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Volumn 6, Issue 3, 2011, Pages 550-560

Design and Synthesis of Novel Cyclooxygenase-1 Inhibitors as Analgesics: 5-Amino-2-ethoxy-N-(substituted-phenyl)benzamides

(6) Fukai, Ryosuke a Zheng, Xiaoxia a Motoshima, Kazunori a Tai, Akihiro b Yazama, Futoshi b Kakuta, Hiroki a

a OKAYAMA UNIVERSITY (Japan)

b PREFECTURAL UNIVERSITY OF HIROSHIMA (Japan)

Author keywords

Analgesics; Cyclooxygenase 1; Gastric damage; Inhibitors; Phenylbenzamides

Indexed keywords

5 AMINO 2 ETHOXY N (2 METHOXYPHENYL)BENZAMIDE; 5 AMINO 2 ETHOXY N (3 TRIFLUOROMETHYLPHENYL)BENZAMIDE; ANALGESIC AGENT; CYCLOOXYGENASE 1 INHIBITOR; INDOMETACIN; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT; STOMACH INJURY; WRITHING TEST;

ANALGESICS; ANIMALS; BENZAMIDES; BINDING SITES; COMPUTER SIMULATION; CYCLOOXYGENASE 1; CYCLOOXYGENASE INHIBITORS; DRUG DESIGN; EDEMA; MALE; MICE;

EID: 79952092559 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000462 Document Type: Article

Times cited : (8)

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