SCOPUS 정보 검색 플랫폼

Volumn 6, Issue 4, 2011, Pages 1048-1056

A strategy for neuraminidase inhibitors using mechanism-based labeling information

(16) Hinou, Hiroshi a Miyoshi, Risho a Takasu, Yasuaki a Kai, Hirokazu a Kurogochi, Masaki a Arioka, Shingo b Gao, Xiao Dong a Miura, Nobuaki a Fujitani, Naoki a Omoto, Shinya b Yoshinaga, Tomokazu b Fujiwara, Tamio b Noshi, Takeshi b Togame, Hiroko b Takemoto, Hiroshi b Nishimura, Shin Ichiro a

a HOKKAIDO UNIVERSITY (Japan)

b SHIONOGI AND CO LTD (Japan)

Author keywords

drug design; hydrolases; inhibitors; sialic acid; structure activity relationship

Indexed keywords

COMBINED STRUCTURE; DRUG DESIGN; HIGH SELECTIVITY; INHIBITION PROPERTY; INHIBITORS; LINEWEAVER-BURK PLOTS; LOOP STRUCTURE; MECHANISM-BASED LABELING; N-ACETYLNEURAMINIC ACID; NEURAMINIDASE; POTENT INHIBITION; POTENT INHIBITOR; SIALIC ACIDS; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTITUTION GROUPS; VALIDATION STUDY; VIBRIO CHOLERAE;

AMINO ACIDS; CARBOXYLIC ACIDS; DESIGN; ENZYMES; HYDROLASES;

INFORMATION USE;

ENZYME INHIBITOR; SIALIC ACID DERIVATIVE; SIALIDASE;

ARTICLE; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; ENZYME ACTIVE SITE; ENZYMOLOGY; METABOLISM; PROTEIN TERTIARY STRUCTURE; STRUCTURE ACTIVITY RELATION; VIBRIO CHOLERAE;

CATALYTIC DOMAIN; DRUG DESIGN; ENZYME INHIBITORS; NEURAMINIDASE; PROTEIN STRUCTURE, TERTIARY; SIALIC ACIDS; STRUCTURE-ACTIVITY RELATIONSHIP; VIBRIO CHOLERAE;

EID: 79953039574 PISSN: 18614728 EISSN: 1861471X Source Type: Journal
DOI: 10.1002/asia.201000594 Document Type: Article

Times cited : (10)

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