-
1
-
-
69349100378
-
Towards Physico-Relevant Dissolution Testing: The Importance of Solid-State Analysis in Dissolution
-
Aaltonen, J.; Rades, T. Towards Physico-Relevant Dissolution Testing: The Importance of Solid-State Analysis in Dissolution Dissolution Technol. 2009, 16, 47-54
-
(2009)
Dissolution Technol.
, vol.16
, pp. 47-54
-
-
Aaltonen, J.1
Rades, T.2
-
2
-
-
0030638567
-
Characteristics and significance of the amorphous state in pharmaceutical systems
-
Hancock, B. C.; Zografi, G. Characteristics and significance of the amorphous state in pharmaceutical systems J. Pharm. Sci. 1997, 86 (1) 1-12
-
(1997)
J. Pharm. Sci.
, vol.86
, Issue.1
, pp. 1-12
-
-
Hancock, B.C.1
Zografi, G.2
-
3
-
-
1142303337
-
What is the true solubility advantage for amorphous pharmaceuticals?
-
DOI 10.1023/A:1007516718048
-
Hancock, B. C.; Parks, M. What is the True Solubility Advantage for Amorphous Pharmaceuticals? Pharm. Res. 2000, 17 (4) 397-404 (Pubitemid 30395293)
-
(2000)
Pharmaceutical Research
, vol.17
, Issue.4
, pp. 397-404
-
-
Hancock, B.C.1
Parks, M.2
-
4
-
-
5144219871
-
Amorphous drug delivery systems: Molecular aspects, design, and performance
-
DOI 10.1615/CritRevTherDrugCarrierSyst.v21.i3.10
-
Kaushal, A. M.; Gupta, P.; Bansal, A. K. Amorphous drug delivery systems: Molecular aspects, design and performance Crit. Rev. Ther. Drug Carrier Syst. 2004, 21, 133-193 (Pubitemid 41647581)
-
(2004)
Critical Reviews in Therapeutic Drug Carrier Systems
, vol.21
, Issue.3
, pp. 133-193
-
-
Kaushal, A.M.1
Gupta, P.2
Bansal, A.K.3
-
5
-
-
0033663452
-
Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25
-
Van den Mooter, G.; Wuyts, M.; Blaton, N.; Busson, R.; Grobet, P.; Augustijns, P.; Kinget, R. Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25 Eur. J. Pharm. Sci. 2001, 12 (3) 261-269
-
(2001)
Eur. J. Pharm. Sci.
, vol.12
, Issue.3
, pp. 261-269
-
-
Van Den Mooter, G.1
Wuyts, M.2
Blaton, N.3
Busson, R.4
Grobet, P.5
Augustijns, P.6
Kinget, R.7
-
6
-
-
0035095847
-
Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with hydrophilic amorphous polymers
-
DOI 10.1211/0022357011775532
-
Forster, A.; Hempenstall, J.; Rades, T. Characterization of glass solutions of poorly water-soluble drugs produced by melt extrusion with hydrophilic amorphous polymers J. Pharm. Pharmacol. 2001, 53 (3) 303-315 (Pubitemid 32229189)
-
(2001)
Journal of Pharmacy and Pharmacology
, vol.53
, Issue.3
, pp. 303-315
-
-
Forster, A.1
Hempenstall, J.2
Rades, T.3
-
7
-
-
36549042006
-
Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs
-
DOI 10.1016/j.drudis.2007.09.005, PII S1359644607003753
-
Vasconcelos, T.; Sarmento, B.; Costa, P. Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs Drug Discovery Today 2007, 12 (23-24) 1068-1075 (Pubitemid 350186132)
-
(2007)
Drug Discovery Today
, vol.12
, Issue.23-24
, pp. 1068-1075
-
-
Vasconcelos, T.1
Sarmento, B.2
Costa, P.3
-
8
-
-
0032885450
-
Solid dispersion of poorly water-soluble drugs: Early promises, subsequent problems, and recent breakthroughs
-
Serajuddin, A. T. M. Solid dispersion of poorly water-soluble drugs: Early promises, subsequent problems, and recent breakthroughs J. Pharm. Sci. 1999, 88 (10) 1058-1066
-
(1999)
J. Pharm. Sci.
, vol.88
, Issue.10
, pp. 1058-1066
-
-
Serajuddin, A.T.M.1
-
9
-
-
61849159945
-
Design, Optimization, Preparation and Evaluation of Dispersion Granules of Valsartan and Formulation into Tablets
-
Shrivastava, A. R.; Ursekar, B.; Kapadia, C. J. Design, Optimization, Preparation and Evaluation of Dispersion Granules of Valsartan and Formulation into Tablets Curr. Drug Delivery 2009, 6, 28-37
-
(2009)
Curr. Drug Delivery
, vol.6
, pp. 28-37
-
-
Shrivastava, A.R.1
Ursekar, B.2
Kapadia, C.J.3
-
10
-
-
0019298791
-
Comparison of polyethylene glycol and polyoxyethylene stearate as excipients for solid dispersion systems of griseofulvin and tolbutamide II: Dissolution and solubility studies
-
DOI 10.1002/jps.2600691122
-
Kaur, R.; Grant, D. J. W.; Eaves, T. Comparison of polyethylene glycol and polyoxyethylene stearate as excipients for solid dispersion systems of griseofulvin and tolbutamide II J. Pharm. Sci. 1980, 69 (11) 1321-1326 (Pubitemid 11162729)
-
(1980)
Journal of Pharmaceutical Sciences
, vol.69
, Issue.11
, pp. 1321-1326
-
-
Kaur, R.1
Grant, D.J.W.2
Eaves, T.3
-
11
-
-
57349179076
-
Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation
-
Chieng, N.; Aaltonen, J.; Saville, D.; Rades, T. Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation Eur. J. Pharm. Biopharm. 2009, 71 (1) 47-54
-
(2009)
Eur. J. Pharm. Biopharm.
, vol.71
, Issue.1
, pp. 47-54
-
-
Chieng, N.1
Aaltonen, J.2
Saville, D.3
Rades, T.4
-
12
-
-
67349087395
-
Enhanced dissolution rate and synchronized release of drugs in binary systems through formulation: Amorphous naproxen-cimetidine mixtures prepared by mechanical activation
-
Allesa, M.; Chieng, N.; Rehder, S.; Rantanen, J.; Rades, T.; Aaltonen, J. Enhanced dissolution rate and synchronized release of drugs in binary systems through formulation: Amorphous naproxen-cimetidine mixtures prepared by mechanical activation J. Controlled Release 2009, 136 (1) 45-53
-
(2009)
J. Controlled Release
, vol.136
, Issue.1
, pp. 45-53
-
-
Allesa, M.1
Chieng, N.2
Rehder, S.3
Rantanen, J.4
Rades, T.5
Aaltonen, J.6
-
13
-
-
0034595299
-
Physicochemical properties of amorphous precipitates of cimetidine-indomethacin binary system
-
DOI 10.1016/S0939-6411(00)00060-6, PII S0939641100000606
-
Yamamura, S.; Gotoh, H.; Sakamoto, Y.; Momose, Y. Physicochemical properties of amorphous precipitates of cimetidine-indomethacin binary system Eur. J. Pharm. Biopharm. 2000, 49 (3) 259-265 (Pubitemid 30229875)
-
(2000)
European Journal of Pharmaceutics and Biopharmaceutics
, vol.49
, Issue.3
, pp. 259-265
-
-
Yamamura, S.1
Gotoh, H.2
Sakamoto, Y.3
Momose, Y.4
-
14
-
-
0037173525
-
Physicochemical properties of amorphous salt of cimetidine and diflunisal system
-
DOI 10.1016/S0378-5173(02)00195-3, PII S0378517302001953
-
Yamamura, S.; Gotoh, H.; Sakamoto, Y.; Momose, Y. Physicochemical properties of amorphous salt of cimetidine and diflunisal system Int. J. Pharm. 2002, 241 (2) 213-221 (Pubitemid 34718023)
-
(2002)
International Journal of Pharmaceutics
, vol.241
, Issue.2
, pp. 213-221
-
-
Yamamura, S.1
Gotoh, H.2
Sakamoto, Y.3
Momose, Y.4
-
16
-
-
0015124656
-
Pharmaceutical applications of solid dispersion systems
-
Chiou, W. L.; Riegelman, S. Pharmaceutical applications of solid dispersion systems J. Pharm. Sci. 1971, 60 (9) 1281-1302
-
(1971)
J. Pharm. Sci.
, vol.60
, Issue.9
, pp. 1281-1302
-
-
Chiou, W.L.1
Riegelman, S.2
-
17
-
-
33344473894
-
Characterization of the molecular distribution of drugs in glassy solid dispersions at the nano-meter scale, using differential scanning calorimetry and gravimetric water vapour sorption techniques
-
DOI 10.1016/j.ijpharm.2005.12.007, PII S0378517305008203
-
van Drooge, D. J.; Hinrichs, W. L. J.; Visser, M. R.; Frijlink, H. W. Characterization of the molecular distribution of drugs in glassy solid dispersions at the nano-meter scale, using differential scanning calorimetry and gravimetric water vapour sorption techniques Int. J. Pharm. 2006, 310 (1-2) 220-229 (Pubitemid 43287987)
-
(2006)
International Journal of Pharmaceutics
, vol.310
, Issue.1-2
, pp. 220-229
-
-
Van Drooge, D.J.1
Hinrichs, W.L.J.2
Visser, M.R.3
Frijlink, H.W.4
-
18
-
-
8844234199
-
Synthesis and characterization of layered double hydroxides (LDH) intercalated with non-steroidal anti-inflammatory drugs (NSAID)
-
del Arco, M.; Gutiérrez, S.; Martín, C.; Rives, V.; Rocha, J. Synthesis and characterization of layered double hydroxides (LDH) intercalated with non-steroidal anti-inflammatory drugs (NSAID) J. Solid State Chem. 2004, 177 (11) 3954-3962
-
(2004)
J. Solid State Chem.
, vol.177
, Issue.11
, pp. 3954-3962
-
-
Del Arco, M.1
Gutiérrez, S.2
Martín, C.3
Rives, V.4
Rocha, J.5
-
20
-
-
55649112715
-
Perspectives in the use of spectroscopy to characterise pharmaceutical solids
-
Aaltonen, J.; Gordon, K. C.; Strachan, C. J.; Rades, T. Perspectives in the use of spectroscopy to characterise pharmaceutical solids Int. J. Pharm. 2008, 364 (2) 159-169
-
(2008)
Int. J. Pharm.
, vol.364
, Issue.2
, pp. 159-169
-
-
Aaltonen, J.1
Gordon, K.C.2
Strachan, C.J.3
Rades, T.4
-
21
-
-
0031423468
-
Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions
-
DOI 10.1023/A:1012167410376
-
Taylor, L. S.; Zografi, G. Spectroscopic Characterization of Interactions Between PVP and Indomethacin in Amorphous Molecular Dispersions Pharm. Res. 1997, 14 (12) 1691-1698 (Pubitemid 28062912)
-
(1997)
Pharmaceutical Research
, vol.14
, Issue.12
, pp. 1691-1698
-
-
Taylor, L.S.1
Zografi, G.2
-
22
-
-
57449095886
-
Understanding the solid-state forms of fenofibrate - A spectroscopic and computational study
-
Heinz, A.; Gordon, K. C.; McGoverin, C. M.; Rades, T.; Strachan, C. J. Understanding the solid-state forms of fenofibrate-A spectroscopic and computational study Eur. J. Pharm. Biopharm. 2009, 71 (1) 100-108
-
(2009)
Eur. J. Pharm. Biopharm.
, vol.71
, Issue.1
, pp. 100-108
-
-
Heinz, A.1
Gordon, K.C.2
McGoverin, C.M.3
Rades, T.4
Strachan, C.J.5
-
23
-
-
33846818758
-
A theoretical and spectroscopic study of γ-crystalline and amorphous indometacin
-
DOI 10.1211/jpp.59.2.0012
-
Strachan, C. J.; Rades, T.; Gordon, K. C. A theoretical and spectroscopic study of γ-crystalline and amorphous indometacin J. Pharm. Pharmacol. 2007, 59 (2) 261-269 (Pubitemid 46203064)
-
(2007)
Journal of Pharmacy and Pharmacology
, vol.59
, Issue.2
, pp. 261-269
-
-
Strachan, C.J.1
Rades, T.2
Gordon, K.C.3
-
24
-
-
0036394705
-
Mechanism for further enhancement in drug dissolution from solid-dispersion granules upon storage
-
DOI 10.1081/PDT-120002236
-
Gupta, M. K.; Bogner, R. H.; Goldman, D.; Tseng, Y.-C. Mechanism for Further Enhancement in Drug Dissolution from Solid-Dispersion Granules upon Storage Pharm. Dev. Technol. 2002, 7 (1) 103-112 (Pubitemid 35154420)
-
(2002)
Pharmaceutical Development and Technology
, vol.7
, Issue.1
, pp. 103-112
-
-
Gupta, M.K.1
Bogner, R.H.2
Goldman, D.3
Tseng, Y.-C.4
-
25
-
-
0008342468
-
Refinement of the structure of naproxen, (+)-6-methoxy-α-methyl-2- naphthaleneacetic acid
-
Kim, Y.; Song, H.; Park, I. Refinement of the structure of naproxen, (+)-6-methoxy-α-methyl-2-naphthaleneacetic acid Arch. Pharmacal Res. 1987, 10 (4) 232-238
-
(1987)
Arch. Pharmacal Res.
, vol.10
, Issue.4
, pp. 232-238
-
-
Kim, Y.1
Song, H.2
Park, I.3
-
26
-
-
34248334514
-
Inhibiting surface crystallization of amorphous indomethacin by nanocoating
-
DOI 10.1021/la070050i
-
Wu, T.; Sun, Y.; Li, N.; de Villiers, M. M.; Yu, L. Inhibiting Surface Crystallization of Amorphous Indomethacin by Nanocoating Langmuir 2007, 23 (9) 5148-5153 (Pubitemid 46732007)
-
(2007)
Langmuir
, vol.23
, Issue.9
, pp. 5148-5153
-
-
Wu, T.1
Sun, Y.2
Li, N.3
De Villiers, M.M.4
Yu, L.5
-
27
-
-
0008819067
-
Non-crystalline solids: Glasses and amorphous solids
-
Gupta, P. K. Non-crystalline solids: glasses and amorphous solids J. Non-Cryst. Solids 1996, 195 (1-2) 158-164 (Pubitemid 126347265)
-
(1996)
Journal of Non-Crystalline Solids
, vol.195
, Issue.1-2
, pp. 158-164
-
-
Gupta, P.K.1
-
28
-
-
0030284632
-
The effects of co-lyophilized polymeric additives on the glass transition temperature and crystallization of amorphous sucrose
-
Shamblin, S. L.; Huang, E. Y.; Zografi, G. The effects of co-lyophilized polymeric additives on the glass transition temperature and crystallization of amorphous sucrose J. Therm. Anal. Calorim. 1996, 47 (5) 1567-1579 (Pubitemid 126794510)
-
(1996)
Journal of Thermal Analysis
, vol.47
, Issue.5
, pp. 1567-1579
-
-
Shamblin, S.L.1
Huang, E.Y.2
Zografi, G.3
-
29
-
-
0031797174
-
Sugar-polymer hydrogen bond interactions in lyophilized amorphous mixtures
-
DOI 10.1021/js9800174
-
Taylor, L. S.; Zografi, G. Sugar-polymer hydrogen bond interactions in lyophilized amorphous mixtures J. Pharm. Sci. 1998, 87 (12) 1615-1621 (Pubitemid 28559651)
-
(1998)
Journal of Pharmaceutical Sciences
, vol.87
, Issue.12
, pp. 1615-1621
-
-
Taylor, L.S.1
-
30
-
-
0031807819
-
Mixing behavior of colyophilized binary systems
-
DOI 10.1021/JS9704801
-
Shamblin, S. L.; Taylor, L. S.; Zografi, G. Mixing behavior of colyophilized binary systems J. Pharm. Sci. 1998, 87 (6) 694-701 (Pubitemid 28268567)
-
(1998)
Journal of Pharmaceutical Sciences
, vol.87
, Issue.6
, pp. 694-701
-
-
Shamblin, S.L.1
Taylor, L.S.2
Zografi, G.3
-
31
-
-
27144512688
-
Role of molecular interaction in stability of celecoxib-PVP amorphous systems
-
DOI 10.1021/mp050004g
-
Gupta, P.; Thilagavathi, R.; Chakraborti, A. K.; Bansal, A. K. Role of Molecular Interaction in Stability of Celecoxib-PVP Amorphous Systems Mol. Pharmaceutics 2005, 2 (5) 384-391 (Pubitemid 41503679)
-
(2005)
Molecular Pharmaceutics
, vol.2
, Issue.5
, pp. 384-391
-
-
Gupta, P.1
Thilagavathi, R.2
Chakraborti, A.K.3
Bansal, A.K.4
-
32
-
-
0034868680
-
The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion
-
DOI 10.1081/DDC-100105180
-
Forster, A.; Hempenstall, J.; Tucker, I.; Rades, T. The Potential of Small-Scale Fusion Experiments and the Gordon-Taylor Equation to Predict the Suitability of Drug/Polymer Blends for Melt Extrusion Drug Dev. Ind. Pharm. 2001, 27 (6) 549-560 (Pubitemid 32803574)
-
(2001)
Drug Development and Industrial Pharmacy
, vol.27
, Issue.6
, pp. 549-560
-
-
Forster, A.1
Hempenstall, J.2
Tucker, I.3
Rades, T.4
-
33
-
-
1842865536
-
Melt extrusion: From process to drug delivery technology
-
DOI 10.1016/S0939-6411(02)00061-9, PII S0939641102000619
-
Breitenbach, J. Melt extrusion: from process to drug delivery technology Eur. J. Pharm. Biopharm. 2002, 54 (2) 107-117 (Pubitemid 34919382)
-
(2002)
European Journal of Pharmaceutics and Biopharmaceutics
, vol.54
, Issue.2
, pp. 107-117
-
-
Breitenbach, J.1
|