Synthesis and evaluation of analgesic and anti-inflammatory activities of most active free radical scavenging derivatives of embelin - A Structure-activity relationship

Chemical and Pharmaceutical Bulletin

Volumn 59, Issue 8, 2011, Pages 913-919

  Mahendran, Sekar ^a   Badami, Shrishailappa ^b   Ravi, Subban ^c   Thippeswamy, Boreddy Shivanandappa ^b   Veerapur, Veeresh Prabhakar ^b  

^a JSS COLLEGE OF PHARMACY   (India)

^b SREE SIDDAGANGA COLLEGE OF PHARMACY   (India)

^c KARPAGAM UNIVERSITY   (India)

Author keywords

Analgesic; Anti inflammatory; Antioxidant; Embelin; Structure activity relationship

Indexed keywords

1,1 DIPHENYL 2 PICRYLHYDRAZYL; 1,4 BENZOQUINONE DERIVATIVE; 2,2' AZINOBIS(3 ETHYLBENZOTHIAZOLINE 6 SULFONIC ACID); ACETIC ACID; ANALGESIC AGENT; ANTIINFLAMMATORY AGENT; ANTIOXIDANT; ASCORBIC ACID; DICLOFENAC; EMBELIN; PENTAZOCINE; RUTOSIDE; SCAVENGER; SULFONE DERIVATIVE;

ANALGESIC ACTIVITY; ANTIINFLAMMATORY ACTIVITY; ANTIOXIDANT ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; EMBELIA; EMBELIA RIBES; IN VITRO STUDY; MOTOR DYSFUNCTION; NONHUMAN; PAW EDEMA; RAT; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION; WRITHING;

ANIMALS; ANTI-INFLAMMATORY AGENTS; BENZOQUINONES; BENZOTHIAZOLES; EDEMA; EMBELIA; FREE RADICAL SCAVENGERS; FRUIT; HINDLIMB; MICE; PAIN; PLANT EXTRACTS; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONIC ACIDS;

EID: 79961108124     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.59.913     Document Type: Article

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