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Volumn , Issue , 2010, Pages 129-153

Controlled release using bilayer osmotic tablet technology: reducing theory to practice

Author keywords

Bilayer osmotic tablets functional swelling layer and manufactured delivery port; Controlled release using bilayer osmotic tablet technology reducing theory to practice; in vitro performance testing tablet release rate measures, in vitro characterization using dissolution testing

Indexed keywords


EID: 79958258569     PISSN: None     EISSN: None     Source Type: Book    
DOI: 10.1002/9780470640487.ch9     Document Type: Chapter
Times cited : (13)

References (66)
  • 2
    • 85056041650 scopus 로고    scopus 로고
    • In Amidon GL. Lee PI, Topp EM, editors. Marcel Dekkar, New York
    • Cardinal JR. In Amidon GL, Lee PI, Topp EM, editors. Transport Processes in Pharmaceutical Systems, Marcel Dekkar, New York, 2000, pp. 411-444.
    • (2000) Transport Processes in Pharmaceutical Systems , pp. 411-444
    • Cardinal, J.R.1
  • 4
    • 0029076668 scopus 로고
    • Osmotic drug delivery: a review of the patent literature
    • Santus G, Baker RW. Osmotic drug delivery: a review of the patent literature. J. Control. Release 1995;35:1-21.
    • (1995) J. Control. Release , vol.35 , pp. 1-21
    • Santus, G.1    Baker, R.W.2
  • 5
    • 0016830071 scopus 로고
    • Elementary osmotic pump
    • Theeuwes F. Elementary osmotic pump. J. Pharm. Sci. 1975; 64:1987-1991.
    • (1975) J. Pharm. Sci. , vol.64 , pp. 1987-1991
    • Theeuwes, F.1
  • 6
    • 77049235472 scopus 로고
    • A continuous long-term injector
    • Rose S, Nelson JF. A continuous long-term injector. Aust. J. Exp. Biol. 1955;33:415-420.
    • (1955) Aust. J. Exp. Biol. , vol.33 , pp. 415-420
    • Rose, S.1    Nelson, J.F.2
  • 8
    • 0034044857 scopus 로고    scopus 로고
    • Osmotically controlled oral drug delivery
    • Verma RK, Mishra B, Garg S. Osmotically controlled oral drug delivery. Drug Dev. Ind. Pharm. 2000;26(7):695-708.
    • (2000) Drug Dev. Ind. Pharm. , vol.26 , Issue.7 , pp. 695-708
    • Verma, R.K.1    Mishra, B.2    Garg, S.3
  • 10
    • 38149101751 scopus 로고    scopus 로고
    • Factors affecting the release of nifedipine from a swellable elementary osmotic pump
    • Nokhodchi A, Momin MN, Shokri J, Shahsavari M, Rashidi PA. Factors affecting the release of nifedipine from a swellable elementary osmotic pump. Drug Deliv. 2008;15(1): 43-48.
    • (2008) Drug Deliv. , vol.15 , Issue.1 , pp. 43-48
    • Nokhodchi, A.1    Momin, M.N.2    Shokri, J.3    Shahsavari, M.4    Rashidi, P.A.5
  • 11
    • 34648818167 scopus 로고    scopus 로고
    • Studies on bi-layer osmotic pump tablets of water-insoluble allopurinol with large dose: in vitro and in vivo
    • Wang X, Nie S-F, Li W, Luan L, Pan W. Studies on bi-layer osmotic pump tablets of water-insoluble allopurinol with large dose: in vitro and in vivo. Drug Dev. Ind. Pharm. 2007;33(9): 1024-1029.
    • (2007) Drug Dev. Ind. Pharm. , vol.33 , Issue.9 , pp. 1024-1029
    • Wang, X.1    Nie, S.-F.2    Li, W.3    Luan, L.4    Pan, W.5
  • 12
    • 24944523675 scopus 로고    scopus 로고
    • Assessment of the feasibility of oral controlled release in an exploratory development setting
    • Thombre AG. Assessment of the feasibility of oral controlled release in an exploratory development setting. Drug Discov. Today 2005;10(17):1159-1166.
    • (2005) Drug Discov. Today , vol.10 , Issue.17 , pp. 1159-1166
    • Thombre, A.G.1
  • 15
    • 0023514452 scopus 로고
    • In vitro study of gastrointestinal diffusion system using disopyramide phosphate
    • Jedras Z, Janicki S. In vitro study of gastrointestinal diffusion system using disopyramide phosphate. Pharmazie 1987;42 (12): 842-844.
    • (1987) Pharmazie , vol.42 , Issue.12 , pp. 842-844
    • Jedras, Z.1    Janicki, S.2
  • 16
    • 0021729931 scopus 로고
    • Oral dosage forms design: status and goals of oral osmotic systems technology
    • Theeuwes F. Oral dosage forms design: status and goals of oral osmotic systems technology. Pharm. Int. 1984;5:293-296.
    • (1984) Pharm. Int. , vol.5 , pp. 293-296
    • Theeuwes, F.1
  • 17
    • 0042782044 scopus 로고    scopus 로고
    • Feasibility assessment and rapid development of oral controlled release prototypes.
    • Controlled Drug Delivery
    • Thombre AG. Feasibility assessment and rapid development of oral controlled release prototypes. ACS Symp. Ser.; 752 (Controlled Drug Delivery): 2000, 69-77.
    • (2000) ACS Symp. Ser. , vol.752 , pp. 69-77
    • Thombre, A.G.1
  • 18
    • 43249121029 scopus 로고    scopus 로고
    • Gut instincts: explorations in intestinal physiology and drug delivery
    • McConnell EL, Fadda HM, Basit AW. Gut instincts: explorations in intestinal physiology and drug delivery. Int. J. Pharm. 2008;364(2):213-226.
    • (2008) Int. J. Pharm. , vol.364 , Issue.2 , pp. 213-226
    • McConnell, E.L.1    Fadda, H.M.2    Basit, A.W.3
  • 21
    • 41549164293 scopus 로고    scopus 로고
    • Dissolution: fundamentals of in vitro release and the biopharmaceutics classification system
    • Pharmaceutical Product Development
    • Johnson KC. Dissolution: fundamentals of in vitro release and the biopharmaceutics classification system. Drugs Pharm. Sci. 2007;165(Pharmaceutical Product Development):1-28.
    • (2007) Drugs Pharm. Sci. , vol.165 , pp. 1-28
    • Johnson, K.C.1
  • 22
    • 0027275798 scopus 로고
    • Dissolution modeling: factors affecting the dissolution rates of polydisperse powders
    • Lu ATK, Frisella ME, Johnson KC. Dissolution modeling: factors affecting the dissolution rates of polydisperse powders. Pharm. Res. 1993;10(9):1308-1314.
    • (1993) Pharm. Res. , vol.10 , Issue.9 , pp. 1308-1314
    • Lu, A.TK.1    Frisella, M.E.2    Johnson, K.C.3
  • 23
    • 34648818167 scopus 로고    scopus 로고
    • Studies on bi-layer osmotic pump tablets of water-insoluble allopurinol with large dose: in vitro and in vivo
    • Nie S-F, Li W, Luan L, Pan W, Wang X. Studies on bi-layer osmotic pump tablets of water-insoluble allopurinol with large dose: in vitro and in vivo. Drug Dev. Ind. Pharm. 2007;33 (9):1024-1029.
    • (2007) Drug Dev. Ind. Pharm. , vol.33 , Issue.9 , pp. 1024-1029
    • Nie, S.-F.1    Li, W.2    Luan, L.3    Pan, W.4    Wang, X.5
  • 24
    • 0031017250 scopus 로고    scopus 로고
    • Atenolol gastrointestinal therapeutic system. I. Screening of formulation variables
    • Sastry SV, DeGennaro MD, Reddy IK, Khan MA. Atenolol gastrointestinal therapeutic system. I. Screening of formulation variables. Drug Dev. Ind. Pharm. 1997;23(2):157-165.
    • (1997) Drug Dev. Ind. Pharm. , vol.23 , Issue.2 , pp. 157-165
    • Sastry, S.V.1    DeGennaro, M.D.2    Reddy, I.K.3    Khan, M.A.4
  • 26
    • 35348941520 scopus 로고
    • Osmotic devices having composite walls
    • US Patent 4,077,407
    • Theeuwes F,Ayer AD. Osmotic devices having composite walls US Patent 4,077,407, 1978.
    • (1978)
    • Theeuwes, F.1    Ayer, A.D.2
  • 30
    • 0031742446 scopus 로고    scopus 로고
    • Controlled, multidose, pharmacokinetic evaluation of two extended-release carbamazepine formulations (Carbatrol and Tegretol-XR)
    • Stevens RE, Limsakun T, Evans G, Mason DH, Jr. Controlled, multidose, pharmacokinetic evaluation of two extended-release carbamazepine formulations (Carbatrol and Tegretol-XR). J. Pharm. Sci. 1998;87(12):1531-1534.
    • (1998) J. Pharm. Sci. , vol.87 , Issue.12 , pp. 1531-1534
    • Stevens, R.E.1    Limsakun, T.2    Evans, G.3    Mason Jr, D.H.4
  • 31
    • 0027318239 scopus 로고
    • Effects of plasticizers on water permeation and mechanical properties of cellulose acetate: antiplasticization in slightly plasticized polymer film
    • Guo JH. Effects of plasticizers on water permeation and mechanical properties of cellulose acetate: antiplasticization in slightly plasticized polymer film. Drug Dev. Ind. Pharm. 1993;19(13):1541-1545.
    • (1993) Drug Dev. Ind. Pharm. , vol.19 , Issue.13 , pp. 1541-1545
    • Guo, J.H.1
  • 32
    • 0347572406 scopus 로고    scopus 로고
    • Effects of polyethylene glycol on morphology, thermomechanical properties, and water vapor permeability of cellulose acetate-free films
    • 64, 66, 68, 70, 72, 74
    • Yuan J, Shang PP, Wu SH. Effects of polyethylene glycol on morphology, thermomechanical properties, and water vapor permeability of cellulose acetate-free films. Pharm. Technol. North Am. 2001;25(10):62, 64, 66, 68, 70, 72, 74.
    • (2001) Pharm. Technol. North Am. , vol.25 , Issue.10 , pp. 62
    • Yuan, J.1    Shang, P.P.2    Wu, S.H.3
  • 33
    • 39549106484 scopus 로고    scopus 로고
    • Preparation of bilayer-core osmotic pump tablet by coating the indented core tablet
    • Liu L, Xu X. Preparation of bilayer-core osmotic pump tablet by coating the indented core tablet. Int. J. Pharm. 2008; 352 (1-2):225-230.
    • (2008) int. J. Pharm. , Issue.1-2 , pp. 225-230
    • Liu, L.1    Xu, X.2
  • 34
    • 0028902188 scopus 로고
    • Compression behavior and tensile strength of heat-treated polyethylene glycols
    • Lin C-W, Cham T-M. Compression behavior and tensile strength of heat-treated polyethylene glycols. Int. J. Pharm. 1995;118:169-179.
    • (1995) Int. J. Pharm. , vol.118 , pp. 169-179
    • Lin, C.-W.1    Cham, T.-M.2
  • 35
    • 0029826865 scopus 로고    scopus 로고
    • Characterization of compressibility and compactibility of poly(ethylene oxide) polymers for modified release application by compaction simulator
    • Yang L, Venkatesh G, Fassihi R. Characterization of compressibility and compactibility of poly(ethylene oxide) polymers for modified release application by compaction simulator. J. Pharm. Sci. 1996;85(10):1085-1090.
    • (1996) J. Pharm. Sci. , vol.85 , Issue.10 , pp. 1085-1090
    • Yang, L.1    Venkatesh, G.2    Fassihi, R.3
  • 36
    • 0030919390 scopus 로고    scopus 로고
    • Compaction simulator study of a novel triple-layer tablet matrix for industrial tableting
    • Yang L,Venkatesh G, Fassihi R. Compaction simulator study of a novel triple-layer tablet matrix for industrial tableting. Int. J. Pharm. 1997;152(1):45-52.
    • (1997) Int. J. Pharm. , vol.152 , Issue.1 , pp. 45-52
    • Yang, L.1    Venkatesh, G.2    Fassihi, R.3
  • 37
    • 0013858092 scopus 로고
    • Compression and dry granulation
    • Jaminet F, Hess H. Compression and dry granulation. Pharm. Acta Helv. 1966;41(1):39-58.
    • (1966) Pharm. Acta Helv. , vol.41 , Issue.1 , pp. 39-58
    • Jaminet, F.1    Hess, H.2
  • 38
    • 0036183094 scopus 로고    scopus 로고
    • Effect of molecular mass on the melting temperature, enthalpy and entropy of hydroxy-terminated PEO
    • Sanchez-Soto PJ, Gines JM, Arias MJ, Novak C, Ruiz-Conde A. Effect of molecular mass on the melting temperature, enthalpy and entropy of hydroxy-terminated PEO. J. Therm. Anal. Calorim. 2002;67(1):189-197.
    • (2002) J. Therm. Anal. Calorim. , vol.67 , Issue.1 , pp. 189-197
    • Sanchez-Soto, P.J.1    Gines, J.M.2    Arias, M.J.3    Novak, C.4    Ruiz-Conde, A.5
  • 39
    • 0022975569 scopus 로고
    • Osmotically controlled drug delivery systems produced from organic solutions and aqueous dispersions of cellulose acetate
    • Bindschaedler C, Gurny R, Doelker E. Osmotically controlled drug delivery systems produced from organic solutions and aqueous dispersions of cellulose acetate. J. Control. Release 1986;4(3):203-212.
    • (1986) J. Control. Release , vol.4 , Issue.3 , pp. 203-212
    • Bindschaedler, C.1    Gurny, R.2    Doelker, E.3
  • 40
    • 0026600895 scopus 로고
    • Evaluation of a cellulose acetate (ca) latex as coating material for controlled release products
    • Kelbert M, Bechard SR. Evaluation of a cellulose acetate (ca) latex as coating material for controlled release products. Drug Dev. Ind. Pharm. 1992;18(5):519-538.
    • (1992) Drug Dev. Ind. Pharm. , vol.18 , Issue.5 , pp. 519-538
    • Kelbert, M.1    Bechard, S.R.2
  • 41
    • 14644404381 scopus 로고    scopus 로고
    • A thermodynamic model for organic and aqueous tablet film coating
    • Am Ende MT, Berchielli A. A thermodynamic model for organic and aqueous tablet film coating. Pharm. Dev. Technol. 2005;10(1):47-58.
    • (2005) Pharm. Dev. Technol. , vol.10 , Issue.1 , pp. 47-58
    • Am Ende, M.T.1    Berchielli, A.2
  • 43
    • 33646412301 scopus 로고    scopus 로고
    • Raman spectroscopy for tablet coating thickness quantification and coating characterization in the presence of strong fluorescent interference
    • Romero-Torres S, Perez-Ramos JD, Morris KR, Grant ER. Raman spectroscopy for tablet coating thickness quantification and coating characterization in the presence of strong fluorescent interference. J. Pharm. Biomed. Anal. 2006;41(3): 811-819.
    • (2006) J. Pharm. Biomed. Anal. , vol.41 , Issue.3 , pp. 811-819
    • Romero-Torres, S.1    Perez-Ramos, J.D.2    Morris, K.R.3    Grant, E.R.4
  • 47
    • 0002667968 scopus 로고
    • Stability of the polyoxyethylene chain
    • Nonionic Surfactants
    • DonbrowM. Stability of the polyoxyethylene chain. Surfactant Sci. Ser. 1987;23(Nonionic Surfactants):1011-1072.
    • (1987) Surfactant Sci. Ser. , vol.23 , pp. 1011-1072
    • Donbrow, M.1
  • 48
    • 0030862261 scopus 로고    scopus 로고
    • Thermal/oxidative degradation and stabilization of polyethylene glycol
    • Han S, Kim C, Kwon D. Thermal/oxidative degradation and stabilization of polyethylene glycol. Polymer 1997;38: 317-323.
    • (1997) Polymer , vol.38 , pp. 317-323
    • Han, S.1    Kim, C.2    Kwon, D.3
  • 49
    • 84885566198 scopus 로고
    • Oxidative degradation of polymers and organic compounds via unimolecular decomposition of peroxy radicals
    • Marchal J. Oxidative degradation of polymers and organic compounds via unimolecular decomposition of peroxy radicals. Cent. Rech. Macromol., CNRS 1972.
    • (1972) Cent. Rech. Macromol.CNR
    • Marchal, J.1
  • 50
    • 14644399287 scopus 로고    scopus 로고
    • Use of the antioxidant BHT in asymmetric membrane tablet coatings to stabilize the core to the acid catalyzed peroxide oxidation of a thioether drug
    • Puz MJ, Johnson BA, Murphy BJ. Use of the antioxidant BHT in asymmetric membrane tablet coatings to stabilize the core to the acid catalyzed peroxide oxidation of a thioether drug. Pharm. Dev. Technol. 2005;10(1):115-125.
    • (2005) Pharm. Dev. Technol. , vol.10 , Issue.1 , pp. 115-125
    • Puz, M.J.1    Johnson, B.A.2    Murphy, B.J.3
  • 51
    • 0014350683 scopus 로고
    • Solubilization of griseofulvin by nonionic surfactants
    • Elworthy PH, Lipscomb FJ. Solubilization of griseofulvin by nonionic surfactants. J. Pharm. Pharmacol. 1968;20(11): 817-824.
    • (1968) J. Pharm. Pharmacol. , vol.20 , Issue.11 , pp. 817-824
    • Elworthy, P.H.1    Lipscomb, F.J.2
  • 52
    • 55049133105 scopus 로고    scopus 로고
    • Pharmaceutical development of solid dispersion based osmotic drug delivery system for nifedipine
    • Kanagale P, Patel V, Venkatesan N, Jain M, Patel P, Misra A. Pharmaceutical development of solid dispersion based osmotic drug delivery system for nifedipine. Curr. Drug Deliv. 2008;5 (4):306-311.
    • (2008) Curr. Drug Deliv. , vol.5 , Issue.4 , pp. 306-311
    • Kanagale, P.1    Patel, V.2    Venkatesan, N.3    Jain, M.4    Patel, P.5    Misra, A.6
  • 53
    • 0028340095 scopus 로고
    • Physical characteristics and dissolution kinetics of solid dispersions of ketoprofen and polyethylene glycol 6000
    • MargaritMV, Rodriguez IC, Cerezo A. Physical characteristics and dissolution kinetics of solid dispersions of ketoprofen and polyethylene glycol 6000. Int. J. Pharm. 1994;108(2): 101-107.
    • (1994) Int. J. Pharm. , vol.108 , Issue.2 , pp. 101-107
    • Margarit, M.V.1    Rodriguez, I.C.2    Cerezo, A.3
  • 55
    • 60349129366 scopus 로고    scopus 로고
    • Preparation and thermal characterization of poly(ethylene oxide)/griseofulvin solid dispersions for biomedical applications
    • Stachurek I, Pielichowski K. Preparation and thermal characterization of poly(ethylene oxide)/griseofulvin solid dispersions for biomedical applications. J. Appl. Polym. Sci. 2009; 111(4):1690-1696.
    • (2009) J. Appl. Polym. Sci. , vol.111 , Issue.4 , pp. 1690-1696
    • Stachurek, I.1    Pielichowski, K.2
  • 56
    • 3543091054 scopus 로고    scopus 로고
    • Solid state NMR perspective of drug-polymer solid solutions: a model system based on poly(ethylene oxide)
    • Schachter DM, Xiong J, Tirol GC. Solid state NMR perspective of drug-polymer solid solutions: a model system based on poly(ethylene oxide). Int. J. Pharm. 2004;281(1-2): 89-101.
    • (2004) Int. J. Pharm. , vol.281 , Issue.1-2 , pp. 89-101
    • Schachter, D.M.1    Xiong, J.2    Tirol, G.C.3
  • 57
    • 52449113421 scopus 로고    scopus 로고
    • Spontaneous crystallinity loss of drugs in the disordered regions of poly(ethylene oxide) in the presence of water
    • Marsac PJ, Romary DP, Shamblin SL, Baird JA, Taylor LS. Spontaneous crystallinity loss of drugs in the disordered regions of poly(ethylene oxide) in the presence of water. J. Pharm. Sci. 2008;97(8):3182-3194.
    • (2008) J. Pharm. Sci. , vol.97 , Issue.8 , pp. 3182-3194
    • Marsac, P.J.1    Romary, D.P.2    Shamblin, S.L.3    Baird, J.A.4    Taylor, L.S.5
  • 58
    • 2442680307 scopus 로고    scopus 로고
    • Polyethylene oxides: protection potential against polymorphic transitions of drugs
    • Schmidt AG, Wartewig S, Picker KM. Polyethylene oxides: protection potential against polymorphic transitions of drugs?. J. Raman Spectrosc. 2004;35(5):360-367.
    • (2004) J. Raman Spectrosc. , vol.35 , Issue.5 , pp. 360-367
    • Schmidt, A.G.1    Wartewig, S.2    Picker, K.M.3
  • 59
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals
    • Hancock BC, Parks M. What is the true solubility advantage for amorphous pharmaceuticals?. Pharm. Res. 2000;17(4): 397-404.
    • (2000) Pharm. Res. , vol.17 , Issue.4 , pp. 397-404
    • Hancock, B.C.1    Parks, M.2
  • 60
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and significance of the amorphous state in pharmaceutical systems
    • Hancock BC, Zografi G. Characteristics and significance of the amorphous state in pharmaceutical systems. J. Pharm. Sci. 1997;86:1-12.
    • (1997) J. Pharm. Sci. , vol.86 , pp. 1-12
    • Hancock, B.C.1    Zografi, G.2
  • 64
    • 33846242938 scopus 로고    scopus 로고
    • Evaluation of various properties of alternative salt forms of sulfobutylether-b-cyclodextrin, (SBE)7M-b-CD
    • Sotthivirat S, Haslam JL, Stella VJ. Evaluation of various properties of alternative salt forms of sulfobutylether-b-cyclodextrin, (SBE)7M-b-CD. Int. J. Pharm. 2007;330(1-2):73-81.
    • (2007) Int. J. Pharm. , vol.330 , Issue.1-2 , pp. 73-81
    • Sotthivirat, S.1    Haslam, J.L.2    Stella, V.J.3
  • 65
    • 0032779325 scopus 로고    scopus 로고
    • Release of testosterone from an osmotic pump tablet utilizing (SBE)7M-beta-cyclodextrin as both a solubilizing and an osmotic pump agent
    • Okimoto K, Rajewski RA, Stella VJ. Release of testosterone from an osmotic pump tablet utilizing (SBE)7M-beta-cyclodextrin as both a solubilizing and an osmotic pump agent. J. Control. Release 1999;58(1):29-38.
    • (1999) J. Control. Release , vol.58 , Issue.1 , pp. 29-38
    • Okimoto, K.1    Rajewski, R.A.2    Stella, V.J.3


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