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Volumn 76, Issue 10-11, 2011, Pages 1082-1097

Investigation of new acyloxy derivatives of cholic acid and their esters as drug absorption modifiers

(12) Mrózek, Lech a Dvořáková, Lenka b Mandelová, Zuzana b Rárová, Lucie c Řezáčová, Anna b Plaček, Lukáš a Opatřilová, Radka b Dohnal, Jiří b Paleta, Oldřich d Král, Vladimír d Drašar, Pavel d Jampílek, Josef b

a BorsodChem MCHZ Sro ^* (Czech Republic)

b UNIVERSITY OF VETERINARY AND PHARMACEUTICAL SCIENCES (Czech Republic)

c PALACKÝ UNIVERSITY (Czech Republic)

d INSTITUTE OF CHEMICAL TECHNOLOGY (Czech Republic)

Author keywords

Cholic acid derivatives; In vitro cytotoxicity; Intestinal absorption promoters; Lipophilicity; Solubility; Transdermal penetration enhancers

Indexed keywords

CHOLIC ACID DERIVATIVE; ESTER; PENETRATION ENHANCING AGENT;

ARTICLE; BREAST ADENOCARCINOMA; CANCER CELL CULTURE; CANCER INHIBITION; CARBON NUCLEAR MAGNETIC RESONANCE; CHEMICAL ANALYSIS; CHEMICAL STRUCTURE; CONTROLLED STUDY; CYTOTOXICITY; HUMAN; HUMAN CELL; HYDROPHOBICITY; IN VITRO STUDY; INFRARED SPECTROSCOPY; INTESTINE ABSORPTION; LIPOPHILICITY; LYMPHATIC LEUKEMIA; MASS SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE; SKIN FIBROBLAST; SKIN PENETRATION; SOLUBILITY; SYNTHESIS; THIN LAYER CHROMATOGRAPHY;

ANIMALS; CELL LINE; CELL LINE, TUMOR; CHOLIC ACID; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; ESTERS; EXCIPIENTS; HUMANS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; MAGNETIC RESONANCE SPECTROSCOPY; SKIN; SKIN ABSORPTION; STRUCTURE-ACTIVITY RELATIONSHIP; SWINE; THEOPHYLLINE;

EID: 79960456607 PISSN: 0039128X EISSN: 18785867 Source Type: Journal
DOI: 10.1016/j.steroids.2011.04.014 Document Type: Article

Times cited : (30)

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