메뉴 건너뛰기




Volumn 15, Issue 12, 2010, Pages 9174-9183

Synthesis and biological activity of trans-tiliroside derivatives as potent anti-diabetic agents

Author keywords

Anti diabetic activity; Derivative synthesis; Novozyme435; Trans tiliroside

Indexed keywords

ANTIDIABETIC AGENT; FLAVONOID; GLUCOSE; METFORMIN; TILIROSIDE;

EID: 78650647699     PISSN: None     EISSN: 14203049     Source Type: Journal    
DOI: 10.3390/molecules15129174     Document Type: Article
Times cited : (33)

References (29)
  • 3
    • 0036170309 scopus 로고    scopus 로고
    • Molecular modeling of protein tyrosine phosphatase 1B (PTP 1B) inhibitors
    • Murthy, V.S.; Kulkarni, V.M. Molecular modeling of protein tyrosine phosphatase 1B (PTP 1B) inhibitors. Bioorg. Med. Chem. 2002, 10, 897-906.
    • (2002) Bioorg. Med Chem. , vol.10 , pp. 897-906
    • Murthy, V.S.1    Kulkarni, V.M.2
  • 4
    • 0036336284 scopus 로고    scopus 로고
    • Synthesis and biological activity of a novel class of pyridazine analogues as non-competitive reversible inhibitors of protein tyrosine phosphatase 1B (PTP1B)
    • DOI 10.1016/S0968-0896(02)00176-1, PII S0968089602001761
    • Liljebris, C.; Martinsson, J.; Tedenborg, L.; Williams, M.; Barker, E.; Duffy, J.E.S.; Nygren, A.; James, S. Synthesis and biological activity of a novel class of pyridazine analogues non-competitive reversible inhibitors of protein tyrosine phosphatase 1B (PTP 1B). Bioorg. Med. Chem. 2002, 10, 3197-3212. (Pubitemid 34855393)
    • (2002) Bioorganic and Medicinal Chemistry , vol.10 , Issue.10 , pp. 3197-3212
    • Liljebris, C.1    Martinsson, J.2    Tedenborg, L.3    Williams, M.4    Barker, E.5    Duffy, J.E.S.6    Nygren, A.7    James, S.8
  • 5
    • 33748791911 scopus 로고    scopus 로고
    • Efficacy of Potentilla chinesis in patients with type 2 diabetes mellitus
    • Ma, Y.; Wen, S.Z. Efficacy of Potentilla chinesis in patients with type 2 diabetes mellitus. Chin. Trad. Herb. Drugs 2002, 33, 644-644.
    • (2002) Chin. Trad. Herb. Drugs , vol.33 , pp. 644-644
    • Ma, Y.1    Wen, S.Z.2
  • 6
    • 41749105985 scopus 로고    scopus 로고
    • Study on anti-diabetes active fraction and consituents from Potentilla Chinesis
    • Zhao, C.; Qiao, W.; Zhang, Y.W.; Lu, B.; Duan, H.Q. Study on anti-diabetes active fraction and consituents from Potentilla Chinesis. J .Chin. Mater. Med. 2008, 33, 680-682.
    • (2008) J .Chin. Mater. Med. , vol.33 , pp. 680-682
    • Zhao, C.1    Qiao, W.2    Zhang, Y.W.3    Lu, B.4    Duan, H.Q.5
  • 8
    • 77951608965 scopus 로고    scopus 로고
    • Anti-diabetic effect of standardized extract of potentilla discolor bunge and identification of its active components
    • Yang, J.; Chen, H.; Zhang, L.;Wang, Q.;Lai, M.X. Anti-Diabetic Effect of Standardized Extract of Potentilla discolor Bunge and Identification of its Active Components. Drug Develop. Res. 2010, 71, 127-132.
    • (2010) Drug Develop. Res. , vol.71 , pp. 127-132
    • Yang, J.1    Chen, H.2    Zhang, L.3    Wang, Q.4    Lai, M.X.5
  • 10
    • 85007856292 scopus 로고
    • Isolation of flavonoid-glycodides in onion and identification by chemical synthesis of the glycosides
    • Tsushida, T.; Suzuki, M. Isolation of flavonoid-glycodides in onion and identification by chemical synthesis of the glycosides. Jpn. Food Sci. Technol. 1995, 42, 100-108.
    • (1995) Jpn. Food Sci Technol. , vol.42 , pp. 100-108
    • Tsushida, T.1    Suzuki, M.2
  • 11
    • 0029998244 scopus 로고    scopus 로고
    • A two-step efficient chemoenzymatic synthesis of flavonoid glycoside malonates
    • Bruno, D.; Monica, L. A two-step efficient chemoenzymatic synthesis of flavonoid glycoside malonates. J. Nat. Prod. 1996, 5, 618-621.
    • (1996) J. Nat Prod. , vol.5 , pp. 618-621
    • Bruno, D.1    Monica, L.2
  • 12
    • 0027730791 scopus 로고
    • Chemo-enzymatic synthesis of 6-O-(3-Arylprop-2-enoyl) derivatives of the flavonol glucoside isoquercitrin
    • Bruno, D.; Andrea, B. Chemo-enzymatic synthesis of 6"-O-(3-Arylprop- 2-enoyl) derivatives of the flavonol glucoside isoquercitrin. Helv. Chim. Acta 1993, 76, 2981-2991.
    • (1993) Helv. Chim. Acta , vol.76 , pp. 2981-2991
    • Bruno, D.1    Andrea, B.2
  • 13
    • 0037179159 scopus 로고    scopus 로고
    • Regio-and stereoselective of the major metabolite of quercetin, quercetin-3-O-b-D-glucuronide
    • Mohamed, B.; Aziz, A.; Christian, R. Regio-and stereoselective of the major metabolite of quercetin, quercetin-3-O-b-D-glucuronide. Tetrahedron Lett. 2002, 43, 6263-6266.
    • (2002) Tetrahedron Lett. , vol.43 , pp. 6263-6266
    • Mohamed, B.1    Aziz, A.2    Christian, R.3
  • 14
    • 40849120177 scopus 로고    scopus 로고
    • The enzymatic synthesis of glucosylmyristate as a reaction model for general considerations on 'sugar esters' production
    • Cauglia, F.; Canepa, P. The enzymatic synthesis of glucosylmyristate as a reaction model for general considerations on 'sugar esters' production. Bioresour. Technol. 2008, 99, 4065-4072.
    • (2008) Bioresour. Technol. , vol.99 , pp. 4065-4072
    • Cauglia, F.1    Canepa, P.2
  • 15
    • 84985131464 scopus 로고
    • Structure elucidation and synthesis of flavonol acylglycosides
    • Barbara, V.; Vedanta, M.C.; Hildebert, W. Structure elucidation and synthesis of flavonol acylglycosides. Helv. Chim. Acta 1981, 64, 1964-1967.
    • (1981) Helv. Chim. Acta , vol.64 , pp. 1964-1967
    • Barbara, V.1    Vedanta, M.C.2    Hildebert, W.3
  • 16
    • 0031712627 scopus 로고    scopus 로고
    • Action of novel antidiabetic thiazolidinedione, T-174, in animal models of non-insulin-dependent diabetes mellitus (NIDDM) and in cultured muscle cells
    • Kenji, A.; Tomomi, I.; Masamichi, A.; Masanori, I.; Akira, S.; Katsuo, I. Action of novel antidiabetic thiazolidinedione, T-174, in animal models of non-insulin-dependent diabetes mellitus (NIDDM) and in cultured muscle cells. Br. J. Pharm. 1998, 125, 429-436.
    • (1998) Br. J. Pharm. , vol.125 , pp. 429-436
    • Kenji, A.1    Tomomi, I.2    Masamichi, A.3    Masanori, I.4    Akira, S.5    Katsuo, I.6
  • 17
    • 33746065836 scopus 로고    scopus 로고
    • Establishing and identifying insulin-resistance HepG2 cell line
    • Li, C.G.; Ning, G.; Chen, J.L. Establishing and identifying insulin-resistance HepG2 cell line. Chin. J. Diabetes 1999, 7, 198-200.
    • (1999) Chin. J. Diabetes , vol.7 , pp. 198-200
    • Li, C.G.1    Ning, G.2    Chen, J.L.3
  • 18
    • 33746084454 scopus 로고    scopus 로고
    • Effect of ethanolic extracts of Ananas comosus L. leaves on insulin sensitivity in rats and HepG2
    • Xie, W.D.; Wang, W.; Su, H.; Xing, D.M.; Pan, Y.; Du, L.J. Effect of ethanolic extracts of Ananas comosus L. leaves on insulin sensitivity in rats and HepG2. Comp. Biochem. Physiol. Part C 2006, 143, 429-435.
    • (2006) Comp. Biochem. Physiol. Part C , Issue.143 , pp. 429-435
    • Xie, W.D.1    Wang, W.2    Su, H.3    Xing, D.M.4    Pan, Y.5    Du, L.J.6
  • 19
    • 33645892889 scopus 로고    scopus 로고
    • Effect of citrus flavonoids on lipid metabolism and glucose-regulating enzyme mRNA levels in type-2 diabetic mice
    • Jung, U.J.; Lee, M.K.; Park, Y.B.; Kang, M.A.; Choi, M.S. Effect of citrus flavonoids on lipid metabolism and glucose-regulating enzyme mRNA levels in type-2 diabetic mice. Int. J. Biochem. Cell Biol. 2006, 38, 1134-1145.
    • (2006) Int. J. Biochem. Cell Biol. , vol.38 , pp. 1134-1145
    • Jung, U.J.1    Lee, M.K.2    Park, Y.B.3    Kang, M.A.4    Choi, M.S.5
  • 20
    • 77950917531 scopus 로고    scopus 로고
    • A comparative study of flavonoid analogues on streptozotocin-nicotinamide induced diabetic rats: Quercetin as a potential antidiabetic agent acting via 11β-Hydroxysteroid dehydrogenase type 1 inhibition
    • Mariana, T.P.; Rolffy, O.A.; Rafael, V.M.; Narender, S.; Jose, L.M.F.; Scott, P.W.; Margaret, B.; Gabriel, N.V.; Samuel, E.S.A comparative study of flavonoid analogues on streptozotocin-nicotinamide induced diabetic rats: Quercetin as a potential antidiabetic agent acting via 11β-Hydroxysteroid dehydrogenase type 1 inhibition. Eur. J. Med. Chem. 2010, 45, 2606-2612.
    • (2010) Eur. J. Med. Chem. , vol.45 , pp. 2606-2612
    • Mariana, T.P.1    Rolffy, O.A.2    Rafael, V.M.3    Narender, S.4    Jose, L.M.F.5    Scott, P.W.6    Margaret, B.7    Gabriel, N.V.8    Samuel, E.S.9
  • 22
    • 0031887718 scopus 로고    scopus 로고
    • Antidiabetic principles of natural medicines.II. Aldose reductase and alpha-glucosidase inhibitors from Brazilian natural medicine, the leaves of Myrcia multiflora DC. (Myrtaceae): Structures of myrciacitrins I and II and myrciaphenones A and B
    • Yoshikawa, M.; Shimada, H.; Nishida, N.; Li, Y.; Toguchida, I.; Yamahara, J.; Matsuda, H. Antidiabetic principles of natural medicines.II. Aldose reductase and alpha-glucosidase inhibitors from Brazilian natural medicine, the leaves of Myrcia multiflora DC. (Myrtaceae): Structures of myrciacitrins I and II and myrciaphenones A and B. Chem. Pharm. Bull. (Tokyo) 1998, 46, 113-119.
    • (1998) Chem. Pharm. Bull. (Tokyo) , vol.46 , pp. 113-119
    • Yoshikawa, M.1    Shimada, H.2    Nishida, N.3    Li, Y.4    Toguchida, I.5    Yamahara, J.6    Matsuda, H.7
  • 23
    • 0030048414 scopus 로고    scopus 로고
    • Insulinomimetic effects of myricetin on lipogenesis and glucose transport in rat adipocytes but not glucose transport translocation
    • Kian, C.O.; Hoon, E.K. Insulinomimetic effects of myricetin on lipogenesis and glucose transport in rat adipocytes but not glucose transport translocation. Biochem. Pharmacol. 1996, 51, 423-429.
    • (1996) Biochem. Pharmacol. , vol.51 , pp. 423-429
    • Kian, C.O.1    Hoon, E.K.2
  • 24
    • 0041589462 scopus 로고    scopus 로고
    • Antidiabetic effects of quercetin in streptozocin-induced diabetic rats
    • Vessal, M.; Hemmati, M. Antidiabetic effects of quercetin in streptozocin-induced diabetic rats. Comp. Biochem. Physiol. Part C 2003, 135, 357-364.
    • (2003) Comp. Biochem. Physiol. Part C , vol.135 , pp. 357-364
    • Vessal, M.1    Hemmati, M.2
  • 25
    • 77954870511 scopus 로고    scopus 로고
    • The potential mechanism of tiliroside-dependent inhibition of t-butylhydroperoxide-induced oxidative stress in endometrial carcinoma cells
    • Tomczyk, M.; Tumanov, A.; Zaniewska, A.; Surazynski, A. The potential mechanism of tiliroside-dependent inhibition of t-butylhydroperoxide-induced oxidative stress in endometrial carcinoma cells. Planta Med. 2010, 76, 963-968.
    • (2010) Planta Med. , vol.76 , pp. 963-968
    • Tomczyk, M.1    Tumanov, A.2    Zaniewska, A.3    Surazynski, A.4
  • 26
    • 74249119381 scopus 로고    scopus 로고
    • Tyrosinase inhibitory effect and inhibitory mechanism of tiliroside from raspberry
    • Lu, Y.H.; Chen, J.; Wei, D.Z.; Wang, Z.T.; Tao, X.Y. Tyrosinase inhibitory effect and inhibitory mechanism of tiliroside from raspberry. J. Enzyme Inhib. Med. Chem. 2009, 24, 1154-1160.
    • (2009) J. Enzyme Inhib. Med. Chem. , vol.24 , pp. 1154-1160
    • Lu, Y.H.1    Chen, J.2    Wei, D.Z.3    Wang, Z.T.4    Tao, X.Y.5
  • 27
    • 56749157730 scopus 로고    scopus 로고
    • Studies on the phenylethanoid glycosides with anti-complement activity from Paulownia tomentosa var. tomentosa wood
    • Si, C.L.; Deng, X.J.; Liu, Z.; Kim, J.K.; Bae, Y.S. Studies on the phenylethanoid glycosides with anti-complement activity from Paulownia tomentosa var. tomentosa wood. J. Asian Nat. Prod. Res. 2008, 10, 1003-1008.
    • (2008) J. Asian Nat. Prod. Res. , vol.10 , pp. 1003-1008
    • Si, C.L.1    Deng, X.J.2    Liu, Z.3    Kim, J.K.4    Bae, Y.S.5
  • 28
    • 34848848083 scopus 로고    scopus 로고
    • Acetylcholinesterase inhibition by flavonoids from Agrimonia pilosa
    • Jung, M.; Park, M. Acetylcholinesterase inhibition by flavonoids from Agrimonia pilosa. Molecules 2007, 12, 2130-2139.
    • (2007) Molecules , vol.12 , pp. 2130-2139
    • Jung, M.1    Park, M.2
  • 29
    • 34247895642 scopus 로고    scopus 로고
    • Potent anti-obese principle from Rosa canina:Structrual requirements and mode of action of trans-tiliroside
    • Kiyofumi, N. Hisashi, M.; Mizuho, K.; Toshio, M.; Norihisa, N.; Masayuki, Y. Potent anti-obese principle from Rosa canina:Structrual requirements and mode of action of trans-tiliroside. Bioorg. Med. Chem. Lett. 2007, 17, 3059-3064.
    • (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 3059-3064
    • Kiyofumi, N.1    Hisashi, M.2    Mizuho, K.3    Toshio, M.4    Norihisa, N.5    Masayuki, Y.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.