Synthesis and antimalarial activity of new 1,12-bis(N,N′-acetamidinyl)dodecane derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 3, 2007, Pages 593-596

  Ouattara, Mahama ^a,b,c   Wein, Sharon ^a   Calas, Michèle ^d   Hoang, Yen Vo ^b   Vial, Henri ^a   Escale, Roger ^b  

^a UNIVERSITÉ DE MONTPELLIER   (France)

^b UNIV MONTPELLIER   (France)

^c UFR Sciences Économiques et de Gestion   (France)

^d CNRS   (France)

Author keywords

Antimalarial agents; Bis alkylamidine; Bis alkylamidoxime; O substituted bis alkylamidoxime; Prodrugs

Indexed keywords

ACETAMIDINE DERIVATIVE; CHLOROQUINE;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIMALARIAL ACTIVITY; ARTICLE; DRUG POTENCY; DRUG SYNTHESIS; EVALUATION; MOUSE; NONHUMAN; SUBSTITUTION REACTION;

EID: 33846343962     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.11.013     Document Type: Article

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