Exploration of dimensions of estrogen potency: Parsing ligand binding and coactivator binding affinities

Journal of Biological Chemistry

Volumn 286, Issue 15, 2011, Pages 12971-12982

  Jeyakumar, M ^a   Carlson, Kathryn E ^a   Gunther, Jillian R ^a   Katzenellenbogen, John A ^a  

^a UNIVERSITY OF ILLINOIS AT URBANA CHAMPAIGN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING AFFINITIES; CELLULAR RESPONSE; COACTIVATORS; ESTROGEN RECEPTOR; GOOD CORRELATIONS; HIGH AFFINITY; HORMONE BINDING; IN-CELL; IN-VITRO; LIGAND BINDING; LIGAND BINDING AFFINITY; LIGAND BINDING DOMAIN; LIGAND COMPLEXES; MOLECULAR BASIS; MOLECULAR EVENTS; RECEPTOR BINDING; REGULATED TRANSCRIPTION FACTORS; TARGET CELLS; TARGET TISSUES; THREE PARAMETERS; TIME-RESOLVED;

BINDING ENERGY; COMPLEXATION; EMPLOYMENT; GENES; TRANSCRIPTION; TRANSCRIPTION FACTORS;

LIGANDS;

17ALPHA ESTRADIOL; CONJUGATED ESTROGEN; DIETHYLSTILBESTROL; DIMETHYLSTILBESTROL; EQUILENIN; ESTRADIOL; ESTRIOL; ESTROGEN; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; ESTRONE; GENISTEIN; STEROID RECEPTOR COACTIVATOR 3;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; FLUORESCENCE RESONANCE ENERGY TRANSFER; HORMONE ACTION; HORMONE RECEPTOR INTERACTION; IN VITRO STUDY; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN EXPRESSION; QUANTITATIVE ANALYSIS;

CELL LINE; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; ESTROGENS; HUMANS; LIGANDS; NUCLEAR RECEPTOR COACTIVATORS; PROTEIN BINDING; PROTEIN STRUCTURE, QUATERNARY; PROTEIN STRUCTURE, TERTIARY;

EID: 79953905621     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M110.205112     Document Type: Article

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