SCOPUS 정보 검색 플랫폼

Volumn 17, Issue 9, 2011, Pages 2297-2303

Biological and docking studies of topoisomerase IV inhibition by thiosemicarbazides

(8) Siwek, Agata a Sta̧czek, Paweł b Wujec, Monika a Stefańska, Joanna c Kosikowska, Urszula a Malm, Anna a Jankowski, Stefan d Paneth, Piotr d

a MEDICAL UNIVERSITY OF LUBLIN (Poland)

b UNIVERSITY OF LODZ (Poland)

c MEDICAL UNIVERSITY OF WARSAW (Poland)

d LODZ UNIVERSITY OF TECHNOLOGY (Poland)

Author keywords

Antibacterial activity; Bacterial topoisomerase IV; Docking; Enzyme inhibitor; Thiosemicarbazide derivative

Indexed keywords

1,4 DIBENZOYLTHIOSEMICARBAZIDE; 4 BENZOYL 1 (4 METHYL IMIDAZOL 5 YL)CARBONYLTHIOSEMICARBAZIDE; 4 BENZOYL 1 (INDOL 2 YL)CARBONYLTHIOSEMICARBAZIDE; ADENOSINE TRIPHOSPHATE; ANTIBIOTIC AGENT; CEFUROXIME; CIPROFLOXACIN; DNA TOPOISOMERASE (ATP HYDROLYSING); DNA TOPOISOMERASE INHIBITOR; DNA TOPOISOMERASE IV; THIOSEMICARBAZIDE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; BACILLUS CEREUS; BACILLUS SUBTILIS; BACTERIAL GROWTH; BACTERIAL STRAIN; BORDETELLA BRONCHISEPTICA; CONFERENCE PAPER; CONTROLLED STUDY; DNA SUPERCOILING; DRUG BINDING SITE; DRUG POTENCY; DRUG SYNTHESIS; DRUG TARGETING; ENZYME INHIBITION; ESCHERICHIA COLI; IC 50; KLEBSIELLA PNEUMONIAE; MICROCOCCUS LUTEUS; MINIMUM INHIBITORY CONCENTRATION; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; PROTEUS MIRABILIS; PROTEUS VULGARIS; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS; STREPTOCOCCUS PNEUMONIAE;

ANTI-BACTERIAL AGENTS; BACILLUS CEREUS; BACILLUS SUBTILIS; BINDING SITES; COMPUTER SIMULATION; DISK DIFFUSION ANTIMICROBIAL TESTS; DNA TOPOISOMERASE IV; ENZYME ASSAYS; IMIDAZOLES; MICROBIAL SENSITIVITY TESTS; MICROCOCCUS LUTEUS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PROTEIN BINDING; SEMICARBAZIDES; STAPHYLOCOCCUS AUREUS; STAPHYLOCOCCUS EPIDERMIDIS;

BACTERIA (MICROORGANISMS); POSIBACTERIA;

EID: 80054879796 PISSN: 16102940 EISSN: 09485023 Source Type: Journal
DOI: 10.1007/s00894-010-0889-z Document Type: Conference Paper

Times cited : (33)

References (24)

1
- 54849420897
- 10.1016/j.coph.2008.04.009 1:CAS:528:DC%2BD1cXhtlaqsLvI
- BJ Bradbury MJ Pucci 2008 Curr Opin Pharmacol 8 574 581 10.1016/j.coph.2008.04.009 1:CAS:528:DC%2BD1cXhtlaqsLvI
- (2008) Curr Opin Pharmacol , vol.8 , pp. 574-581
- Bradbury, B.J.¹ Pucci, M.J.²

2
- 34948830988
- Discovery of novel DNA gyrase inhibitors by high-throughput virtual screening
- DOI 10.1128/AAC.00392-07
- DA Ostrov JA Hernández Prada PE Corsino KA Finton N Le TC Rowe 2007 Antimicrob Agents Chemother 51 3688 3698 10.1128/AAC.00392-07 1:CAS:528:DC%2BD2sXhtFGhtbnI (Pubitemid 47519360)
- (2007) Antimicrobial Agents and Chemotherapy , vol.51 , Issue.10 , pp. 3688-3698
- Ostrov, D.A.¹ Hernandez Prada, J.A.² Corsino, P.E.³ Finton, K.A.⁴ Le, N.⁵ Rowe, T.C.⁶

3
- 26844521517
- In silico fragment-based discovery of indolin-2-one analogues as potent DNA gyrase inhibitors
- DOI 10.1016/j.bmcl.2005.08.068, PII S0960894X05010991
- M Oblak SG Grdadolnik M Kotnik R Jerala M Filipič T Šolmajer 2005 Bioorg Med Chem Lett 15 5207 5210 10.1016/j.bmcl.2005.08. 068 1:CAS:528:DC%2BD2MXhtFCntrbJ (Pubitemid 41463648)
- (2005) Bioorganic and Medicinal Chemistry Letters , vol.15 , Issue.23 , pp. 5207-5210
- Oblak, M.¹ Grdadolnik, S.G.² Kotnik, M.³ Jerala, R.⁴ Filipic, M.⁵ Solmajer, T.⁶

4
- 33748925426
- Biophysical characterization of an indolinone inhibitor in the ATP-binding site of DNA gyrase
- DOI 10.1016/j.bbrc.2006.08.172, PII S0006291X06019437
- M Oblak S Golič Grdadolnik M Kotnik A Poterszman RA Atkinson H Nierengarten D Desplancq D Moras T Solmajer 2006 Biochem Biophys Res Commun 349 1206 1213 10.1016/j.bbrc.2006.08.172 1:CAS:528:DC%2BD28XpvFGjs78%3D (Pubitemid 44430194)
- (2006) Biochemical and Biophysical Research Communications , vol.349 , Issue.4 , pp. 1206-1213
- Oblak, M.¹ Grdadolnik, S.G.² Kotnik, M.³ Poterszman, A.⁴ Atkinson, R.A.⁵ Nierengarten, H.⁶ Desplancq, D.⁷ Moras, D.⁸ Solmajer, T.⁹

5
- 50649101663
- 10.1017/S003358350800468X 1:CAS:528:DC%2BD1cXhtVGnsbfE
- AJ Schoeffler JM Berger 2008 Q Rev Biophys 41 41 101 10.1017/ S003358350800468X 1:CAS:528:DC%2BD1cXhtVGnsbfE
- (2008) Q Rev Biophys , vol.41 , pp. 41-101
- Schoeffler, A.J.¹ Berger, J.M.²

6
- 37549023863
- 10.1038/nature06396 1:CAS:528:DC%2BD2sXhsVGjsL%2FN
- KC Dong JM Berger 2007 Nature 450 1201 1205 10.1038/nature06396 1:CAS:528:DC%2BD2sXhsVGjsL%2FN
- (2007) Nature , vol.450 , pp. 1201-1205
- Dong, K.C.¹ Berger, J.M.²

7
- 0036724716
- Fluoroquinolone resistance among Gram-positive cocci
- DOI 10.1016/S1473-3099(02)00369-9
- DC Hooper 2002 Lancet Infect Dis 2 530 538 10.1016/S1473-3099(02)00369-9 1:CAS:528:DC%2BD38XnsFOjtbg%3D (Pubitemid 34966356)
- (2002) Lancet Infectious Diseases , vol.2 , Issue.9 , pp. 530-538
- Hooper, D.C.¹

8
- 1842830032
- A multidrug efflux pump inhibitor reduces Fluoroquinolone resistance in Pseudomonas aeruginosa isolates
- DOI 10.1159/000077280
- AY Coban B Ekinci B Durupinar 2004 Chemotherapy 50 22 26 10.1159/000077280 (Pubitemid 38490195)
- (2004) Chemotherapy , vol.50 , Issue.1 , pp. 22-26
- Coban, A.Y.¹ Ekinci, B.² Durupinar, B.³

9
- 2142814314
- Crystal Structures of Escherichia coli Topoisomerase IV ParE Subunit (24 and 43 Kilodaltons): A Single Residue Dictates Differences in Novobiocin Potency against Topoisomerase IV and DNA Gyrase
- DOI 10.1128/AAC.48.5.1856-1864.2004
- S Bellon JD Parsons Y Wei K Hayakawa LL Swenson PS Charifson JA Lippke R Aldape ChH Gross 2004 Antimicrob Agents Chemother 48 1856 1864 10.1128/AAC.48.5.1856-1864.2004 1:CAS:528:DC%2BD2cXjslCksLk%3D (Pubitemid 38544398)
- (2004) Antimicrobial Agents and Chemotherapy , vol.48 , Issue.5 , pp. 1856-1864
- Bellon, S.¹ Parsons, J.D.² Wei, Y.³ Hayakawa, K.⁴ Swenson, L.L.⁵ Charifson, P.S.⁶ Lippke, J.A.⁷ Aldape, R.⁸ Gross, C.H.⁹

10
- 4644248307
- Synthesis and antibacterial activity of novel and potent DNA gyrase inhibitors with azole ring
- DOI 10.1016/j.bmc.2004.08.010, PII S0968089604006133
- A Tanitame Y Oyamada K Ofuji M Fujimoto K Suzuki T Ueda H Terauchi M Kawasaki K Nagai M Wachi J-i Yamagishi 2004 Bioorg Med Chem 12 5515 5524 10.1016/j.bmc.2004.08.010 1:CAS:528:DC%2BD2cXotF2itLo%3D (Pubitemid 39304051)
- (2004) Bioorganic and Medicinal Chemistry , vol.12 , Issue.21 , pp. 5515-5524
- Tanitame, A.¹ Oyamada, Y.² Ofuji, K.³ Fujimoto, M.⁴ Suzuki, K.⁵ Ueda, T.⁶ Terauchi, H.⁷ Kawasaki, M.⁸ Nagai, K.⁹ Wachi, M.¹⁰ Yamagishi, J.-I.¹¹

11
- 34248232578
- 10.1007/s00706-007-0600-y 1:CAS:528:DC%2BD2sXkvF2mtLs%3D
- S Cunha FC Macedo Jr GAN Costa MT Rodrigues Jr RBV Verde LC de Souza Neta I Vencato C Lariucci FP Sá 2007 Monatsh Chem 138 511 516 10.1007/s00706-007-0600-y 1:CAS:528:DC%2BD2sXkvF2mtLs%3D
- (2007) Monatsh Chem , vol.138 , pp. 511-516
- Cunha, S.¹ Macedo Jr., F.C.² Costa, G.A.N.³ Rodrigues Jr., M.T.⁴ Verde, R.B.V.⁵ De Souza Neta, L.C.⁶ Vencato, I.⁷ Lariucci, C.⁸ Sá, F.P.⁹

12
- 38649109136
- 10.1016/j.carres.2007.11.024 1:CAS:528:DC%2BD1cXhsFWqur4%3D
- Z Zhong R Xing S Liu L Wang S Cai P Li 2008 Carbohydr Res 343 566 570 10.1016/j.carres.2007.11.024 1:CAS:528:DC%2BD1cXhsFWqur4%3D
- (2008) Carbohydr Res , vol.343 , pp. 566-570
- Zhong, Z.¹ Xing, R.² Liu, S.³ Wang, L.⁴ Cai, S.⁵ Li, P.⁶

13
- 80255138917
- Polish Patent Aplication No. P-390774
- Siwek A, Paneth P, Sta̧czek P, Stefańska J (2010) Polish Patent Aplication No. P-390774
- (2010)
- Siwek, A.P.¹

14
- 72149099079
- 10.1016/j.ejmech.2009.10.016 1:CAS:528:DC%2BD1MXhsF2ju7nK
- NAH Farag W El-Tayeb 2010 Eur J Med Chem 45 317 325 10.1016/j.ejmech. 2009.10.016 1:CAS:528:DC%2BD1MXhsF2ju7nK
- (2010) Eur J Med Chem , vol.45 , pp. 317-325
- Farag, N.A.H.¹ El-Tayeb, W.²

15
- 33646696219
- Clinical and Laboratory Standards Institute. Clinical and Laboratory Standards Institute Wayne, PA
- Clinical and Laboratory Standards Institute (2006) Performance standards for antimicrobial disc susceptibility tests; document M2-A9. Clinical and Laboratory Standards Institute, Wayne, PA
- (2006) Performance Standards for Antimicrobial Disc Susceptibility Tests; Document M2-A9

16
- 33646693907
- Clinical and Laboratory Standards Institute. Clinical and Laboratory Standards Institute Wayne, PA
- Clinical and Laboratory Standards Institute (2006) Methods for dilution antimicrobial susceptibility tests for bacteria that grow aerobically; document M7-A7. Clinical and Laboratory Standards Institute, Wayne, PA
- (2006) Methods for Dilution Antimicrobial Susceptibility Tests for Bacteria That Grow Aerobically; Document M7-A7

17
- 11644261806
- 10.1002/(SI CI)1096-98 7X(19981 115)19:14<163 9::AID-JC C10>3.0.CO;2-B 1:CAS:528:Dya K1cXntFem ur4%3D
- GM Morris DS Goodsell RS Halliday R Huey WE Hart RK Belew AJ Olson 1998 J Comput Chem 19 1639 166 10.1002/(SICI)1096-987X(19981115)19:14<1639::AID- JCC10>3.0.CO;2-B 1:CAS:528:DyaK1cXntFemur4%3D
- (1998) J Comput Chem , vol.19 , pp. 1639-166
- Morris, G.M.¹ Goodsell, D.S.² Halliday, R.S.³ Huey, R.⁴ Hart, W.E.⁵ Belew, R.K.⁶ Olson, A.J.⁷

18
- 0033545622
- A general and fast scoring function for protein-ligand interactions: A simplified potential approach
- DOI 10.1021/jm980536j
- I Muegge Y Martin 1999 J Med Chem 42 791 804 10.1021/jm980536j 1:CAS:528:DyaK1MXht1aksrk%3D (Pubitemid 29136170)
- (1999) Journal of Medicinal Chemistry , vol.42 , Issue.5 , pp. 791-804
- Muegge, I.¹ Martin, Y.C.²

19
- 0029011701
- 10.1021/ja00124a002 1:CAS:528:DyaK2MXlsFertrc%3D
- WD Cornell P Cieplak CI Bayly IR Gould KM Merz Jr DM Ferguson DC Spellmeyer T Fox JW Caldwell PA Kollman 1995 J Am Chem Soc 117 5179 5197 10.1021/ja00124a002 1:CAS:528:DyaK2MXlsFertrc%3D
- (1995) J Am Chem Soc , vol.117 , pp. 5179-5197
- Cornell, W.D.¹ Cieplak, P.² Bayly, C.I.³ Gould, I.R.⁴ Merz Jr., K.M.⁵ Ferguson, D.M.⁶ Spellmeyer, D.C.⁷ Fox, T.⁸ Caldwell, J.W.⁹ Kollman, P.A.¹⁰

20
- 38849090006
- Sulfonamide-1,2,4-triazole derivatives as antifungal and antibacterial agents: Synthesis, biological evaluation, lipophilicity, and conformational studies
- DOI 10.1016/j.bmc.2007.10.082, PII S0968089607009509
- IR Ezabadi C Camoutsis P Zoumpoulakis A Geronikaki M Soković J Glamoćilija A Ćirić 2008 Bioorg Med Chem 16 1150 1161 10.1016/j.bmc.2007.10.082 1:CAS:528:DC%2BD1cXhvVWhtbc%3D (Pubitemid 351193036)
- (2008) Bioorganic and Medicinal Chemistry , vol.16 , Issue.3 , pp. 1150-1161
- Ezabadi, I.R.¹ Camoutsis, C.² Zoumpoulakis, P.³ Geronikaki, A.⁴ Sokovic, M.⁵ Glamocilija, J.⁶ Ciric, A.⁷

21
- 42149101677
- Synthesis and antioxidant properties of novel N-methyl-1,3,4-thiadiazol- 2-amine and 4-methyl-2H-1,2,4-triazole-3(4H)-thione derivatives of benzimidazole class
- DOI 10.1016/j.bmc.2008.02.077, PII S0968089608001995
- C Kuş G Ayhan-KIlcIgil S Özbey FB Kaynak M Kaya T Çoban B Can-Eke 2008 Bioorg Med Chem 16 4294 4303 10.1016/j.bmc.2008.02. 077 (Pubitemid 351539047)
- (2008) Bioorganic and Medicinal Chemistry , vol.16 , Issue.8 , pp. 4294-4303
- Kus, C.¹ Ayhan-Kilcigil, G.² Ozbey, S.³ Kaynak, F.B.⁴ Kaya, M.⁵ Coban, T.⁶ Can-Eke, B.⁷

22
- 40949124294
- Synthesis and antimicrobial activity of new 1,2,4-triazole and 1,3,4-thiadiazole derivatives
- DOI 10.1080/14756360701408697, PII 791443763
- T Önkol DS Doǧruer L Uzun S Adak S Özkan MFJ Şahin 2008 J Enzym Inhib Med Chem 23 277 284 10.1080/14756360701408697 (Pubitemid 351404849)
- (2008) Journal of Enzyme Inhibition and Medicinal Chemistry , vol.23 , Issue.2 , pp. 277-284
- Onkol, T.¹ Dogruer, D.² Uzun, L.³ Adak, S.⁴ Ozkan, S.⁵ Sahin, M.F.⁶

23
- 33847358707
- 10.1080/10426500600892776 1:CAS:528:DC%2BD2sXhtFWisbo%3D
- HZ Shams RM Mohareb MH Helal AE Mahmoud 2007 Phosphorus Sulfur Silicon Relat Elem 182 237 263 10.1080/10426500600892776 1:CAS:528:DC%2BD2sXhtFWisbo%3D
- (2007) Phosphorus Sulfur Silicon Relat Elem , vol.182 , pp. 237-263
- Shams, H.Z.¹ Mohareb, R.M.² Helal, M.H.³ Mahmoud, A.E.⁴

24
- 30444434889
- Isothiazolopyridones: Synthesis, structure, and biological activity of a new class of antibacterial agents
- DOI 10.1021/jm051066d
- JA Wiles A Hashimoto JA Thanassi J Cheng ChD Incarvito M Deshpande MJ Pucci BJ Bradbury 2006 J Med Chem 49 39 42 10.1021/jm051066d 1:CAS:528:DC%2BD2MXht12rtbjP (Pubitemid 43077320)
- (2006) Journal of Medicinal Chemistry , vol.49 , Issue.1 , pp. 39-42
- Wiles, J.A.¹ Hashimoto, A.² Thanassi, J.A.³ Cheng, J.⁴ Incarvito, C.D.⁵ Deshpande, M.⁶ Pucci, M.J.⁷ Bradbury, B.J.⁸

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.