Interpretation of the effects of protein kinase C inhibitors on human UDP-glucuronosyltransferase 1A (UGT1A) proteins in cellulo

Drug Metabolism and Pharmacokinetics

Volumn 26, Issue 3, 2011, Pages 256-265

  Abe, Yuko ^a   Fujiwara, Ryoichi ^a   Oda, Shingo ^a   Yokoi, Tsuyoshi ^a   Nakajima, Miki ^a  

^a KANAZAWA UNIVERSITY   (Japan)

Author keywords

Degradation; Glucuronidation; Inhibition; Phosphorylation; UGT

Indexed keywords

CALPHOSTIN C; CURCUMIN; GLUCURONOSYLTRANSFERASE; GLUCURONOSYLTRANSFERASE 1A9; MESSENGER RNA; PHOSPHOPROTEIN; POLYHISTIDINE TAG; PROTEASOME; UDP GLUCURONOSYLTRANSFERASE 1A; UNCLASSIFIED DRUG;

ARTICLE; AUTOPHAGY; CELL STRAIN HEK293; CONCENTRATION RESPONSE; CONTROLLED STUDY; ENZYME ACTIVITY; ENZYME DEGRADATION; ENZYME INHIBITION; GENE EXPRESSION SYSTEM; HUMAN; HUMAN CELL; IMMUNOBLOTTING; IMMUNOPRECIPITATION; IN VITRO STUDY; PROTEIN EXPRESSION; PROTEIN PHOSPHORYLATION; PROTEIN PURIFICATION;

EID: 79959974678     PISSN: 13474367     EISSN: 18800920     Source Type: Journal    
DOI: 10.2133/dmpk.DMPK-10-RG-121     Document Type: Article

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