-
1
-
-
14444272751
-
Synthesis and evaluation of a series of novel 2-[(4- chlorophenoxy) methyl]-benzimidazoles as selective neuropeptide Y Y1 receptor antagonists hamideh zarrinmayeh
-
Zarrinmayeh, H.; Nunes, A. M.; Ornstein, P. L.; Zimmerman, D. M.; Brian Arnold, M.; Schober, D. A.; Gackenheimer, S. L.; Bruns, R. F.; Hipskind, P. A.; Britton, T. C.; Cantrell, B. E.; Gehlert, D. R. Synthesis and evaluation of a series of novel 2-[(4- chlorophenoxy)methyl]-benzimidazoles as selective neuropeptide Y Y1 receptor antagonists hamideh zarrinmayeh. J. Med. Chem., 1998, 41, 2709.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 2709
-
-
Zarrinmayeh, H.1
Nunes, A.M.2
Ornstein, P.L.3
Zimmerman, D.M.4
Brian Arnold, M.5
Schober, D.A.6
Gackenheimer, S.L.7
Bruns, R.F.8
Hipskind, P.A.9
Britton, T.C.10
Cantrell, B.E.11
Gehlert, D.R.12
-
2
-
-
0034597569
-
Resistance-modifying agents. 9.1 synthesis and biological properties of benzimidazole inhibitors of the DNA repair enzyme poly (ADP-ribose) polymerase
-
White, A. W.; Almassy, R.; Calvert, A. H.; Curtin, N. J.; Griffin, R. J.; Hostomsky, Z.; Maegley, K.; Newell, D. R.; Srinivasan, S.; Golding, B. T. Resistance-modifying agents. 9.1 synthesis and biological properties of benzimidazole inhibitors of the DNA repair enzyme poly (ADP-ribose) polymerase. J. Med. Chem., 2000, 43, 4084.
-
(2000)
J. Med. Chem.
, vol.43
, pp. 4084
-
-
White, A.W.1
Almassy, R.2
Calvert, A.H.3
Curtin, N.J.4
Griffin, R.J.5
Hostomsky, Z.6
Maegley, K.7
Newell, D.R.8
Srinivasan, S.9
Golding, B.T.10
-
3
-
-
77956444015
-
Synthesis of novel tripodal-benzimidazole from 2,4,6-tris(p- formylphenoxy)-1,3,5-triazine: Structural, electrochemical and antimicrobial studies
-
Koc, Z. E.; Bingol, H.; Saf, A. O.; Torlak, E.; Coskun, A. Synthesis of novel tripodal-benzimidazole from 2,4,6-tris(p-formylphenoxy)-1,3,5-triazine: structural, electrochemical and antimicrobial studies. J. Hazard. Mater., 2010, 183, 251.
-
(2010)
J. Hazard. Mater.
, vol.183
, pp. 251
-
-
Koc, Z.E.1
Bingol, H.2
Saf, A.O.3
Torlak, E.4
Coskun, A.5
-
4
-
-
77955904687
-
Synthesis characterization, and biological evaluation of benzimidazole derivatives as potential anxiolytics
-
Nannapaneni, D.; Gupta Atyam, V.; Reddy, M.; Raidu, S. Synthesis, characterization, and biological evaluation of benzimidazole derivatives as potential anxiolytics. J. Young Pharmacists, 2010, 2, 273.
-
(2010)
J. Young Pharmacists
, vol.2
, pp. 273
-
-
Nannapaneni, D.1
Gupta, A.V.2
Reddy, M.3
Raidu, S.4
-
5
-
-
0032499283
-
Design, synthesis, and antiviral evaluations of 1- (substituted benzyl)-2-substituted-5,6-dichlorobenzimidazoles as nonnucleoside analogues of 2,5,6-trichloro-1-(β-d-ribofuranosyl) benzimidazole
-
Porcari, A. R.; Devivar, R. V.; Kucera, L. S.; Drach, J. C.; Townsend, L. B. Design, synthesis, and antiviral evaluations of 1- (substituted benzyl)-2-substituted-5,6-dichlorobenzimidazoles as nonnucleoside analogues of 2,5,6-trichloro-1-(β-d-ribofuranosyl) benzimidazole. J. Med. Chem., 1998, 41, 1252.
-
(1998)
J. Med. Chem.
, Issue.41
, pp. 1252
-
-
Porcari, A.R.1
Devivar, R.V.2
Kucera, L.S.3
Drach, J.C.4
Townsend, L.B.5
-
6
-
-
0031463691
-
Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase. 2- aryl-substituted benzimidazoles
-
Roth, T.; Morningstar, M. L.; Boyer, P. L.; Hughes, S. H.; Buckheit, R. W. Jr.; Michejda, C. J. Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase. 2- aryl-substituted benzimidazoles. J. Med. Chem., 1997, 40, 4199
-
(1997)
J. Med. Chem.
, vol.40
, pp. 4199
-
-
Roth, T.1
Morningstar, M.L.2
Boyer, P.L.3
Hughes, S.H.4
Buckheit Jr., R.W.5
Michejda, C.J.6
-
7
-
-
0032499278
-
-
Design, synthesis, and antiviral activity of α-nucleosides: D- and L-isomers of lyxofuranosyl- and (5-deoxylyxofuranosyl)benzimidazoles
-
Migawa, M. T.; Girardet, J. L.; Walker II, J. A.; Koszalka, G. W.; Chamberlain, S. D.; Drach, J. C.; Townsend, L. B. Design, synthesis, and antiviral activity of α-nucleosides: D- and L-isomers of lyxofuranosyl- and (5-deoxylyxofuranosyl)benzimidazoles. J. Med. Chem., 1998, 41, 1242.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 1242
-
-
Migawa, M.T.1
Girardet, J.L.2
Walker II, J.A.3
Koszalka, G.W.4
Chamberlain, S.D.5
Drach, J.C.6
Townsend, L.B.7
-
8
-
-
0017915202
-
Halobenzimidazole ribosides and RNA synthesis of cells and viruses
-
Tamm, I.; Seghal, P. B. Halobenzimidazole ribosides and RNA synthesis of cells and viruses. Adv. Virus Res., 1978, 22, 187.
-
(1978)
Adv. Virus Res.
, vol.22
, pp. 187
-
-
Tamm, I.1
Seghal, P.B.2
-
9
-
-
37049243363
-
Inhibition of influenza and mumps virus multiplication by 4,5,6-(or 5,6,7-) trichloro-1-β-D-ribofuranosylbenzimidazole
-
Tamm, I. Inhibition of influenza and mumps virus multiplication by 4,5,6-(or 5,6,7-) trichloro-1-β-D-ribofuranosylbenzimidazole. Science, 1954, 120, 847.
-
(1954)
Science
, Issue.120
, pp. 847
-
-
Tamm, I.1
-
10
-
-
33947458464
-
The chemistry of the benzimidazoles
-
Wright, J. B. The chemistry of the benzimidazoles. Chem. Rev., 1951, 48, 397.
-
(1951)
Chem. Rev.
, vol.48
, pp. 397
-
-
Wright, J.B.1
-
11
-
-
0019167326
-
Synthesis of imidazo[4,5-b]- and [4,5-c]pyridines
-
Middleton, R. W.; George Wibberley, D. Synthesis of imidazo[4,5-b]- and [4,5-c]pyridines. J. Heterocycl. Chem., 1980, 17, 1757.
-
(1980)
J. Heterocycl. Chem.
, vol.17
, pp. 1757
-
-
Middleton, R.W.1
George, W.D.2
-
12
-
-
31344432191
-
Derivatives of 2-phenylbenzimidazole
-
Rope, M.; Isensee, R. W.; Joseph, L. Derivatives of 2- phenylbenzimidazole. J. Am. Chem. Soc., 1952, 74, 1095.
-
(1952)
J. Am. Chem. Soc.
, vol.74
, pp. 1095
-
-
Rope, M.1
Isensee, R.W.2
Joseph, L.3
-
13
-
-
0001291624
-
Synthesis of monocationic and dicationic analogs of hoechst 33258
-
Czarny, A.; Wilson, W. D.; Boykin, D. W. Synthesis of monocationic and dicationic analogs of hoechst 33258. J. Heterocycl. Chem., 1996, 33, 1393.
-
(1996)
J. Heterocycl. Chem.
, vol.33
, pp. 1393
-
-
Czarny, A.1
Wilson, W.D.2
Boykin, D.W.3
-
14
-
-
0017872205
-
Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring
-
Inhibitors of arginine-specific esteroproteases
-
Tidwell, R. R.; Geratz, J. D.; Dann, O.; Volz, G.; Zeh, D.; Loewe, H. Diarylamidine derivatives with one or both of the aryl moieties consisting of an indole or indole-like ring. Inhibitors of arginine-specific esteroproteases. J. Med. Chem., 1978, 21, 613.
-
(1978)
J. Med. Chem.
, vol.21
, pp. 613
-
-
Tidwell, R.R.1
Geratz, J.D.2
Dann, O.3
Volz, G.4
Zeh, D.5
Loewe, H.6
-
15
-
-
0027253921
-
Structure, DNA minor groove binding, and base pair specificity of alkyl- and aryl-linked bis(amidinobenzimidazoles) and bis(amidinoindoles)
-
Fairley, T. A.; Tidwell, R. R.; Donkor, I.; Naiman, N. A.; Ohemeng, K. A.; Lombardy, R. J.; Bentley, J. A.; Cory, M. Structure, DNA minor groove binding, and base pair specificity of alkyl- and aryl-linked bis(amidinobenzimidazoles) and bis(amidinoindoles). J. Med. Chem., 1993, 36, 1746.
-
(1993)
J. Med. Chem.
, vol.36
, pp. 1746
-
-
Fairley, T.A.1
Tidwell, R.R.2
Donkor, I.3
Naiman, N.A.4
Ohemeng, K.A.5
Lombardy, R.J.6
Bentley, J.A.7
Cory, M.8
-
16
-
-
0032500083
-
Trois nouvelles voies de synthèse des dérivés 1,3-azoliques sous micro-ondes
-
Bougrin, K.; Loupy, A.; Soufiaoui, M. Trois nouvelles voies de synthèse des dérivés 1,3-azoliques sous micro-ondes. Tetrahedron, 1998, 54, 8055
-
(1998)
Tetrahedron
, vol.54
, pp. 8055
-
-
Bougrin, K.1
Loupy, A.2
Soufiaoui, M.3
-
17
-
-
0036324238
-
A simple and efficient method for the synthesis of novel trifluoromethyl benzimidazoles under microwave irradiation conditions
-
Venkat Reddy, G.; Rama Rao, V. V. V. N. S.; Narsaiah, B.; Shanthan Rao, P. A simple and efficient method for the synthesis of novel trifluoromethyl benzimidazoles under microwave irradiation conditions. Synth. Commun., 2002, 32, 2467
-
(2002)
Synth. Commun.
, Issue.32
, pp. 2467
-
-
Venkat, R.G.1
Rama, R.V.V.V.N.S.2
Narsaiah, B.3
Shanthan, R.P.4
-
18
-
-
0032543469
-
Benzimidazoles: Oxydation hétérocyclisante par le nitrobenzène ou le diméthylsulfoxyde sur silice et sous irradiation micro-ondes ou ultra-violet
-
Ben-Alloum, A.; Bakkas, S.; Soufiaoui, M. Benzimidazoles: oxydation hétérocyclisante par le nitrobenzène ou le diméthylsulfoxyde sur silice et sous irradiation micro-ondes ou ultra-violet. Tetrahedron Lett., 1998, 39, 4481
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 4481
-
-
Ben-Alloum, A.1
Bakkas, S.2
Soufiaoui, M.3
-
19
-
-
4143063050
-
Convenient routes to substituted benzimidazoles and imidazolo[4,5-b] pyridines using nitrobenzene as oxidant
-
Yadagiri, B.; William Lown, J. Convenient routes to substituted benzimidazoles and imidazolo[4,5-b]pyridines using nitrobenzene as oxidant. Synth. Commun., 1990, 20, 955.
-
(1990)
Synth. Commun.
, Issue.20
, pp. 955
-
-
Yadagiri, B.1
William Lown, J.2
-
20
-
-
0035899191
-
Development of serine protease inhibitors displaying a multicentered short (>2.3 A) hydrogen bond binding mode: Inhibitors of urokinase-type plasminogen activator and factor Xa
-
Verner, E.; Katz, B. A.; Spencer, J. R.; Allen, D.; Hataye, J.; Hruzewicz, W.; Hui, H. C.; Kolesnikov, A.; Li, Y.; Luong, C.; Martelli, A.; Radika, K.; Rai, R.; She, M.; Shrader, W.; Sprengeler, P. A.; Trapp, S.; Wang, J.; Young, W. B.; Mackman, R. L. Development of serine protease inhibitors displaying a multicentered short (>2.3 A) hydrogen bond binding mode: inhibitors of urokinase-type plasminogen activator and factor Xa. J. Med. Chem., 2001, 44,2753.
-
(2001)
J. Med. Chem.
, vol.44
, pp. 2753
-
-
Verner, E.1
Katz, B.A.2
Spencer, J.R.3
Allen, D.4
Hataye, J.5
Hruzewicz, W.6
Hui, H.C.7
Kolesnikov, A.8
Li, Y.9
Luong, C.10
Martelli, A.11
Radika, K.12
Rai, R.13
She, M.14
Shrader, W.15
Sprengeler, P.A.16
Trapp, S.17
Wang, J.18
Young, W.B.19
Mackman, R.L.20
more..
-
21
-
-
0029061671
-
2,3- Dichloro-5,6-dicyano-1,4-benzoquinone, a mild catalyst for the formation of carbon-nitrogen bonds
-
Eynde, J. J. V.; Delfosse, F.; Lor, P.; Haverbeke, Y. V. 2,3- Dichloro-5,6-dicyano-1,4-benzoquinone, a mild catalyst for the formation of carbon-nitrogen bonds. Tetrahedron, 1995, 51, 5813.
-
(1995)
Tetrahedron
, vol.51
, pp. 5813
-
-
Eynde, J.J.V.1
Delfosse, F.2
Lor, P.3
Haverbeke, Y.V.4
-
22
-
-
0035687467
-
Traceless solid-phase synthesis of 5-benzoylbenzimidazoles
-
Lee, K. J.; Janda, K. D. Traceless solid-phase synthesis of 5- benzoylbenzimidazoles. Can. J. Chem., 2001, 79, 1556.
-
(2001)
Can. J. Chem.
, vol.79
, pp. 1556
-
-
Lee, K.J.1
Janda, K.D.2
-
23
-
-
0000997887
-
In situ generation and synthetic application of 2- phenylbenzimidazoline to the selective reduction of carbon-carbon double bonds of electron-deficient olefins
-
Chikashita, H.; Nishida, S.; Miyazaki, M.; Morita, Y.; Itoh, K. In situ generation and synthetic application of 2- phenylbenzimidazoline to the selective reduction of carbon-carbon double bonds of electron-deficient olefins. Bull. Chem. Soc. Jpn., 1987, 60, 737.
-
(1987)
Bull. Chem. Soc. Jpn.
, vol.60
, pp. 737
-
-
Chikashita, H.1
Nishida, S.2
Miyazaki, M.3
Morita, Y.4
Itoh, K.5
-
24
-
-
40549107132
-
New one-pot procedure for the synthesis of 2-substituted benzimidazoles
-
Sharghi, H.; Asemani, O.; Khalifeh, R. New one-pot procedure for the synthesis of 2-substituted benzimidazoles. Synth. Commun., 2008, 38, 1128.
-
(2008)
Synth. Commun.
, vol.38
, pp. 1128
-
-
Sharghi, H.1
Asemani, O.2
Khalifeh, R.3
-
25
-
-
0000586488
-
Oxidation with metal oxides-II : Oxidation of chalcone phenylhydrazones, pyrazolines, oaminobenzylidine anils and o-hydroxy benzylidine anils with manganese dioxide
-
Bhatnagar, I.; George, M. V. Oxidation with metal oxides-II : oxidation of chalcone phenylhydrazones, pyrazolines, oaminobenzylidine anils and o-hydroxy benzylidine anils with manganese dioxide. Tetrahedron, 1968, 24, 1293.
-
(1968)
Tetrahedron
, vol.24
, pp. 1293
-
-
Bhatnagar, I.1
George, M.V.2
-
26
-
-
0037631073
-
Synthèse chimiosélective des benzimidazoles sur silice traitée par le chlorure du thionyle
-
Alloum, A. B.; Bougrinb, K.; Soufiaouib, M. Synthèse chimiosélective des benzimidazoles sur silice traitée par le chlorure du thionyle. Tetrahedron Lett., 2003, 44, 5935.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 5935
-
-
Alloum, A.B.1
Bougrinb, K.2
Soufiaouib, M.3
-
27
-
-
0043240483
-
Practical oxone®- Mediated, high-throughput, solution-phase synthesis of benzimidazoles from 1,2-phenylenediamines and aldehydes and its application to preparative scale synthesis
-
Beaulieu, P. L.; Haché, B.; von Moos, E. A Practical Oxone®- Mediated, High-Throughput, Solution-Phase Synthesis of Benzimidazoles from 1,2-Phenylenediamines and Aldehydes and its Application to Preparative Scale Synthesis. Synthesis, 2003, 1683.
-
(2003)
Synthesis
, pp. 1683
-
-
Beaulieu, P.L.1
Haché, B.2
Von, M.E.A.3
-
28
-
-
33745685573
-
Application of sulfamic acid as an eco-friendly catalyst in an expedient synthesis of benzimidazoles
-
Chakrabarty, M.; Karmakar, S.; Mukherji, A.; Arima, S.; Harigaya, Y. Application of sulfamic acid as an eco-friendly catalyst in an expedient synthesis of benzimidazoles. Heterocycles, 2006, 68, 967
-
(2006)
Heterocycles
, vol.68
, pp. 967
-
-
Chakrabarty, M.1
Karmakar, S.2
Mukherji, A.3
Arima, S.4
Harigaya, Y.5
-
29
-
-
51849108118
-
Sulfonic acid functionalized silica as an efficient heterogeneous recyclable catalyst for one-pot synthesis of 2-substituted benziimidazoles
-
Das, B.; Kanth, B. S.; Reddy, K. R.; Kumar, A. S. Sulfonic acid functionalized silica as an efficient heterogeneous recyclable catalyst for one-pot synthesis of 2-substituted benziimidazoles. J. Heterocycl. Chem., 2008, 45, 1499.
-
(2008)
J. Heterocycl. Chem.
, vol.45
, pp. 1499
-
-
Das, B.1
Kanth, B.S.2
Reddy, K.R.3
Kumar, A.S.4
-
30
-
-
28544451672
-
An efficient and one-pot synthesis of imidazolines and benzimidazoles via anaerobic oxidation of carbon- nitrogen bonds in water
-
Gogoi, P.; Konwar, D. An efficient and one-pot synthesis of imidazolines and benzimidazoles via anaerobic oxidation of carbon- nitrogen bonds in water. Tetrahedron Lett., 2006, 47, 79
-
(2006)
Tetrahedron Lett.
, vol.47
, pp. 79
-
-
Gogoi, P.1
Konwar, D.2
-
31
-
-
33745398367
-
Iodine-mediated synthesis of 2- arylbenzoxazoles, 2-arylbenzimidazoles, and 1,3,5-trisubstituted pyrazoles
-
Ponnala, S.; Sahu, D. P. Iodine-mediated synthesis of 2- arylbenzoxazoles, 2-arylbenzimidazoles, and 1,3,5-trisubstituted pyrazoles. Synth. Commun., 2006, 36, 2189.
-
(2006)
Synth. Commun.
, Issue.36
, pp. 2189
-
-
Ponnala, S.1
Sahu, D.P.2
-
32
-
-
31544450237
-
A convenient one-pot synthesis of 2-substituted benzimidazoles
-
Trivedi, R.; De, S. K.; Gibbs, R. A. A convenient one-pot synthesis of 2-substituted benzimidazoles. J. Mol. Cat. A: Chem., 2006, 245, 8.
-
(2006)
J. Mol. Cat. A: Chem.
, vol.245
, pp. 8
-
-
Trivedi, R.1
De, S.K.2
Gibbs, R.A.3
-
33
-
-
4143104652
-
Ytterbium triflate promoted synthesis of benzimidazole derivatives
-
Curini, M.; Epifano, F.; Montanari, F.; Rosati, O.; Taccone, S. Ytterbium triflate promoted synthesis of benzimidazole derivatives. Synlett, 2004, 1832.
-
(2004)
Synlett
, vol.1832
-
-
Curini, M.1
Epifano, F.2
Montanari, F.3
Rosati, O.4
Taccone, S.5
-
34
-
-
33644905184
-
Synthesis of 2- Arylbenzothiazoles and imidazoles using scandium triflate as a catalyst for both a ring closing and an oxidation steps
-
Itoh, T.; Nagata, K.; Ishikawa, H.; Ohsawa, A. Synthesis of 2- arylbenzothiazoles and imidazoles using scandium triflate as a catalyst for both a ring closing and an oxidation steps. Heterocycles, 2004, 63, 2769
-
(2004)
Heterocycles
, vol.63
, pp. 2769
-
-
Itoh, T.1
Nagata, K.2
Ishikawa, H.3
Ohsawa, A.4
-
35
-
-
0345761268
-
Synthesis of 2-substituted benzimidazoles by reaction of ophenylenediamine with aldehydes in the presence of Sc(OTf)3
-
Nagata, K.; Itoh, T.; Ishikawa, H.; Ohsawa, A. Synthesis of 2-substituted benzimidazoles by reaction of ophenylenediamine with aldehydes in the presence of Sc(OTf)3. Heterocycles, 2003, 61, 93.
-
(2003)
Heterocycles
, Issue.61
, pp. 93
-
-
Nagata, K.1
Itoh, T.2
Ishikawa, H.3
Ohsawa, A.4
-
36
-
-
33749321211
-
A simple KHSO4 promoted synthesis of 2-arylsubstituted benzimidazoles by oxidative condensation of alde hydes with o-phenylenediamine
-
Ma, H. Q.; Wang, Y. L.; Wang, J. Y. A simple KHSO4 promoted synthesis of 2-arylsubstituted benzimidazoles by oxidative condensation of alde hydes with o-phenylenediamine. Heterocycles, 2006, 68, 1669.
-
(2006)
Heterocycles
, vol.68
, pp. 1669
-
-
Ma, H.Q.1
Wang, Y.L.2
Wang, J.Y.3
|