Pentobarbital inhibition of human recombinant α 1A P/Q-type voltage-gated calcium channels involves slow, open channel block

British Journal of Pharmacology

Volumn 161, Issue 2, 2010, Pages 365-383

  Schober, A ^a   Sokolova, E ^a   Gingrich, K J ^a  

^a NEW YORK UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

Ca V2.1; electrophysiology; P Q Ca +2 channels; pentobarbital; pharmacology; recombinant proteins

Indexed keywords

CALCIUM; CALCIUM CHANNEL P TYPE; CALCIUM CHANNEL Q TYPE; PENTOBARBITAL;

ARTICLE; CALCIUM CELL LEVEL; CALCIUM CURRENT; CELL STRAIN HEK293; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYTOSOL; DRUG EFFECT; DRUG MECHANISM; FREQUENCY MODULATION; HUMAN; HUMAN CELL; IC 50; NERVE CELL PLASTICITY; NEUROTRANSMITTER RELEASE; PATCH CLAMP; PRIORITY JOURNAL; STEADY STATE; WHOLE CELL;

CALCIUM CHANNEL BLOCKERS; CALCIUM CHANNELS; CELL CULTURE TECHNIQUES; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGICAL PHENOMENA; HUMANS; ION CHANNEL GATING; PENTOBARBITAL; RECOMBINANT PROTEINS; TIME FACTORS; TRANSFECTION;

EID: 77956026094     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.2010.00886.x     Document Type: Article

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