Discovery of carboranes as inducers of 20S proteasome activity

ChemMedChem

Volumn 5, Issue 8, 2010, Pages 1236-1241

  Ban, Hyun Seung ^a   Minegishi, Hidemitsu ^a   Shimizu, Kazuki ^a   Maruyama, Minako ^a   Yasui, Yuka ^a   Nakamura, Hiroyuki ^a  

^a GAKUSHUIN UNIVERSITY   (Japan)

Author keywords

20S proteasome; Activators; Caspase like activity; Drug discovery; Trypsin like activity

Indexed keywords

2 (4 CARBORANYLPHENOXY)N PHENYLACETAMIDE; CARBORANE DERIVATIVE; CASPASE; CHYMOTRYPSIN; PROTEASOME; PROTEASOME 20S; TRYPSIN; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; PRIORITY JOURNAL; SIGNAL TRANSDUCTION;

ACETANILIDES; ACETIC ACIDS; BENZOPHENONES; BORON; BORON COMPOUNDS; CARBON; DRUG EVALUATION, PRECLINICAL; HELA CELLS; HUMANS; PROTEASOME ENDOPEPTIDASE COMPLEX;

EID: 77955120232     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.201000112     Document Type: Article

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