메뉴 건너뛰기




Volumn 38, Issue 7, 2011, Pages 1035-1041

Biodistribution and human dosimetry of enantiomer-1 of the synthetic leucine analog anti-1-amino-2-fluorocyclopentyl-1-carboxylic acid

Author keywords

Amino acid; Anti 2 18F FACPC; Anti 3 18F FACBC; Biodistribution; Dosimetry; FACBC; FACPC; Positron emission tomography

Indexed keywords

1 AMINO 2 FLUOROCYCLOPENTYL 1 CARBOXYLIC ACID F 18; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

EID: 80053612717     PISSN: 09698051     EISSN: 18729614     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2011.03.007     Document Type: Article
Times cited : (2)

References (33)
  • 1
    • 0000067486 scopus 로고
    • The uptake of a variety of amino acids into nuclear proteins of tumors and other tissues
    • Busch H., Davis J.R., Honig G.R., Anderson D.C., Nair P.V., Nyhan W.L. The uptake of a variety of amino acids into nuclear proteins of tumors and other tissues. Cancer Res 1959, 19:1030-1039.
    • (1959) Cancer Res , vol.19 , pp. 1030-1039
    • Busch, H.1    Davis, J.R.2    Honig, G.R.3    Anderson, D.C.4    Nair, P.V.5    Nyhan, W.L.6
  • 2
    • 0015525722 scopus 로고
    • Sugar and amino acid transport by cells in culture - differences between normal and malignant cells
    • Isselbacher K.J. Sugar and amino acid transport by cells in culture - differences between normal and malignant cells. N Engl J Med 1972, 286(17):929-933.
    • (1972) N Engl J Med , vol.286 , Issue.17 , pp. 929-933
    • Isselbacher, K.J.1
  • 3
    • 0025095302 scopus 로고
    • Role of amino acid transport and countertransport in nutrition and metabolism
    • Christensen H.N. Role of amino acid transport and countertransport in nutrition and metabolism. Physiol Rev 1990, 70(1):43-77.
    • (1990) Physiol Rev , vol.70 , Issue.1 , pp. 43-77
    • Christensen, H.N.1
  • 4
    • 33745616802 scopus 로고    scopus 로고
    • Differential Expression and functional characterization of system l amino acid transporters in human normal osteoblast cells and osteogenic sarcoma cells
    • Kim S.G., Kim H.H., Kim H.K., et al. Differential Expression and functional characterization of system l amino acid transporters in human normal osteoblast cells and osteogenic sarcoma cells. Anticancer Res 2006, 26(3A):1989-1996.
    • (2006) Anticancer Res , vol.26 , Issue.3 A , pp. 1989-1996
    • Kim, S.G.1    Kim, H.H.2    Kim, H.K.3
  • 5
    • 20044374008 scopus 로고    scopus 로고
    • Expression of L-type amino acid transporter 1 (LAT1) in esophageal carcinoma
    • Kobayashi H., Ishii Y., Takayama T. Expression of L-type amino acid transporter 1 (LAT1) in esophageal carcinoma. J Surg Oncol 2005, 90(4):233-238.
    • (2005) J Surg Oncol , vol.90 , Issue.4 , pp. 233-238
    • Kobayashi, H.1    Ishii, Y.2    Takayama, T.3
  • 6
    • 12144287436 scopus 로고    scopus 로고
    • L-type amino acid transporter-1 overexpression and melphalan sensitivity in Barrett's adenocarcinoma
    • Lin J., Raoof D.A., Thomas D.G., et al. L-type amino acid transporter-1 overexpression and melphalan sensitivity in Barrett's adenocarcinoma. Neoplasia 2004, 6(1):74-84.
    • (2004) Neoplasia , vol.6 , Issue.1 , pp. 74-84
    • Lin, J.1    Raoof, D.A.2    Thomas, D.G.3
  • 7
    • 4243389920 scopus 로고    scopus 로고
    • Human L-type amino acid transporter 1 (LAT1): characterization of function and expression in tumor cell lines
    • Yanagida O., Kanai Y., Chairoungdua A., et al. Human L-type amino acid transporter 1 (LAT1): characterization of function and expression in tumor cell lines. Biochim Biophys Acta 2001, 1514(2):291-302.
    • (2001) Biochim Biophys Acta , vol.1514 , Issue.2 , pp. 291-302
    • Yanagida, O.1    Kanai, Y.2    Chairoungdua, A.3
  • 8
    • 33646540633 scopus 로고    scopus 로고
    • L-type amino acid transporter 1 as a potential molecular target in human astrocytic tumors
    • Nawashiro H., Otani N., Shinomiya N., et al. L-type amino acid transporter 1 as a potential molecular target in human astrocytic tumors. Int J Cancer 2006, 119(3):484-492.
    • (2006) Int J Cancer , vol.119 , Issue.3 , pp. 484-492
    • Nawashiro, H.1    Otani, N.2    Shinomiya, N.3
  • 9
    • 0032869487 scopus 로고    scopus 로고
    • Investigation of transport mechanism and uptake kinetics of O-(2-[18F]fluoroethyl)-l-tyrosine in vitro and in vivo
    • Heiss P., Mayer S., Herz M., Wester H.J., Schwaiger M., Senekowitsch-Schmidtke R. Investigation of transport mechanism and uptake kinetics of O-(2-[18F]fluoroethyl)-l-tyrosine in vitro and in vivo. J Nucl Med 1999, 40(8):1367-1373.
    • (1999) J Nucl Med , vol.40 , Issue.8 , pp. 1367-1373
    • Heiss, P.1    Mayer, S.2    Herz, M.3    Wester, H.J.4    Schwaiger, M.5    Senekowitsch-Schmidtke, R.6
  • 10
    • 0025858860 scopus 로고
    • Increased amino acid transport into brain tumors measured by PET of L-(2-18F)fluorotyrosine
    • Wienhard K., Herholz K., Coenen H.H., et al. Increased amino acid transport into brain tumors measured by PET of L-(2-18F)fluorotyrosine. J Nucl Med 1991, 32(7):1338-1346.
    • (1991) J Nucl Med , vol.32 , Issue.7 , pp. 1338-1346
    • Wienhard, K.1    Herholz, K.2    Coenen, H.H.3
  • 11
    • 52549133776 scopus 로고    scopus 로고
    • Non-natural amino acids for tumor imaging using positron emission tomography and single photon emission computed tomography
    • McConathy J., Goodman M.M. Non-natural amino acids for tumor imaging using positron emission tomography and single photon emission computed tomography. Cancer Metastasis Rev 2008, 27(4):555-573.
    • (2008) Cancer Metastasis Rev , vol.27 , Issue.4 , pp. 555-573
    • McConathy, J.1    Goodman, M.M.2
  • 12
    • 0018651869 scopus 로고
    • 1-aminocyclobutane[11C]carboxylic acid, a potential tumor-seeking agent
    • Washburn L.C., Sun T.T., Byrd B., Hayes R.L., Butler T.A. 1-aminocyclobutane[11C]carboxylic acid, a potential tumor-seeking agent. J Nucl Med 1979, 20(10):1055-1061.
    • (1979) J Nucl Med , vol.20 , Issue.10 , pp. 1055-1061
    • Washburn, L.C.1    Sun, T.T.2    Byrd, B.3    Hayes, R.L.4    Butler, T.A.5
  • 13
    • 0032588608 scopus 로고    scopus 로고
    • Synthesis and evaluation of [18F]1-amino-3-fluorocyclobutane-1-carboxylic acid to image brain tumors
    • Shoup T.M., Olson J., Hoffman J.M., et al. Synthesis and evaluation of [18F]1-amino-3-fluorocyclobutane-1-carboxylic acid to image brain tumors. J Nucl Med 1999, 40(2):331-338.
    • (1999) J Nucl Med , vol.40 , Issue.2 , pp. 331-338
    • Shoup, T.M.1    Olson, J.2    Hoffman, J.M.3
  • 14
    • 33847291423 scopus 로고    scopus 로고
    • Initial experience with the radiotracer anti-1-amino-3-18F-fluorocyclobutane-1-carboxylic acid with PET/CT in prostate carcinoma
    • Schuster D.M., Votaw J.R., Nieh P.T., et al. Initial experience with the radiotracer anti-1-amino-3-18F-fluorocyclobutane-1-carboxylic acid with PET/CT in prostate carcinoma. J Nucl Med 2007, 48(1):56-63.
    • (2007) J Nucl Med , vol.48 , Issue.1 , pp. 56-63
    • Schuster, D.M.1    Votaw, J.R.2    Nieh, P.T.3
  • 15
    • 33847309910 scopus 로고    scopus 로고
    • A preliminary study of anti-1-amino-3-18F-fluorocyclobutyl-1-carboxylic acid for the detection of prostate cancer
    • Oka S., Hattori R., Kurosaki F., et al. A preliminary study of anti-1-amino-3-18F-fluorocyclobutyl-1-carboxylic acid for the detection of prostate cancer. J Nucl Med 2007, 48(1):46-55.
    • (2007) J Nucl Med , vol.48 , Issue.1 , pp. 46-55
    • Oka, S.1    Hattori, R.2    Kurosaki, F.3
  • 16
    • 80053603496 scopus 로고    scopus 로고
    • Characterization of the two enantiomers of anti-18F-FACPC as PET tumor agents
    • 2_MeetingAbstracts
    • Jarkas N., Voll R., Camp V., Zhang Z., Goodman M. Characterization of the two enantiomers of anti-18F-FACPC as PET tumor agents. J Nucl Med Meeting Abstracts 2010, 51:1516. 2_MeetingAbstracts.
    • (2010) J Nucl Med Meeting Abstracts , vol.51 , pp. 1516
    • Jarkas, N.1    Voll, R.2    Camp, V.3    Zhang, Z.4    Goodman, M.5
  • 17
    • 84855694794 scopus 로고    scopus 로고
    • Pilot evaluation of 1-amino-2-[18F] fluorocyclopentane-1-carboxylic acid (anti-2-[18F] FACPC) PET-CT in recurrent prostate carcinoma
    • 2_MeetingAbstracts
    • Savir-Baruch B., Schuster D., Jarkas N., et al. Pilot evaluation of 1-amino-2-[18F] fluorocyclopentane-1-carboxylic acid (anti-2-[18F] FACPC) PET-CT in recurrent prostate carcinoma. J Nucl Med Meeting Abstracts 2010, 51:1266. 2_MeetingAbstracts.
    • (2010) J Nucl Med Meeting Abstracts , vol.51 , pp. 1266
    • Savir-Baruch, B.1    Schuster, D.2    Jarkas, N.3
  • 18
    • 77956754523 scopus 로고    scopus 로고
    • (R,S)-Anti-1-amino-2-[18F]fluorocyclopentyl-1-carboxylic acid: synthesis from racemic 2-benzyloxycyclopentanone and biological evaluation for brain tumor imaging with positron emission tomography
    • Jarkas N., Voll R.J., Williams L., Camp V.M., Goodman M.M. (R,S)-Anti-1-amino-2-[18F]fluorocyclopentyl-1-carboxylic acid: synthesis from racemic 2-benzyloxycyclopentanone and biological evaluation for brain tumor imaging with positron emission tomography. J Med Chem 2010, 53(18):6603-6607.
    • (2010) J Med Chem , vol.53 , Issue.18 , pp. 6603-6607
    • Jarkas, N.1    Voll, R.J.2    Williams, L.3    Camp, V.M.4    Goodman, M.M.5
  • 19
    • 0038241522 scopus 로고    scopus 로고
    • Improved synthesis of anti-[18F]FACBC: improved preparation of labeling precursor and automated radiosynthesis
    • McConathy J., Voll R.J., Yu W., Crowe R.J., Goodman M.M. Improved synthesis of anti-[18F]FACBC: improved preparation of labeling precursor and automated radiosynthesis. Appl Radiat Isot 2003, 58(6):657-666.
    • (2003) Appl Radiat Isot , vol.58 , Issue.6 , pp. 657-666
    • McConathy, J.1    Voll, R.J.2    Yu, W.3    Crowe, R.J.4    Goodman, M.M.5
  • 20
    • 77249087166 scopus 로고    scopus 로고
    • Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain tumors
    • Yu W., McConathy J., Williams L., et al. Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain tumors. J Med Chem 2010, 53(2):876-886.
    • (2010) J Med Chem , vol.53 , Issue.2 , pp. 876-886
    • Yu, W.1    McConathy, J.2    Williams, L.3
  • 21
    • 16544364015 scopus 로고    scopus 로고
    • Performance characteristics of a newly developed PET/CT scanner using NEMA standards in 2D and 3D modes
    • Mawlawi O., Podoloff D.A., Kohlmyer S., et al. Performance characteristics of a newly developed PET/CT scanner using NEMA standards in 2D and 3D modes. J Nucl Med 2004, 45(10):1734-1742.
    • (2004) J Nucl Med , vol.45 , Issue.10 , pp. 1734-1742
    • Mawlawi, O.1    Podoloff, D.A.2    Kohlmyer, S.3
  • 23
    • 0030002992 scopus 로고    scopus 로고
    • MIRDOSE: personal computer software for internal dose assessment in nuclear medicine
    • Stabin M.G. MIRDOSE: personal computer software for internal dose assessment in nuclear medicine. J Nucl Med 1996, 37(3):538-546.
    • (1996) J Nucl Med , vol.37 , Issue.3 , pp. 538-546
    • Stabin, M.G.1
  • 24
    • 61349145115 scopus 로고    scopus 로고
    • Stereoselective synthesis and biological evaluation of syn-1-amino-3-[18F]fluorocyclobutyl-1-carboxylic acid as a potential positron emission tomography brain tumor imaging agent
    • Yu W., Williams L., Camp V.M., Malveaux E., Olson J.J., Goodman M.M. Stereoselective synthesis and biological evaluation of syn-1-amino-3-[18F]fluorocyclobutyl-1-carboxylic acid as a potential positron emission tomography brain tumor imaging agent. Bioorg Med Chem 2009, 17(5):1982-1990.
    • (2009) Bioorg Med Chem , vol.17 , Issue.5 , pp. 1982-1990
    • Yu, W.1    Williams, L.2    Camp, V.M.3    Malveaux, E.4    Olson, J.J.5    Goodman, M.M.6
  • 25
    • 0037161594 scopus 로고    scopus 로고
    • Synthesis of syn- and anti-1-amino-3-[18F]fluoromethyl-cyclobutane-1-carboxylic acid (FMACBC), potential pet ligands for tumor detection
    • Martarello L., McConathy J., Camp V.M., et al. Synthesis of syn- and anti-1-amino-3-[18F]fluoromethyl-cyclobutane-1-carboxylic acid (FMACBC), potential pet ligands for tumor detection. J Med Chem 2002, 45(11):2250-2259.
    • (2002) J Med Chem , vol.45 , Issue.11 , pp. 2250-2259
    • Martarello, L.1    McConathy, J.2    Camp, V.M.3
  • 26
    • 0032921707 scopus 로고    scopus 로고
    • Synthesis and radiopharmacology of O-(2-[18F]fluoroethyl)-l-tyrosine for tumor imaging
    • Wester H.J., Herz M., Weber W., et al. Synthesis and radiopharmacology of O-(2-[18F]fluoroethyl)-l-tyrosine for tumor imaging. J Nucl Med 1999, 40(1):205-212.
    • (1999) J Nucl Med , vol.40 , Issue.1 , pp. 205-212
    • Wester, H.J.1    Herz, M.2    Weber, W.3
  • 27
    • 0038669336 scopus 로고    scopus 로고
    • Whole-body distribution and dosimetry of O-(2-[18F]fluoroethyl)-l-tyrosine
    • Pauleit D., Floeth F., Herzog H., et al. Whole-body distribution and dosimetry of O-(2-[18F]fluoroethyl)-l-tyrosine. Eur J Nucl Med Mol Imaging 2003, 30(4):519-524.
    • (2003) Eur J Nucl Med Mol Imaging , vol.30 , Issue.4 , pp. 519-524
    • Pauleit, D.1    Floeth, F.2    Herzog, H.3
  • 28
  • 29
    • 0031833854 scopus 로고    scopus 로고
    • Estimation of internal absorbed dose of l-[methyl-11C]methionine using whole-body positron emission tomography
    • Deloar H.M., Fujiwara T., Nakamura T., et al. Estimation of internal absorbed dose of l-[methyl-11C]methionine using whole-body positron emission tomography. Eur J Nucl Med 1998, 25(6):629-633.
    • (1998) Eur J Nucl Med , vol.25 , Issue.6 , pp. 629-633
    • Deloar, H.M.1    Fujiwara, T.2    Nakamura, T.3
  • 30
    • 34250323369 scopus 로고    scopus 로고
    • Biodistribution and radiation dosimetry of the synthetic nonmetabolized amino acid analogue anti-18F-FACBC in humans
    • Nye J.A., Schuster D.M., Yu W., Camp V.M., Goodman M.M., Votaw J.R. Biodistribution and radiation dosimetry of the synthetic nonmetabolized amino acid analogue anti-18F-FACBC in humans. J Nucl Med 2007, 48(6):1017-1020.
    • (2007) J Nucl Med , vol.48 , Issue.6 , pp. 1017-1020
    • Nye, J.A.1    Schuster, D.M.2    Yu, W.3    Camp, V.M.4    Goodman, M.M.5    Votaw, J.R.6
  • 31
    • 0035057021 scopus 로고    scopus 로고
    • Whole-body kinetics and dosimetry of cis-4-[18F]fluoro-l-proline
    • Börner A.R., Langen K.J., Herzog H., et al. Whole-body kinetics and dosimetry of cis-4-[18F]fluoro-l-proline. Nucl Med Biol 2001, 28(3):287-292.
    • (2001) Nucl Med Biol , vol.28 , Issue.3 , pp. 287-292
    • Börner, A.R.1    Langen, K.J.2    Herzog, H.3
  • 32
    • 80053613606 scopus 로고    scopus 로고
    • Pilot Evaluation of anti-1-amino-2-[18F]fluorocyclopentane-1-carboxylic acid (anti-2-[18F]FACPC) PET-CT in recurrent prostate carcinoma. Molecular Imaging and Biology. in press.
    • Savir-Baruch B, Schuster DM, Jarkas N, et al. Pilot Evaluation of anti-1-amino-2-[18F]fluorocyclopentane-1-carboxylic acid (anti-2-[18F]FACPC) PET-CT in recurrent prostate carcinoma. Molecular Imaging and Biology. in press.
    • Savir-Baruch, B.1    Schuster, D.M.2    Jarkas, N.3
  • 33
    • 78650679160 scopus 로고    scopus 로고
    • ICRP publication 103: recommendations of the ICRP†
    • Charles M.W. ICRP publication 103: recommendations of the ICRP†. Radiat Prot Dosimetry 2008, 129(4):500-507.
    • (2008) Radiat Prot Dosimetry , vol.129 , Issue.4 , pp. 500-507
    • Charles, M.W.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.