Synthesis and characterisation of a novel tubulin-directed DO3A-colchicine conjugate with potential theranostic features

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 11, 2011, Pages 3346-3348

  Wardle, Nicholas J ^a   Kalber, Tammy ^b   Bell, Jimmy D ^b   Bligh, S W Annie ^a  

^a LONDON METROPOLITAN UNIVERSITY   (United Kingdom)

^b HAMMERSMITH HOSPITAL   (United Kingdom)

Author keywords

Colchicine; Contrast agent; Gadolinium; Magnetic resonance imaging; Tubulin

Indexed keywords

COLCHICINE DERIVATIVE; DEACETYLCOLCHICINE; GADOTERIDOL; PROTON;

ARTICLE; CARCINOMA CELL; DRUG BINDING; DRUG EFFICACY; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; IN VITRO STUDY; OVARY CARCINOMA;

CELL LINE, TUMOR; COLCHICINE; FEMALE; HUMANS; MOLECULAR STRUCTURE; ORGANOMETALLIC COMPOUNDS; OVARIAN NEOPLASMS; TUBULIN;

EID: 79956118061     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.04.014     Document Type: Article

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