고
    • Skin bioavailability of dietary vitamin E, carotenoids, polyphenols, vitamin C, zinc and selenium
    • DOI 10.1079/BJN20061817
    • Richelle M., Sabatier M., Steiling H., Williamson G. (2006): Skin bioavailability of dietary vitamin E, carotenoids, polyphenols, vitamin C, zinc and selenium. Br. J. Nutr. 96, 227-238 http://dx.doi.org/10.1079/BJN20061817 (Pubitemid 46476322)
    • (2006) British Journal of Nutrition , vol.96 , Issue.2 , pp. 227-238
    • Richelle, M.1    Sabatier, M.2    Steiling, H.3    Williamson, G.4
  • 49
    • 0033638022 scopus 로고    scopus 로고
    • + channel mKv1.3 by the phenylalkylamine verapamil: Kinetic aspects of block and disruption of accumulation of block by a single point mutation
    • + channel mKv1.3 by the phenylalkylamine verapamil: kinetic aspects of block and disruption of accumulation of block by a single point mutation. Br J Pharmacol. 131, 1275-1284 http://dx.doi.org/10.1038/sj.bjp.0703723
    • (2000) Br J Pharmacol. , vol.131 , pp. 1275-1284
    • Robe, R.J.1    Grissmer, S.2
  • 52
    • 0030013986 scopus 로고    scopus 로고
    • The IVS6 segment of the L-type calcium channel is critical for the action of dihydropyridines and phenylalkylamines
    • Schuster A., Lacinova L., Klugbauer N., Ito H., Birnbaumer L., Hofmann F. (1996): The IVS6 segment of the L-type calcium channel is critical for the action of dihydropyridines and phenylalkylamines. Embo. J. 15, 2365-2370 (Pubitemid 26156562)
    • (1996) EMBO Journal , vol.15 , Issue.10 , pp. 2365-2370
    • Schuster, A.1    Lacinova, L.2    Klugbauer, N.3    Ito, H.4    Birnbaumer, L.5    Hofmann, F.6
  • 53
    • 34548203177 scopus 로고    scopus 로고
    • 2+ sensitivity of high- And low-voltage activated calcium channels
    • 2+ sensitivity of high- and low-voltage activated calcium channels. Biophys. J. 93, 1175-1183 http://dx.doi.org/10.1529/biophysj.106.103333
    • (2007) Biophys. J. , vol.93 , pp. 1175-1183
    • Sun, H.S.1    Hui, K.2    Lee, D.W.3    Feng, Z.P.4
  • 54
    • 33750319950 scopus 로고    scopus 로고
    • 2+ channels
    • DOI 10.1007/s00424-006-0129-7
    • Talavera K., Nilius B. (2006): Evidence for common structural determinants of activation and inactivation in T-type Ca2+ channels. Pflugers Arch. 453, 189-201 http://dx.doi.org/10.1007/s00424-006-0129-7 (Pubitemid 44630453)
    • (2006) Pflugers Archiv European Journal of Physiology , vol.453 , Issue.2 , pp. 189-201
    • Talavera, K.1    Nilius, B.2
  • 56
    • 33845788095 scopus 로고    scopus 로고
    • Subunit-specific modulation of T-type calcium channels by zinc
    • DOI 10.1113/jphysiol.2006.114496
    • Traboulsie A., Chemin J., Chevalier M., Quignard J. F., Nargeot J., Lory P. (2007): Subunit-specific modulation of T-type calcium channels by zinc. J Physiol. 578, 159-171 http://dx.doi.org/10.1113/jphysiol.2006.114496 (Pubitemid 44971117)
    • (2007) Journal of Physiology , vol.578 , Issue.1 , pp. 159-171
    • Traboulsie, A.1    Chemin, J.2    Chevalier, M.3    Quignard, J.-F.4    Nargeot, J.5    Lory, P.6
  • 57
    • 34249049430 scopus 로고    scopus 로고
    • Calcium channel antagonists: Clinical uses - Past, present and future
    • Triggle D. J. (2007): Calcium channel antagonists: clinical uses - past, present and future. Biochem. Pharmacol. 74, 1-9 http://dx.doi.org/10.1016/j.bcp. 2007.01.016
    • (2007) Biochem. Pharmacol. , vol.74 , pp. 1-9
    • Triggle, D.J.1
  • 58
    • 0023778390 scopus 로고
    • Multiple types of neuronal calcium channels and their selective modulation
    • Tsien R. W., Lipscombe D., Madison D. V., Bley K. R., Fox A. P. (1988): Multiple types of neuronal calcium channels and their selective modulation. Trends Neurosci. 11, 431-438 http://dx.doi.org/10.1016/0166-2236(88)90194-4
    • (1988) Trends Neurosci. , vol.11 , pp. 431-438
    • Tsien, R.W.1    Lipscombe, D.2    Madison, D.V.3    Bley, K.R.4    Fox, A.P.5
  • 61
    • 0029120855 scopus 로고
    • Extracellular site of action of phenylalkylamines on L-type calcium current in rat ventricular myocytes
    • Wegener J. W., Nawrath H. (1995): Extracellular site of action of phenylalkylamines on L-type calcium current in rat ventricular myocytes. Naunyn Schmiedebergs Arch. Pharmacol. 352, 322-330 http://dx.doi.org/10.1007/BF00168564
    • (1995) Naunyn Schmiedebergs Arch. Pharmacol. , vol.352 , pp. 322-330
    • Wegener, J.W.1    Nawrath, H.2
  • 62
    • 0032926279 scopus 로고    scopus 로고
    • Structure and functional characterization of a novel human low-voltage activated calcium channel
    • DOI 10.1046/j.1471-4159.1999.0720791.x
    • Williams M. E., Washburn M. S., Hans M., Urrutia A., Brust P. F., Prodanovich P., Harpold M. M., Stauderman K. A. (1999): Structure and functional characterization of a novel human low-voltage activated calcium channel. J. Neurochem. 72, 791-799 http://dx.doi.org/10.1046/j.1471-4159.1999.0720791.x (Pubitemid 29055245)
    • (1999) Journal of Neurochemistry , vol.72 , Issue.2 , pp. 791-799
    • Williams, M.E.1    Washburn, M.S.2    Hans, M.3    Urrutia, A.4    Brust, P.F.5    Prodanovich, P.6    Harpold, M.M.7    Stauderman, K.A.8
  • 63
    • 0028942570 scopus 로고
    • Pharmacokinetic interaction between isradipine and lovastatin in normal, female and male volunteers
    • Zhou L. X., Finley D. K., Hassell A. E., Holtzman J. L. (1995): Pharmacokinetic interaction between isradipine and lovastatin in normal, female and male volunteers. J. Pharmacol. Exp. Ther. 273, 121-127
    • (1995) J. Pharmacol. Exp. Ther. , vol.273 , pp. 121-127
    • Zhou, L.X.1    Finley, D.K.2    Hassell, A.E.3    Holtzman, J.L.4


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