ATP competitive protein kinase C inhibitors demonstrate distinct state-dependent inhibition

PLoS ONE

Volumn 6, Issue 10, 2011, Pages

  Smith, Ida M ^a   Hoshi, Naoto ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BISINDOLYLMALEIMIDE; BISINDOLYLMALEIMIDE I; BISINDOLYLMALEIMIDE IV; K 252C; PHORBOL DIBUTYRATE; PROTEIN KINASE C; STAUROSPORINE; STAUROSPORINE DERIVATIVE; UNCLASSIFIED DRUG; ADENOSINE TRIPHOSPHATE; INDOLE DERIVATIVE; MALEIMIDE DERIVATIVE; PROTEIN KINASE INHIBITOR;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG DETERMINATION; DRUG INHIBITION; DRUG STRUCTURE; ENZYME ACTIVATION; ENZYME INHIBITION; ENZYME REPRESSION; HUMAN; HUMAN CELL; PROTEIN CONFORMATION; PROTEIN INTERACTION; ANIMAL; BINDING COMPETITION; DRUG ANTAGONISM; KINETICS; METABOLISM; PROTEIN STABILITY;

ADENOSINE TRIPHOSPHATE; ANIMALS; BINDING, COMPETITIVE; HUMANS; INDOLES; KINETICS; MALEIMIDES; PROTEIN CONFORMATION; PROTEIN KINASE C; PROTEIN KINASE INHIBITORS; PROTEIN STABILITY;

EID: 80054767649     PISSN: None     EISSN: 19326203     Source Type: Journal    
DOI: 10.1371/journal.pone.0026338     Document Type: Article

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