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Volumn 3, Issue 3, 2011, Pages 582-600

Application of twin screw extrusion in the manufacture of cocrystals, part I: Four case studies

Author keywords

Cocrystals; Environmentally friendly; Green chemistry; Twin screw extrusion

Indexed keywords

CAFFEINE DERIVATIVE; CAFFEINE OXALIC ACID; CARBAMAZEPINE; CARBAMAZEPINE SACCHARIN; NICOTINAMIDE CINNAMIC ACID; NICOTINAMIDE DERIVATIVE; SOLVENT; THEOPHYLLINE CITRIC ACID; THEOPHYLLINE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 80053001573     PISSN: None     EISSN: 19994923     Source Type: Journal    
DOI: 10.3390/pharmaceutics3030582     Document Type: Article
Times cited : (86)

References (37)
  • 1
    • 0035289779 scopus 로고    scopus 로고
    • Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
    • Lipinski, C.A.; Lombardo, F.; Dominy, B.W.; Feeney, P.J. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Adv. Drug Delivery Rev. 2001, 46, 3-26.
    • (2001) Adv. Drug Delivery Rev , vol.46 , pp. 3-26
    • Lipinski, C.A.1    Lombardo, F.2    Dominy, B.W.3    Feeney, P.J.4
  • 2
    • 34548231676 scopus 로고    scopus 로고
    • What is a co-crystal?
    • Bond, A.D. What is a co-crystal? CrystEngComm 2007, 9, 833-834.
    • (2007) CrystEngComm , vol.9 , pp. 833-834
    • Bond, A.D.1
  • 3
    • 8844275016 scopus 로고    scopus 로고
    • Crystal and co-crystal
    • Desiraju, G.R. Crystal and co-crystal. CrystEngComm 2003, 5, 466-467.
    • (2003) CrystEngComm , vol.5 , pp. 466-467
    • Desiraju, G.R.1
  • 4
    • 8844280262 scopus 로고    scopus 로고
    • Crystal and co-crystal. A second opinion
    • Dunitz, J.D. Crystal and co-crystal. A second opinion. CrystEngComm 2003, 5, 506.
    • (2003) CrystEngComm , vol.5 , pp. 506
    • Dunitz, J.D.1
  • 6
    • 27744484364 scopus 로고    scopus 로고
    • Saccharin Salts of Active Pharmaceutical Ingredients, Their Crystal Structures, and Increased Water Solubilities
    • Banerjee, R.; Bhatt, P.M.; Ravindra, N.V.; Desiraju, G.R. Saccharin Salts of Active Pharmaceutical Ingredients, Their Crystal Structures, and Increased Water Solubilities. Cryst. Growth Des. 2005, 5, 2299-2309.
    • (2005) Cryst. Growth Des , vol.5 , pp. 2299-2309
    • Banerjee, R.1    Bhatt, P.M.2    Ravindra, N.V.3    Desiraju, G.R.4
  • 8
    • 34547486346 scopus 로고    scopus 로고
    • Cocrystals of Piroxicam with Carboxylic Acids
    • Childs, S.L.; Hardcastle, K.I. Cocrystals of Piroxicam with Carboxylic Acids. Cryst. Growth Des. 2007, 7, 1291-1304.
    • (2007) Cryst. Growth Des , vol.7 , pp. 1291-1304
    • Childs, S.L.1    Hardcastle, K.I.2
  • 9
    • 66249101601 scopus 로고    scopus 로고
    • Solubility Advantage of Pharmaceutical Cocrystals
    • Good, D.J.; Rodriguez-Hornedo, N. Solubility Advantage of Pharmaceutical Cocrystals. Cryst. Growth Des. 2009, 9, 2252-2264.
    • (2009) Cryst. Growth Des , vol.9 , pp. 2252-2264
    • Good, D.J.1    Rodriguez-Hornedo, N.2
  • 12
    • 33645320255 scopus 로고    scopus 로고
    • Preparation and Solid-State Characterization of Nonstoichiometric Cocrystals of a Phosphodiesterase-IV Inhibitor and L-Tartaric Acid
    • Variankaval, N.; Wenslow, R.; Murry, J.; Hartman, R.; Helmy, R.; Kwong, E.; Clas, S.-D.; Dalton, C.; Santos, I. Preparation and Solid-State Characterization of Nonstoichiometric Cocrystals of a Phosphodiesterase-IV Inhibitor and L-Tartaric Acid. Cryst. Growth Des. 2006, 6, 690-700.
    • (2006) Cryst. Growth Des , vol.6 , pp. 690-700
    • Variankaval, N.1    Wenslow, R.2    Murry, J.3    Hartman, R.4    Helmy, R.5    Kwong, E.6    Clas, S.-D.7    Dalton, C.8    Santos, I.9
  • 13
    • 19944371772 scopus 로고    scopus 로고
    • Pharmaceutical Cocrystallization: Engineering a Remedy for Caffeine Hydration
    • Trask, A.V.; Motherwell, W.D.S.; Jones, W. Pharmaceutical Cocrystallization: Engineering a Remedy for Caffeine Hydration. Cryst. Growth Des. 2005, 5, 1013-1021.
    • (2005) Cryst. Growth Des , vol.5 , pp. 1013-1021
    • Trask, A.V.1    Motherwell, W.D.S.2    Jones, W.3
  • 14
    • 33746425242 scopus 로고    scopus 로고
    • Physical stability enhancement of theophylline via cocrystallization
    • Trask, A.V.; Motherwell, W.D.S.; Jones, W. Physical stability enhancement of theophylline via cocrystallization. Int. J. Pharm. 2006, 320, 114-123.
    • (2006) Int. J. Pharm , vol.320 , pp. 114-123
    • Trask, A.V.1    Motherwell, W.D.S.2    Jones, W.3
  • 15
    • 70350342771 scopus 로고    scopus 로고
    • Improving mechanical properties of crystalline solids by cocrystal formation: New compressible forms of paracetamol
    • Karki, S.; Friscic, T.; Fabian, L.; Laity, P.R.; Day, G.M.; Jones, W. Improving mechanical properties of crystalline solids by cocrystal formation: new compressible forms of paracetamol. Adv. Mater. (Weinheim Ger.) 2009, 21, 3905-3909.
    • (2009) Adv. Mater. (Weinheim Ger.) , vol.21 , pp. 3905-3909
    • Karki, S.1    Friscic, T.2    Fabian, L.3    Laity, P.R.4    Day, G.M.5    Jones, W.6
  • 16
    • 60849109695 scopus 로고    scopus 로고
    • Improving Mechanical Properties of Caffeine and Methyl Gallate Crystals by Cocrystallization
    • Sun, C.C.; Hou, H. Improving Mechanical Properties of Caffeine and Methyl Gallate Crystals by Cocrystallization. Cryst. Growth Des. 2008, 8, 1575-1579.
    • (2008) Cryst. Growth Des , vol.8 , pp. 1575-1579
    • Sun, C.C.1    Hou, H.2
  • 19
    • 77956879551 scopus 로고    scopus 로고
    • High-throughput cocrystal slurry screening by use of in situ Raman microscopy and multi-well plate
    • Kojima, T.; Tsutsumi, S.; Yamamoto, K.; Ikeda, Y.; Moriwaki, T. High-throughput cocrystal slurry screening by use of in situ Raman microscopy and multi-well plate. Int. J. Pharm. 2010, 399, 52-59.
    • (2010) Int. J. Pharm , vol.399 , pp. 52-59
    • Kojima, T.1    Tsutsumi, S.2    Yamamoto, K.3    Ikeda, Y.4    Moriwaki, T.5
  • 21
    • 53849093843 scopus 로고    scopus 로고
    • Cocrystal Screening of Stanolone and Mestanolone Using Slurry Crystallization
    • Takata, N.; Shiraki, K.; Takano, R.; Hayashi, Y.; Terada, K. Cocrystal Screening of Stanolone and Mestanolone Using Slurry Crystallization. Cryst. Growth Des. 2008, 8, 3032-3037.
    • (2008) Cryst. Growth Des , vol.8 , pp. 3032-3037
    • Takata, N.1    Shiraki, K.2    Takano, R.3    Hayashi, Y.4    Terada, K.5
  • 22
    • 34249106473 scopus 로고    scopus 로고
    • Efficient co-crystal screening using solution-mediated phase transformation
    • Zhang, G.G.Z.; Henry, R.F.; Borchardt, T.B.; Lou, X. Efficient co-crystal screening using solution-mediated phase transformation. J. Pharm. Sci. 2007, 96, 990-995.
    • (2007) J. Pharm. Sci , vol.96 , pp. 990-995
    • Zhang, G.G.Z.1    Henry, R.F.2    Borchardt, T.B.3    Lou, X.4
  • 23
    • 34250545912 scopus 로고
    • Organic molecular compounds and their polymorphism
    • Quehenberger, H. Organic molecular compounds and their polymorphism. Monatsh. Chem. 1949, 80, 595-606.
    • (1949) Monatsh. Chem , vol.80 , pp. 595-606
    • Quehenberger, H.1
  • 25
    • 33845204296 scopus 로고    scopus 로고
    • Screening for inclusion compounds and systematic construction of three-component solids by liquid-assisted grinding
    • Friscic, T.; Trask, A.V.; Jones, W.; Motherwell, W.D.S. Screening for inclusion compounds and systematic construction of three-component solids by liquid-assisted grinding. Angew. Chem. Int. Ed. 2006, 45, 7546-7550.
    • (2006) Angew. Chem. Int , vol.45 , pp. 7546-7550
    • Friscic, T.1    Trask, A.V.2    Jones, W.3    Motherwell, W.D.S.4
  • 27
    • 34547474059 scopus 로고    scopus 로고
    • Making Co-Crystals - The Utility of Ternary Phase Diagrams
    • Chiarella, R.A.; Davey, R.J.; Peterson, M.L. Making Co-Crystals - The Utility of Ternary Phase Diagrams. Cryst. Growth Des. 2007, 7, 1223-1226.
    • (2007) Cryst. Growth Des , vol.7 , pp. 1223-1226
    • Chiarella, R.A.1    Davey, R.J.2    Peterson, M.L.3
  • 28
    • 32644436069 scopus 로고    scopus 로고
    • Phase Solubility Diagrams of Cocrystals Are Explained by Solubility Product and Solution Complexation
    • Nehm, S.J.; Rodriguez-Spong, B.; Rodriguez-Hornedo, N. Phase Solubility Diagrams of Cocrystals Are Explained by Solubility Product and Solution Complexation. Cryst. Growth Des. 2006, 6, 592-600.
    • (2006) Cryst. Growth Des , vol.6 , pp. 592-600
    • Nehm, S.J.1    Rodriguez-Spong, B.2    Rodriguez-Hornedo, N.3
  • 31
    • 60849098457 scopus 로고    scopus 로고
    • Scalable solution cocrystallization: Case of carbamazepine-nicotinamide I
    • Sheikh, A.Y.; Abd Rahim, S.; Hammond, R.B.; Roberts, K.J. Scalable solution cocrystallization: case of carbamazepine-nicotinamide I. CrystEngComm 2009, 11, 501-509.
    • (2009) CrystEngComm , vol.11 , pp. 501-509
    • Sheikh, A.Y.1    Abd Rahim, S.2    Hammond, R.B.3    Roberts, K.J.4
  • 32
    • 77949791492 scopus 로고    scopus 로고
    • Manufacture of pharmaceutical co-crystals using twin screw extrusion: A solvent-less and scalable process
    • Medina, C.; Daurio, D.; Nagapudi, K.; Alvarez-Nunez, F. Manufacture of pharmaceutical co-crystals using twin screw extrusion: a solvent-less and scalable process. J. Pharm. Sci. 2010, 99, 1693-1696.
    • (2010) J. Pharm. Sci , vol.99 , pp. 1693-1696
    • Medina, C.1    Daurio, D.2    Nagapudi, K.3    Alvarez-Nunez, F.4
  • 33
    • 80053022353 scopus 로고    scopus 로고
    • Development of solvent free continuous cocrystallisation technique
    • Dhumal, R.S.; Kelly, A.L.; Paradkar, A.R. Development of solvent free continuous cocrystallisation technique. J. Pharm. Pharmacol. 2010, 62, 1418-1419.
    • (2010) J. Pharm. Pharmacol , vol.62 , pp. 1418-1419
    • Dhumal, R.S.1    Kelly, A.L.2    Paradkar, A.R.3
  • 34
    • 78651333999 scopus 로고    scopus 로고
    • Cocrystallization and Simultaneous Agglomeration Using Hot Melt Extrusion
    • Dhumal, R.S.; Kelly, A.L.; York, P.; Coates, P.D.; Paradkar, A. Cocrystallization and Simultaneous Agglomeration Using Hot Melt Extrusion. Pharm. Res. 2010, 27, 2725-2733.
    • (2010) Pharm. Res , vol.27 , pp. 2725-2733
    • Dhumal, R.S.1    Kelly, A.L.2    York, P.3    Coates, P.D.4    Paradkar, A.5
  • 35
    • 33749449649 scopus 로고    scopus 로고
    • Cocrystal Formation during Cogrinding and Storage is Mediated by Amorphous Phase
    • Jayasankar, A.; Somwangthanaroj, A.; Shao, Z.J.; Rodriguez-Hornedo, N. Cocrystal Formation during Cogrinding and Storage is Mediated by Amorphous Phase. Pharm. Res. 2006, 23, 2381-2392.
    • (2006) Pharm. Res , vol.23 , pp. 2381-2392
    • Jayasankar, A.1    Somwangthanaroj, A.2    Shao, Z.J.3    Rodriguez-Hornedo, N.4
  • 36
    • 34250864401 scopus 로고    scopus 로고
    • Screening for Pharmaceutical Cocrystal Hydrates via Neat and Liquid-Assisted Grinding
    • Karki, S.; Friscic, T.; Jones, W.; Motherwell, W.D.S. Screening for Pharmaceutical Cocrystal Hydrates via Neat and Liquid-Assisted Grinding. Mol. Pharm. 2007, 4, 347-354.
    • (2007) Mol. Pharm , vol.4 , pp. 347-354
    • Karki, S.1    Friscic, T.2    Jones, W.3    Motherwell, W.D.S.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.