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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 23, 2011, Pages 7068-7071

A small molecule that preferentially binds the closed conformation of Hsp90

(4) Alexander, Leslie D b Partridge, James R c Agard, David A c McAlpine, Shelli R a

a UNIVERSITY OF NEW SOUTH WALES (Australia)

b SAN DIEGO STATE UNIVERSITY (United States)

c UNIVERSITY OF CALIFORNIA (United States)

Author keywords

Anistropy; Anticancer; Fluorescein; Fluorescence polarization; Hsp90; Sansalvamide A

Indexed keywords

ADENOSINE TRIPHOSPHATE; AMIDE; FLUORESCEIN; HEAT SHOCK PROTEIN 90; MACROCYCLIC COMPOUND; SANSALVAMIDE A; UNCLASSIFIED DRUG;

ANISOTROPY; ARTICLE; BINDING AFFINITY; CONFORMATION; DRUG MECHANISM; DRUG STRUCTURE; DRUG SYNTHESIS; IC 50; POLARIZATION; PROTEIN CONFORMATION;

ADENOSINE TRIPHOSPHATE; BINDING SITES; DEPSIPEPTIDES; FLUORESCEIN; HSP90 HEAT-SHOCK PROTEINS; MOLECULAR STRUCTURE; PROTEIN BINDING; PROTEIN CONFORMATION;

EID: 80255131088 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.09.096 Document Type: Article

Times cited : (17)

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