In vitro and in vivo characterization of novel 18F-labeled bombesin analogues for targeting GRPR-positive tumors

Bioconjugate Chemistry

Volumn 21, Issue 10, 2010, Pages 1864-1871

  Mu, Linjing ^a   Honer, Michael ^a   Becaud, Jessica ^a   Martic, Miljen ^a   Schubiger, Pius A ^a   Ametamey, Simon M ^a   Stellfeld, Timo ^b   Graham, Keith ^b   Borkowski, Sandra ^b   Lehmann, Lutz ^b   Dinkelborg, Ludger ^b   Srinivasan, Ananth ^b  

^a ETH ZURICH   (Switzerland)

^b BAYER PHARMA AG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING ENERGY; DIAGNOSIS; PEPTIDES;

BOMBESIN ANALOGUES; HUMAN TUMORS; IN-VITRO; IN-VIVO; LINKER SEQUENCE; PEPTIDE RECEPTOR; PEPTIDE SEQUENCES; PET IMAGING; SYNTHESISED; VITRO AND IN VIVO;

TUMORS;

BOMBESIN DERIVATIVE; GASTRIN RELEASING PEPTIDE RECEPTOR; RADIOPHARMACEUTICAL AGENT;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; DRUG UPTAKE; IN VITRO STUDY; IN VIVO STUDY; ISOTOPE LABELING; MOUSE; NONHUMAN; PANCREAS TUMOR; POSITRON EMISSION TOMOGRAPHY; TUMOR;

MUS MUSCULUS;

EID: 77958193859     PISSN: 10431802     EISSN: 15204812     Source Type: Journal    
DOI: 10.1021/bc100222u     Document Type: Article

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