Simple phosphonic inhibitors of human neutrophil elastase

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 5, 2011, Pages 1310-1314

  Sieńczyk, Marcin ^a   Winiarski, Łukasz ^a   Kasperkiewicz, Paulina ^a   Psurski, Mateusz ^a,b   Wietrzyk, Joanna ^b   Oleksyszyn, Józef ^a  

^a WROCLAW UNIVERSITY OF TECHNOLOGY   (Poland)

^b INSTITUTE OF IMMUNOLOGY AND EXPERIMENTAL THERAPY   (Poland)

Author keywords

Aminoalkylphosphonates; Cancer cells; Human neutrophil elastase; Irreversible inhibition; Serine protease inhibitors

Indexed keywords

ALPHA AMINOALKYLPHOSPHONATE DIARYL ESTER; ALPHA AMINOPHOSPHONATE DIARYL ESTER; CHYMOTRYPSIN; LEUKOCYTE ELASTASE; LEUKOCYTE ELASTASE INHIBITOR; PANCREATIC ELASTASE; PHOSPHONIC ACID DERIVATIVE; SERINE PROTEINASE; TRYPSIN; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; ESTERS; HUMANS; LEUKOCYTE ELASTASE; LUNG NEOPLASMS; MOLECULAR STRUCTURE; PHOSPHONIC ACIDS;

SUS;

EID: 79951727060     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.01.083     Document Type: Article

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