Two-headed PROTAC: An effective new tool for targeted protein degradation

ChemBioChem

Volumn 11, Issue 11, 2010, Pages 1531-1534

  Cyrus, Kedra ^a   Wehenkel, Marie ^a   Choi, Eun Young ^a   Swanson, Hollie ^a   Kim, Kyung Bo ^a  

^a UNIVERSITY OF KENTUCKY   (United States)

Author keywords

Estrogen receptor; Ligases; PROTAC; Proteomics; Ubiquitin proteasome pathway

Indexed keywords

PROTEASOME; UBIQUITIN; UBIQUITIN PROTEIN LIGASE E3; ESTROGEN RECEPTOR; LIGASE; PEPTIDE; PROTEIN; SNAKE VENOM PROTEIN C ACTIVATOR;

AMINO ACID SUBSTITUTION; ARTICLE; BINDING AFFINITY; CHIMERA; IMMUNOFLUORESCENCE; MASS SPECTROMETRY; PRIORITY JOURNAL; PROTEIN DEGRADATION; PROTON NUCLEAR MAGNETIC RESONANCE; TECHNOLOGY; UBIQUITINATION; DRUG DELIVERY SYSTEM; DRUG EFFECTS; FEMALE; HUMAN; METABOLISM; PROTEIN STABILITY;

DRUG DELIVERY SYSTEMS; FEMALE; HUMANS; LIGASES; PEPTIDES; PROTEIN STABILITY; PROTEINS; RECEPTORS, ESTROGEN;

EID: 77955162918     PISSN: 14394227     EISSN: 14397633     Source Type: Journal    
DOI: 10.1002/cbic.201000222     Document Type: Article

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