Stilbene derivatives as human 5-HT6 receptor antagonists from the root of Caragana sinica

Biological and Pharmaceutical Bulletin

Volumn 33, Issue 12, 2010, Pages 2024-2028

  Kim, Dong Hyuk ^a,b   Kim, Soon Hee ^a   Kim, Hyoung Ja ^a   Jin, Changbae ^a   Chung, Kwang Chul ^b   Rhim, Hyewhon ^a  

^a Korea Institute of Science and Technology   (South Korea)

^b Yonsei University   (South Korea)

Author keywords

Caragana sinica; Extracellular signal regulated kinase 1 2; FDSS6000; Intracellular Ca2+; Serotonin; Stilbene derivative

Indexed keywords

ACETIC ACID ETHYL ESTER; ALPHA VINIFERIN; CARAGANA SINICA EXTRACT; MITOGEN ACTIVATED PROTEIN KINASE 1; MITOGEN ACTIVATED PROTEIN KINASE 3; MIYABENOL C; PALLIDOL; PLANT EXTRACT; SEROTONIN 6 ANTAGONIST; SEROTONIN 6 RECEPTOR; STILBENE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CARAGANA; CARAGANA SINICA; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG DETERMINATION; DRUG ISOLATION; DRUG MECHANISM; DRUG SCREENING; DRUG SELECTIVITY; ENZYME PHOSPHORYLATION; FRACTIONATION; HUMAN; HUMAN CELL; IC 50; PLANT ROOT; RECEPTOR BLOCKING; STABLE EXPRESSION;

CARAGANA; HEK293 CELLS; HELA CELLS; HUMANS; MITOGEN-ACTIVATED PROTEIN KINASE 3; PLANT EXTRACTS; PLANT ROOTS; POLYCYCLIC COMPOUNDS; SEROTONIN; SEROTONIN ANTAGONISTS; STILBENES;

EID: 78751509219     PISSN: 09186158     EISSN: 13475215     Source Type: Journal    
DOI: 10.1248/bpb.33.2024     Document Type: Article

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