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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 22, 2011, Pages 6705-6708

Identification of a novel RAMP-independent CGRP receptor antagonist

(10) Zartman, C Blair a Bell, Ian M a Gallicchio, Steven N a Graham, Samuel L a Kane, Stefanie A a Mallee, John J a Rutledge, Ruth Z a Salvatore, Christopher A a Vacca, Joseph P a Williams, Theresa M a

a MERCK RESEARCH LABORATORIES (United States)

Author keywords

CGRP; HIV integrase; Hydroxypyridine; RAMP independent

Indexed keywords

CALCITONIN GENE RELATED PEPTIDE RECEPTOR; DIVALENT CATION; INTEGRASE INHIBITOR; PYRIDINOL; RECEPTOR ACTIVITY MODIFYING PROTEIN;

ARTICLE; BINDING SITE; DOG; DRUG BIOAVAILABILITY; DRUG IDENTIFICATION; MOLECULAR WEIGHT; NONHUMAN; RAT; RECEPTOR BINDING;

ANIMALS; CELL LINE; DOGS; HIV; HIV INTEGRASE INHIBITORS; HUMANS; PROTEIN BINDING; PYRIDINES; RATS; RECEPTOR ACTIVITY-MODIFYING PROTEINS; RECEPTORS, CALCITONIN GENE-RELATED PEPTIDE;

CANIS FAMILIARIS; RATTUS;

EID: 80054745704 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.09.056 Document Type: Article

Times cited : (9)

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