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European Journal of Medicinal Chemistry

Volumn 45, Issue 10, 2010, Pages 4418-4426

Synthesis and antimycobacterial activity of new quinoxaline-2-carboxamide 1,4-di-N-oxide derivatives

(6) Moreno, Elsa a Ancizu, Saioa a Pérez Silanes, Silvia a Torres, Enrique a Aldana, Ignacio a Monge, Antonio a

a UNIVERSITY OF NAVARRA (Spain)

Author keywords

Anti tuberculosis agents; Mycobacterium tuberculosis; N oxides; Quinoxaline

Indexed keywords

3 METHYL 7 TRIFLUOROMETHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 CHLOROBENZYLAMIDE 1,4 DI N OXIDE; 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID (2 PHENYLETHYL)AMIDE 1,4 DI N OXIDE; 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 3,7 DIMETHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 6 METHOXY 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 6,7 DICHLORO 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 6,7 DICHLORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 6,7 DICHLORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 7 CHLORO 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 CHLOROBENZYLAMIDE 1,4 DI N OXIDE; 7 CHLORO 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 7 CHLORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID (2 PHENYLETHYL)AMIDE 1,4 DI N OXIDE; 7 CHLORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 7 CHLORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 7 FLUORO 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 7 FLUORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 7 FLUORO 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 7 METHOXY 3 METHYLQUINOXALINE 2 CARBOXYLIC ACID 4 TRIFLUOROMETHYLBENZYLAMIDE 1,4 DI N OXIDE; 7 METHOXY 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 7 METHYL 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 7 METHYL 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; 7 TRIFLUOROMETHYL 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID BENZYLAMIDE 1,4 DI N OXIDE; 7 TRIFLUOROMETHYL 3 PHENYLQUINOXALINE 2 CARBOXYLIC ACID PHENYLAMIDE 1,4 DI N OXIDE; ANTIINFECTIVE AGENT; QUINOXALINE 2 CARBOXAMIDE 1,4 DI N OXIDE DERIVATIVE; QUINOXALINE DERIVATIVE; RIFAMPICIN; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANIMAL CELL; ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; CELL LINE; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; IN VITRO STUDY; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STRUCTURE ACTIVITY RELATION; TUBERCULOSIS;

AMIDES; ANIMALS; ANTITUBERCULAR AGENTS; CELL SURVIVAL; CERCOPITHECUS AETHIOPS; HUMANS; MYCOBACTERIUM TUBERCULOSIS; OXIDES; QUINOXALINES; TUBERCULOSIS; VERO CELLS;

EID: 77956184672 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2010.06.036 Document Type: Article

Times cited : (62)

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