Synthesis and evaluation of esmolol prodrugs for transdermal delivery

Drug Delivery

Volumn 17, Issue 7, 2010, Pages 532-540

  Bijaya, Ghosh ^a   Kaushal, Dave ^b   Sonal, Dubey ^a   Pallavi, K ^a  

^a A Constituent Unit of KLE Academy of Higher Education Research   (India)

^b SOUTH DAKOTA STATE UNIVERSITY   (United States)

Author keywords

Anti hypertensive; Esterase; In vitro; Passive diffusion; Permeability coefficient

Indexed keywords

ESMOLOL; ESMOLOL ACETATE; ESMOLOL BUTYRATE; ESMOLOL PROPIONATE; ESMOLOL VALERATE; PRODRUG; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIHYPERTENSIVE ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; DRUG EFFICACY; DRUG PENETRATION; DRUG STRUCTURE; DRUG SYNTHESIS; ESTERIFICATION; EVALUATION; HYPERTENSION; LIPOPHILICITY; MALE; NONHUMAN; PARAMETER; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; RAT; REACTION ANALYSIS; SKIN PERMEABILITY; SPRAGUE DAWLEY RAT; SWINE;

ADMINISTRATION, CUTANEOUS; ANIMALS; ANTIHYPERTENSIVE AGENTS; BLOOD PRESSURE; DRUG STABILITY; ESTERS; MALE; PERMEABILITY; PRODRUGS; PROPANOLAMINES; RATS; RATS, SPRAGUE-DAWLEY; SKIN ABSORPTION; SOLUBILITY; SWINE;

EID: 77956151821     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.3109/10717544.2010.490248     Document Type: Article

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