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The efficacy was expressed as the percent effect compared to that of the control, 50 μM oleoylethanolamide, defined as 100%
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Log D and solubility measurements were made as described in
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Log D and solubility measurements were made as described in: D. Buttar, N. Colclough, S. Gerhardt, P.A. MacFaul, S.D. Phillips, A. Plowright, P. Whittamore, K. Tam, K. Maskos, S. Steinbacher, and H. Steuber Bioorg. Med. Chem. 18 2010 7486
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For a recent example of LLE being used out-with an inhibitors/antagonists context see
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