Gene polymorphisms involved in triptans pharmacokinetics and pharmacodynamics in migraine therapy

Expert Opinion on Drug Metabolism and Toxicology

Volumn 7, Issue 1, 2011, Pages 39-47

  Gentile, Giovanna ^a   Borro, Marina ^b   Simmaco, Maurizio ^a,b   Missori, Serena ^a   Lala, Noemi ^a   Martelletti, Paolo ^a  

^a SAPIENZA UNIVERSITY OF ROME   (Italy)

^b SAPIENZA UNIVERSITY OF ROME   (Italy)

Author keywords

Migraine; Pharmacogenomics; Polymorphisms; Triptans

Indexed keywords

ALMOTRIPTAN; AMINE OXIDASE (FLAVIN CONTAINING) ISOENZYME A; CYTOCHROME P450; DOPAMINE RECEPTOR; ELETRIPTAN; FROVATRIPTAN; GUANINE NUCLEOTIDE BINDING PROTEIN BETA SUBUNIT; NARATRIPTAN; RIZATRIPTAN; SEROTONIN RECEPTOR; SEROTONIN TRANSPORTER; SUMATRIPTAN; TRIPTAN DERIVATIVE; ZOLMITRIPTAN;

ARTICLE; DNA POLYMORPHISM; DRUG BIOAVAILABILITY; DRUG MECHANISM; DRUG METABOLISM; GENETIC ASSOCIATION; HUMAN; INDEL MUTATION; MIGRAINE; NEUROTRANSMITTER RELEASE; PHARMACODYNAMICS; PHARMACOGENOMICS; SINGLE NUCLEOTIDE POLYMORPHISM; TREATMENT RESPONSE; VARIABLE NUMBER OF TANDEM REPEAT;

CLINICAL TRIALS AS TOPIC; GENETIC ASSOCIATION STUDIES; GENOME, HUMAN; HUMANS; MIGRAINE DISORDERS; MONOAMINE OXIDASE; PAIN; PHARMACOGENETICS; POLYMORPHISM, SINGLE NUCLEOTIDE; SEROTONIN PLASMA MEMBRANE TRANSPORT PROTEINS; TRYPTAMINES;

EID: 78650500631     PISSN: 17425255     EISSN: None     Source Type: Journal    
DOI: 10.1517/17425255.2011.538680     Document Type: Article

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