In vitro and in vivo antiparasital activity against Trypanosoma cruzi of three novel 5-methyl-1,2,4-triazolo[1,5-a]pyrimidin-7(4H)-one-based complexes

Journal of Inorganic Biochemistry

Volumn 105, Issue 6, 2011, Pages 770-776

  Caballero, Ana B ^a   Marín, Clotilde ^a   Rodríguez Diéguez, Antonio ^a   Ramírez Macías, Inmaculada ^a   Barea, Elisa ^a   Sánchez Moreno, Manuel ^a   Salas, Juan M ^a  

^a UNIVERSITY OF GRANADA   (Spain)

Author keywords

Biological properties; Coordination chemistry; Trypanosoma cruzi

Indexed keywords

5 METHYL 1,2,4 TRIAZOLO[1,5 A]PYRIMIDIN 7 (4H) ONE; ANTIPARASITIC AGENT; BENZNIDAZOLE; COPPER COMPLEX; PYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

AMASTIGOTE; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CELL ASSAY; CELL DIVISION; CHAGAS DISEASE; CONTROLLED STUDY; DRUG EFFECT; FEMALE; GROWTH INHIBITION; HYDROGEN BOND; IC 50; IN VITRO STUDY; IN VIVO STUDY; INFECTION RATE; METABOLITE; MOUSE; NONHUMAN; PARASITEMIA; PARASITOSIS; SURVIVAL; TREATMENT DURATION; TRYPANOSOMA CRUZI;

ANIMALS; CERCOPITHECUS AETHIOPS; CHAGAS DISEASE; COORDINATION COMPLEXES; CRYSTALLOGRAPHY, X-RAY; FEMALE; LIGANDS; MICE; MICE, INBRED BALB C; MICROSCOPY, ELECTRON, TRANSMISSION; NITROIMIDAZOLES; PERCHLORIC ACID; PYRIMIDINONES; TRIAZOLES; TRYPANOCIDAL AGENTS; TRYPANOSOMA CRUZI; VERO CELLS;

TRYPANOSOMA CRUZI;

EID: 79953879784     PISSN: 01620134     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jinorgbio.2011.03.015     Document Type: Article

References (35)

1. J.A.R. Navarro, B. Lippert, Coord. Chem. Rev. 185-186 (1999) 653-667.
2. J.A.R. Navarro, E. Barea, M.A. Galindo, J.M. Salas, M.A. Romero, M. Quirós, N. Masciocchi, S. Galli, A. Sironi, B. Lippert, J. Solid State Chem. 178 (2005) 2436-2451.
3. A. Rodríguez-Diéguez, J. Cano, R. Kivekäs, A. Debdoubi, E. Colacio, Inorg. Chem. 46 (2007) 2503-2510.
4. A. Rodríguez-Diéguez, H. Aouryaghal, A.J. Mota, E. Colacio, Acta Cryst E64 (2008) m618/1-m618/7.
5. J. Suárez-Varela, A.J. Mota, H. Aouryaghal, J. Cano, A. Rodríguez-Diéguez, D. Luneau, E. Colacio, Inorg. Chem. 47 (2008) 8143-8158.
6. A.B. Caballero, A. Rodríguez-Diéguez, E. Barea, M. Quirós, J.M. Salas, Cryst Eng Comm 12 (2010) 3038-3045.
7. J.M. Salas, M.A. Romero, M.P. Sánchez, M. Quirós, Coord. Chem. Rev. 193-195 (1999) 1119-1142.
8. R. Gujjar, A. Marwaha, F. El Mazouni, J. White, K.L. White, S. Creason, D.M. Shackleford, J. Baldwin, W.N. Charman, F.S. Buckner, S. Charman, P.K. Rathod, M.A. Phillips, J. Med. Chem. 52 (2009) 1864-1872.
9. W. Tang, D.Q. Shi, J. Heterocycl, Chem 47 (2010) 162-166.
10. Q. Chen, Z.M. Liu, C.N. Chen, L.L. Jiang, G.F. Yang, Chem. Biodivers. 6 (2009) 1254-1265.
11. N.A. El-Koussi, F.A. Omar, S.A. Abdel-Aziz, M.F. Radwan, Bull. Pharm. Sci. 27 (1) (2004) 141-154.
12. R.P. Srivastava, V.V. Kumar, S. Bhatia, S. Sharma, Indian J. Chem. (Sect. B) 34B (3) (1995) 209-214.
13. E. Bakhite, A. Ghafar, A. Pharmazie 50 (1) (1995) 33-35.
14. G. Fischer, Adv. Heterocycl. Chem. 95 (2008) 143-219.
15. I. Lakomska, A. Wojtczak, J. Sitkowski, L. Kozerski, E. Szlyk, Polyhedron 27 (2008) 2765-2770.
16. I. Lakomska, Inorg. Chim. Acta 362 (2009) 669-681.
17. F. Luque, C. Fernández-Ramos, E. Entrala, M.J. Rosales, C. Marín, J.M. Salas, J.A.R. Navarro, M. Sánchez-Moreno, Toxicol. In Vitro 14 (2000) 487-495.
18. F. Luque, C. Fernández-Ramos, E. Entrala, M.J. Rosales, J.A.R. Navarro, M.A. Romero, J.M. Salas, M. Sánchez-Moreno, Comp. Biochem. Phys. C 126 (2000) 39-44.
19. R. Magán, C. Marín, M.J. Rosales, M.A. Barrera, J.M. Salas, M. Sánchez-Moreno, Pharmacology 70 (2004) 83-90.
20. R. Magán, C. Marín, M.J. Rosales, J.M. Salas, M. Sánchez-Moreno, Pharmacology 73 (2005) 41-48.
21. S. Boutaleb-Charki, C. Marín, C.R. Maldonado, M.J. Rosales, J. Urbano, R. Gutiérrez- Sánchez, M. Quirós, J.M. Salas, M. Sánchez-Moreno, Drug Metab. Lett. 3 (2009) 35-44.
22. C. Maldonado, C. Marín, F. Olmo, O. Huertas, M. Quirós, M. Sánchez-Moreno, M.J. Rosales, J.M. Salas, J. Med. Chem. 53 (2010) 6969-6972.
23. J.C. Pinto-Dias, Ann. Intern. Med. 144 (2006) 772-774.
24. J.A.R. Navarro, J.M. Salas, M.A. Romero, R. Vilaplana, F. González-Vílchez, R. Faure, J. Med. Chem. 41 (1998) 332-338.
25. I. Lakomska, J. Biol. Inorg. Chem. 12 (Suppl.1) (2007) S37-PO52.
26. J. Ruiz, M.D. Villa, N. Cutillas, G. López, C. de Haro, D. Bautista, V. Moreno, L. Valencia, Inorg. Chem. 47 (2008) 4490-4505.
27. A.B. Caballero, A. Rodríguez-Diéguez, L. Lezama, E. Barea, J.M. Salas, Dalton Trans. (2011) (in press, doi:10.1039/C0DT01416H).
28. F. Luque, C. Fernández-Ramos, E. Entrala, M.J. Rosales, J.A.R. Navarro, M.A. Romero, J.M. Salas-Peregrín, M. Sánchez-Moreno, Comp. Biochem. Physiol. 126 (2000) 39-44.
29. P. González, C. Marín, I. Rodríguez-González, A.B. Hitos, M.J. Rosales, M. Reina, J.G. Díaz, A. González- Coloma, M. Sánchez-Moreno, Int. J. Antimicrob. Agents 25 (2005) 136-141.
30. C. Fernández-Becerra, M. Sánchez-Moreno, A. Osuna, F.R. Opperdoes, J. Eukaryotic, Microbiology 44 (1997) 523-529.
31. S. Boutaleb-Charki, C. Marín, C.R. Maldonado, M.J. Rosales, J. Urbano, R. Gutiérrez-Sánchez, M. Quirós, J.M. Salas, M. Sánchez-Moreno, Drug Metab. Lett. 3 (2009) 35-44.
32. C. França da Silva, M.M. Batista, D.G.J. Batista, E. Mello de Souza, P. Bernardino da Silva, G. Melo de Oliveira, A.S. Meuser, A.R. Shareef, D.W. Boykin, M.N.C. Soeiro, Antimicrob. Agents Chemother. 52 (2008) 3307-3314.
33. E.M. de Souza, G.M. Oliveira, M.N.C. Soeiro, Drug Target Insights 2 (2007) 61-69.
34. F. Bringaud, L. Rivière, V. Coustou, Mol. Biochem. Parasitol. 149 (2006) 1-9.
35. I. Ramírez-Macías, C. Marín, J.M. Salas, A. Caballero, M.J. Rosales, N. Villegas, A. Rodríguez-Diéguez, E. Barea, M. Sánchez-Moreno, J. Antimicrob. Chemother. 66 (2011) 813-819.