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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 19, 2010, Pages 5815-5817

Reverse-benzamidine antimalarial agents: Design, synthesis, and biological evaluation

(9) Berger, Olivier a Wein, Sharon b Duckert, Jean Frederic a Maynadier, Marjorie b Fangour, Siham El a Escale, Roger a Durand, Thierry a Vial, Henri b Vo Hoang, Yen a

a UNIVERSITÉ DE MONTPELLIER (France)

b UNIVERSITÉ DE MONTPELLIER (France)

Author keywords

Antimalarial agents; Bis N alkylamidines; Chemical design; Reverse benzamidines; Total clearance of parasitemia

Indexed keywords

ANTIMALARIAL AGENT; BENZAMIDINE DERIVATIVE;

ALKALINITY; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; FEMALE; IN VITRO STUDY; LIPOPHILICITY; MOUSE; NONHUMAN; PARASITEMIA;

ANTIMALARIALS; BENZAMIDINES; DRUG DESIGN; PLASMODIUM FALCIPARUM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 77957576119 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.07.124 Document Type: Article

Times cited : (8)

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