Design and synthesis of phthalimide-based fluorescent liver X receptor antagonists

Chemical and Pharmaceutical Bulletin

Volumn 58, Issue 11, 2010, Pages 1524-1528

  Kishida, Kenji ^a   Aoyama, Atsushi ^b   Hashimoto, Yuichi ^b   Miyachi, Hiroyuki ^a  

^a OKAYAMA UNIVERSITY   (Japan)

^b UNIVERSITY OF TOKYO   (Japan)

Author keywords

Fluorescent ligand; Liver X receptor; Liver X receptor antagonist

Indexed keywords

AMINE; LIGAND; LIVER X RECEPTOR; LIVER X RECEPTOR ALPHA; LIVER X RECEPTOR ANTAGONIST; LIVER X RECEPTOR BETA; PHTHALIMIDE DERIVATIVE; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG; FLUORESCENT DYE; ORPHAN NUCLEAR RECEPTOR;

ARTICLE; DRUG BINDING SITE; DRUG DESIGN; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; FLUORESCENCE; FLUORESCENCE SPECTROSCOPY; HUMAN; HUMAN CELL; HYDROPHOBICITY; STRUCTURE ACTIVITY RELATION; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; SYNTHESIS;

CELL LINE; FLUORESCENT DYES; HUMANS; LIGANDS; MOLECULAR STRUCTURE; ORPHAN NUCLEAR RECEPTORS; PHTHALIMIDES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 78049459888     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.58.1525     Document Type: Article

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