Comparative pharmacology of human β-adrenergic receptor subtypes - Characterization of stably transfected receptors in CHO cells

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 369, Issue 2, 2004, Pages 151-159

  Hoffmann, C ^a   Leitz, M R ^a   Oberdorf Maass, S ^a   Lohse, M J ^a   Klotz, K N ^a  

^a UNIVERSITY OF WÜRZBURG   (Germany)

Author keywords

2 receptor; Adrenergic receptor; 1 receptor; 3 receptor; Antagonist; G protein coupled receptors; Inverse agonist; Stable transfection

Indexed keywords

1 (2 ETHYLPHENOXY) 3 (1,2,3,4 TETRAHYDRO 1 NAPHTHYLAMINO) 2 PROPANOL OXALATE; 3 ISOPROPYLAMINO 1 (7 METHYL 4 INDANYLOXY) 2 BUTANOL; 4 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY) 2 BENZIMIDAZOLONE; 4 [2 [[2 (3 CHLOROPHENYL) 2 HYDROXYETHYL]AMINO]PROPYL]PHENOXYACETIC ACID; 5 [2 [[2 HYDROXY 3 [4 (1 METHYL 4 TRIFLUOROMETHYL 2 IMIDAZOLYL)PHENOXY]PROPYL]AMINO]ETHOXY]SALICYLAMIDE; ADENYLATE CYCLASE; ADRENALIN; ALPRENOLOL; ATENOLOL; BETA ADRENERGIC RECEPTOR; BISOPROLOL; BROXATEROL; CARVEDILOL; CYANOPINDOLOL I 125; FENOTEROL; FORMOTEROL; ISOPRENALINE; METOPROLOL; NORADRENALIN; PINDOLOL; PROPRANOLOL; RADIOLIGAND; RECEPTOR SUBTYPE; SALBUTAMOL; SALMETEROL; TERBUTALINE;

ANIMAL CELL; ARTICLE; CELL ISOLATION; CELL MEMBRANE; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; ENZYME ACTIVITY; GENETIC TRANSFECTION; ISOTOPE LABELING; NONHUMAN; PROTEIN EXPRESSION; RECEPTOR AFFINITY;

ADENYLATE CYCLASE; ADRENERGIC BETA-AGONISTS; ADRENERGIC BETA-ANTAGONISTS; ANIMALS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; CRICETULUS; HUMANS; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, BETA; TRANSFECTION;

EID: 1442349847     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00210-003-0860-y     Document Type: Article

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