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Volumn 45, Issue 11, 2010, Pages 5520-5526

Synthesis and biological activities of pyrazolo[3,4-g]quinoxaline derivatives

(6) Gavara, Laurent a,b Saugues, Emmanuelle a,b Alves, Georges a,b Debiton, Eric a Anizon, Fabrice a,b Moreau, Pascale a,b

a UNIVERSITÉ CLERMONT AUVERGNE (France)

b CNRS (France)

Author keywords

In vitro antiproliferative activities; Kinase inhibition; Pyrazolo 3,4 g quinoxaline

Indexed keywords

1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINOXALINE; 1H INDAZOLE 5,6 DIAMINE; 5,6 DINITRO 1H INDAZOLE; 6 METHYL 1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINOXALINE; 6 METHYL 6,9 DIMETHYLMETHANO 6,7,8,9 TETRAHYDRO 1H PYRAZOLO[3,4 B]PHENAZINE; 6,7 DIETHYL 1H PYRAZOLO[3,4 G]QUINOXALINE; 6,7 DIMETHYL1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINOXALINE; 6,7,8,9 TETRAHYDRO 1H PYRAZOLO[3,4 B]PHENAZINE; 7 PHENYL 1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINOXALINE; 7,8 DIMETHYL 1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINOXALINE; 8 METHYL 1,6,7,8 TETRAHYDROCYCLOPENTA[B]PYRAZOLO[3,4 G]QUINAXOLINE; 9 METHYL 6,9 DIMETHYLMETHANO 6,7,8,9 TETRAHYDRO 1H PYRAZOLO[3,4 B]PHENAZINE; PROTEIN KINASE PIM 1; QUINOXALINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CELL PROLIFERATION; DRUG POTENCY; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; FIBROBLAST; HUMAN; HUMAN CELL; IN VITRO STUDY; OUTCOME ASSESSMENT; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; PYRAZOLES; QUINOXALINES; SPECTROMETRY, MASS, ELECTROSPRAY IONIZATION; SPECTROPHOTOMETRY, INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77957833608 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2010.08.067 Document Type: Article

Times cited : (44)

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